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Adenosine A(2A) receptor promotes collagen type III synthesis via β-catenin activation in human dermal fibroblasts.
British journal of pharmacology 20161201
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Enhanced A2A adenosine receptor-mediated increase in coronary flow in type I diabetic mice.
Journal of molecular and cellular cardiology 20160101
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Selective inhibition of KCa3.1 channels mediates adenosine regulation of the motility of human T cells.
Journal of immunology (Baltimore, Md. : 1950) 20131215
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Adenosine A2A receptor and TNF-α regulate the circadian machinery of the human monocytic THP-1 cells.
Inflammation 20130201
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Adenosine A2A receptor modulates vascular response in soluble epoxide hydrolase-null mice through CYP-epoxygenases and PPARγ.
American journal of physiology. Regulatory, integrative and comparative physiology 20130101
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Constitutive activity of the A2A adenosine receptor and compartmentalised cyclic AMP signalling fine-tune noradrenaline release.
Purinergic signalling 20121201
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Stimulation of adenosine receptors in the nucleus accumbens reverses the expression of cocaine sensitization and cross-sensitization to dopamine D2 receptors in rats.
Neuropharmacology 20121101
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Adenosine A(2a) receptor stimulation prevents hepatocyte lipotoxicity and non-alcoholic steatohepatitis (NASH) in rats.
Clinical science (London, England : 1979) 20120901
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A2A adenosine receptor agonists reduce both high-palatability and low-palatability food intake in female rats.
Behavioural pharmacology 20120901
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Trk and cAMP-dependent survival activity of adenosine A(2A) agonist CGS21680 on rat motoneurons in culture.
Neuroscience letters 20120726
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Adenosine A2A receptor activation and hyaluronan fragment inhibition reduce inflammation in mouse articular chondrocytes stimulated with interleukin-1β.
The FEBS journal 20120601
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Adenosine A2A receptor activation prevents wear particle-induced osteolysis.
Science translational medicine 20120523
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Activation of the adenosine A2A receptor attenuates experimental autoimmune myasthenia gravis severity.
European journal of immunology 20120501
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The effect of A(2A) adenosine receptor activation on C-C chemokine receptor 7 expression in human THP1 macrophages during inflammation.
Inflammation 20120401
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Adenosine A2A receptors in the nucleus accumbens bi-directionally alter cocaine seeking in rats.
Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology 20120401
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Differential effects of the adenosine Aâ‚‚A agonist CGS-21680 and haloperidol on food-reinforced fixed ratio responding in the rat.
Psychopharmacology 20120301
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Distinctive immunoregulatory effects of adenosine on T cells of older humans.
FASEB journal : official publication of the Federation of American Societies for Experimental Biology 20120301
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Cholesterol 27-hydroxylase but not apolipoprotein apoE contributes to A2A adenosine receptor stimulated reverse cholesterol transport.
Inflammation 20120201
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Effects of Aâ‚‚A adenosine receptor blockade or stimulation on alcohol intake in alcohol-preferring rats.
Psychopharmacology 20120201
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Endotoxin-induced effects on nucleotide catabolism in mouse kidney.
European journal of pharmacology 20120115
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Evaluation of molecular modeling of agonist binding in light of the crystallographic structure of an agonist-bound Aâ‚‚A adenosine receptor.
Journal of medicinal chemistry 20120112
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Deletion of the BDNF truncated receptor TrkB.T1 delays disease onset in a mouse model of amyotrophic lateral sclerosis.
PloS one 20120101
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Activation of adenosine A2A receptor up-regulates BDNF expression in rat primary cortical neurons.
Neurochemical research 20111201
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CGS 21680, an agonist of the adenosine (A2A) receptor, decreases acute lung inflammation.
European journal of pharmacology 20111001
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CGS 21680, an agonist of the adenosine (A2A) receptor, reduces progression of murine type II collagen-induced arthritis.
The Journal of rheumatology 20111001
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Adenosine A(2A) receptor activation prevents progressive kidney fibrosis in a model of immune-associated chronic inflammation.
Kidney international 20110801
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Adenosine A(2A) agonists as therapy for glomerulonephritis.
Kidney international 20110801
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Synaptically driven state transitions in distal dendrites of striatal spiny neurons.
Nature neuroscience 20110701
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Adenosine 2A receptor is protective against renal injury in MRL/lpr mice.
Lupus 20110601
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Regulation of epithelial sodium channel α-subunit expression by adenosine receptor A₂a in alveolar epithelial cells.
Chinese medical journal 20110501
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Stimulation of A(â‚‚a) adenosine receptor abolishes the inhibitory effect of arachidonic acid on the basolateral 50-pS K channel in the thick ascending limb.
