1233855-46-3 | BIA 10-2474

Packsize	Purity	Availability	Price	Discounted Price
1mg	99%	in stock	$12.00	$9.00
5mg	99%	in stock	$29.00	$20.00
10mg	99%	in stock	$42.00	$30.00
25mg	99%	in stock	$70.00	$49.00
50mg	99%	in stock	$112.00	$79.00

Description

• Catalog Number: AA26326
• Chemical Name: BIA 10-2474
• CAS Number: 1233855-46-3
• Molecular Formula: C16H20N4O2
• Molecular Weight: 300.3556
• MDL Number: MFCD30532661
• SMILES: [O-][n+]1cccc(c1)c1ncn(c1)C(=O)N(C1CCCCC1)C

Computed Properties

• Complexity: 386
• Covalently-Bonded Unit Count: 1
• Heavy Atom Count: 22
• Hydrogen Bond Acceptor Count: 3
• Rotatable Bond Count: 2
• XLogP3: 1.3

Literature

• Discovery of a Potent, Long-Acting, and CNS-Active Inhibitor (BIA 10-2474) of Fatty Acid Amide Hydrolase.

  ChemMedChem 20181022

• Activity-based protein profiling reveals off-target proteins of the FAAH inhibitor BIA 10-2474.

  Science (New York, N.Y.) 20170609

• Fatty acid amide hydrolase inhibitors: a patent review (2009-2014).

  Expert opinion on therapeutic patents 20150101

• The endocannabinoid system as a potential therapeutic target for pain modulation.

  Balkan medical journal 20140601

• Inhibition of fatty acid amide hydrolase (FAAH) as a novel therapeutic strategy in the treatment of pain and inflammatory diseases in the gastrointestinal tract.

  European journal of pharmaceutical sciences : official journal of the European Federation for Pharmaceutical Sciences 20140214