American journal of physiology. Renal physiology 20110401
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Pharmacological postconditioning protects against hepatic ischemia/reperfusion injury.
Liver transplantation : official publication of the American Association for the Study of Liver Diseases and the International Liver Transplantation Society 20110401
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On the existence of a possible A2A-D2-β-Arrestin2 complex: A2A agonist modulation of D2 agonist-induced β-arrestin2 recruitment.
Journal of molecular biology 20110311
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Adenosine A2A receptor activation attenuates tubuloglomerular feedback responses by stimulation of endothelial nitric oxide synthase.
American journal of physiology. Renal physiology 20110201
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Adenosine A(2A) receptor agonist (CGS-21680) prevents endotoxin-induced effects on nucleotidase activities in mouse lymphocytes.
European journal of pharmacology 20110125
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Novel 8-(furan-2-yl)-3-benzyl thiazolo [5,4-e][1,2,4] triazolo [1,5-c] pyrimidine-2(3H)-thione as selective adenosine A(2A) receptor antagonist.
Neuroscience letters 20110113
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Excitatory effect of the A2A adenosine receptor agonist CGS-21680 on spontaneous and K+-evoked acetylcholine release at the mouse neuromuscular junction.
Neuroscience 20110113
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Receptor desensitization and blockade of the suppressive effects of prostaglandin E(2) and adenosine on the cytotoxic activity of human melanoma-infiltrating T lymphocytes.
Cancer immunology, immunotherapy : CII 20110101
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Selective adenosine A2A receptor agonists and antagonists protect against spinal cord injury through peripheral and central effects.
Journal of neuroinflammation 20110101
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A2A and A3 adenosine receptor expression in rheumatoid arthritis: upregulation, inverse correlation with disease activity score and suppression of inflammatory cytokine and metalloproteinase release.
Arthritis research & therapy 20110101
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Contribution of adenosine A(2A) and A(2B) receptors to ischemic coronary dilation: role of K(V) and K(ATP) channels.
Microcirculation (New York, N.Y. : 1994) 20101101
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Peripheral adenosine A2A receptors are involved in carrageenan-induced mechanical hyperalgesia in mice.
Neuroscience 20101027
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Adenosine can mediate its actions through generation of reactive oxygen species.
Journal of cerebral blood flow and metabolism : official journal of the International Society of Cerebral Blood Flow and Metabolism 20101001
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Both A2a and A2b adenosine receptors at reperfusion are necessary to reduce infarct size in mouse hearts.
American journal of physiology. Heart and circulatory physiology 20101001
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Adenosine A1 receptor agonists reduce hyperalgesia after spinal cord injury in rats.
Spinal cord 20100901
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Contraction-induced secretion of VEGF from skeletal muscle cells is mediated by adenosine.
American journal of physiology. Heart and circulatory physiology 20100901
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Ecto-5'-nucleotidase (CD73) attenuates allograft airway rejection through adenosine 2A receptor stimulation.
Journal of immunology (Baltimore, Md. : 1950) 20100715
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Adenosine A(2)A receptor but not HIF-1 mediates Tyrosine hydroxylase induction in hypoxic PC12 cells.
Journal of neuroscience research 20100701
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An adenosine A(2A) agonist injected in the nucleus of the solitary tract prolongs the laryngeal chemoreflex by a GABAergic mechanism in decerebrate piglets.
Experimental physiology 20100701
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Modulation by salt intake of the vascular response mediated through adenosine A(2A) receptor: role of CYP epoxygenase and soluble epoxide hydrolase.
American journal of physiology. Regulatory, integrative and comparative physiology 20100701
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Indirect basal ganglia pathway mediation of repetitive behavior: attenuation by adenosine receptor agonists.
Behavioural brain research 20100626
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Activation of adenosine A2A receptors induces TrkB translocation and increases BDNF-mediated phospho-TrkB localization in lipid rafts: implications for neuromodulation.
The Journal of neuroscience : the official journal of the Society for Neuroscience 20100623
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Activation of adenosine A2A receptor attenuates inflammatory response in a rat model of small-for-size liver transplantation.
Transplantation proceedings 20100601
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Adenosine receptor agonists affect taurine release from mouse brain stem slices in ischemia.
Amino acids 20100501
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Adenosine A2A receptor-selective stimulation reduces signaling pathways involved in the development of intestine ischemia and reperfusion injury.
Shock (Augusta, Ga.) 20100501
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Changes induced by formalin pain in central alpha1-adrenoceptor density are modulated by adenosine receptor agonists.
Journal of neural transmission (Vienna, Austria : 1996) 20100501
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Influence of CGS 21680, a selective adenosine A(2A) receptor agonist, on NMDA receptor function and expression in the brain of Huntington's disease mice.
Brain research 20100406
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Role of adenosine A2 receptors in regulation of cerebral blood flow during induced hypotension.
Journal of cerebral blood flow and metabolism : official journal of the International Society of Cerebral Blood Flow and Metabolism 20100401
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A2A adenosine receptor stimulation decreases foam cell formation by enhancing ABCA1-dependent cholesterol efflux.
Journal of leukocyte biology 20100401
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Adenosine up-regulates vascular endothelial growth factor in human macrophages.
Biochemical and biophysical research communications 20100212
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Post exposure administration of A(1) adenosine receptor agonists attenuates noise-induced hearing loss.
Hearing research 20100201
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The role of nucleus accumbens adenosine-opioid interaction in mediating palatable food intake.
Brain research 20100108
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Selective adenosine A(2a) receptor agonists reduce the apoptosis in an experimental model of spinal cord trauma.
Journal of biological regulators and homeostatic agents 20100101
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Effects of adenosine A(2A) and A(2B) receptor activation on signaling pathways and cytokine production in human uroepithelial cells.
Pharmacology 20100101
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Static magnetic field exposure reproduces cellular effects of the Parkinson's disease drug candidate ZM241385.
PloS one 20100101
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Useful pharmacological parameters for G-protein-coupled receptor homodimers obtained from competition experiments. Agonist-antagonist binding modulation.
Biochemical pharmacology 20091215
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The impact of adenosine and an A2A adenosine receptor agonist on the ACh-induced increase in intracellular calcium of the glomus cells of the cat carotid body.
Brain research 20091208
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The selective adenosine A2A receptor agonist CGS 21680 reduces JNK MAPK activation in oligodendrocytes in injured spinal cord.
Shock (Augusta, Ga.) 20091201
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Theophylline inhibits the differentiation of human monocyte into dendritic cell potentially via adenosine receptor antagonism.
Clinical and experimental allergy : journal of the British Society for Allergy and Clinical Immunology 20091201
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Absence of adenosine-mediated aortic relaxation in A(2A) adenosine receptor knockout mice.
American journal of physiology. Heart and circulatory physiology 20091101
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Effects of adenosine A2A receptor stimulation on cocaine-seeking behavior in rats.
Psychopharmacology 20091001
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Differential regulation of HIF-1alpha isoforms in murine macrophages by TLR4 and adenosine A(2A) receptor agonists.
Journal of leukocyte biology 20090901
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Altered distribution and function of A2A adenosine receptors in the brain of WAG/Rij rats with genetic absence epilepsy, before and after appearance of the disease.
The European journal of neuroscience 20090901
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Platelet function analyzer (PFA-100) offers higher sensitivity and specificity than thromboelastography (TEG) in detection of platelet dysfunction.
Acta anaesthesiologica Taiwanica : official journal of the Taiwan Society of Anesthesiologists 20090901
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The A2A adenosine receptor rescues the urea cycle deficiency of Huntington's disease by enhancing the activity of the ubiquitin-proteasome system.
Human molecular genetics 20090815
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Blocking adenosine A2A receptor reduces peritoneal fibrosis in two independent experimental models.
Nephrology, dialysis, transplantation : official publication of the European Dialysis and Transplant Association - European Renal Association 20090801
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SAR of a series of inhaled A(2A) agonists and comparison of inhaled pharmacokinetics in a preclinical model with clinical pharmacokinetic data.
Bioorganic & medicinal chemistry letters 20090801
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A2A adenosine receptor deficiency leads to impaired tracheal relaxation via NADPH oxidase pathway in allergic mice.
The Journal of pharmacology and experimental therapeutics 20090701
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Spinal NMDA receptor activation is necessary for de novo, but not the maintenance of, A2a receptor-mediated phrenic motor facilitation.
Journal of applied physiology (Bethesda, Md. : 1985) 20090701
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The adenosine A2A receptor antagonist ZM241385 enhances neuronal survival after oxygen-glucose deprivation in rat CA1 hippocampal slices.
British journal of pharmacology 20090701
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Protective effects of adenosine A2A receptor agonist in ventilator-induced lung injury in rats.
Critical care medicine 20090701
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Adenosine A(2A) receptor mediates microglial process retraction.
Nature neuroscience 20090701
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The role of adenosine in hypercarbic hyperemia: in vivo and in vitro studies in adenosine 2(A) receptor knockout and wild-type mice.
Journal of neurosurgery 20090501
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Cardioprotection induced by adenosine A1 receptor agonists in a cardiac cell ischemia model involves cooperative activation of adenosine A2A and A2B receptors by endogenous adenosine.
Journal of cardiovascular pharmacology 20090501
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Functional interaction between purinergic system and opioid withdrawal: in vitro evidence.
Current drug safety 20090501
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Regulation of hind-limb tone by adenosine A2A receptor in rats.
Neuroscience 20090410
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Activation of NTS A2a adenosine receptors differentially resets baroreflex control of renal vs. adrenal sympathetic nerve activity.
American journal of physiology. Heart and circulatory physiology 20090401
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Modification of the cardiovascular response of posterior hypothalamic adenosine A(2A) receptor stimulation by adenylate cyclase and KATP channel blockade in anesthetized rats.
Autonomic neuroscience : basic & clinical 20090312
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High-salt diet enhances mouse aortic relaxation through adenosine A2A receptor via CYP epoxygenases.
American journal of physiology. Regulatory, integrative and comparative physiology 20090301
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GDNF control of the glutamatergic cortico-striatal pathway requires tonic activation of adenosine A receptors.
Journal of neurochemistry 20090301
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Modulation of gamma oscillations by endogenous adenosine through A1 and A2A receptors in the mouse hippocampus.
Neuropharmacology 20090201
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Diminished iron concentrations increase adenosine A(2A) receptor levels in mouse striatum and cultured human neuroblastoma cells.
Experimental neurology 20090201
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Adenosine A(1) and A(2A) receptors in mouse prefrontal cortex modulate acetylcholine release and behavioral arousal.
The Journal of neuroscience : the official journal of the Society for Neuroscience 20090121
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Impact of anti-inflammatory agents on the gene expression profile of stimulated human neutrophils: unraveling endogenous resolution pathways.
PloS one 20090101
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An antagonistic interaction between A2B adenosine and D2 dopamine receptors modulates the function of rat carotid body chemoreceptor cells.
Journal of neurochemistry 20081201
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Adenosine A2A and beta-adrenergic calcium transient and contractile responses in rat ventricular myocytes.
American journal of physiology. Heart and circulatory physiology 20081201
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FGF acts as a co-transmitter through adenosine A(2A) receptor to regulate synaptic plasticity.
Nature neuroscience 20081201
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Adenosine modulates excitatory synaptic transmission and suppresses neuronal death induced by ischaemia in rat spinal motoneurones.
Pflugers Archiv : European journal of physiology 20081101
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Electron probe X-ray microanalysis of intact pathway for human aqueous humor outflow.
American journal of physiology. Cell physiology 20081101
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Adenosine A2A receptor activation reduces infarct size in the isolated, perfused mouse heart by inhibiting resident cardiac mast cell degranulation.
American journal of physiology. Heart and circulatory physiology 20081101
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Role of CYP epoxygenases in A2A AR-mediated relaxation using A2A AR-null and wild-type mice.
American journal of physiology. Heart and circulatory physiology 20081101
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Adenosine and adenosine uptake inhibitors potentiate the neuromuscular blocking action of rocuronium mediated by adenosine A(1) receptors in isolated rat diaphragms.
Acta anaesthesiologica Scandinavica 20081101
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Nucleus accumbens adenosine A2A receptors regulate exertion of effort by acting on the ventral striatopallidal pathway.
The Journal of neuroscience : the official journal of the Society for Neuroscience 20080903
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Intra-accumbens injections of the adenosine A2A agonist CGS 21680 affect effort-related choice behavior in rats.
Psychopharmacology 20080901
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Activation of the A(3) adenosine receptor suppresses superoxide production and chemotaxis of mouse bone marrow neutrophils.
Molecular pharmacology 20080901
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Caffeine stimulates cytochrome oxidase expression and activity in the striatum in a sexually dimorphic manner.
Molecular pharmacology 20080901
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Human equilibrative nucleoside transporters 1 and 2 may be differentially modulated by A2B adenosine receptors in placenta microvascular endothelial cells from pre-eclampsia.
Placenta 20080901
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Effects of binge alcohol exposure in the second trimester on intracerebral arteriolar function in third trimester fetal sheep.
Brain research 20080821
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Molecular modeling of a PAMAM-CGS21680 dendrimer bound to an A2A adenosine receptor homodimer.
Bioorganic & medicinal chemistry letters 20080801
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Brain-derived neurotrophic factor inhibits GABA uptake by the rat hippocampal nerve terminals.
Brain research 20080711
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Adenosine A1 and A2A receptor regulation of protein phosphatase 2A in the murine heart.
Journal of cellular physiology 20080701
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Adenosine-dependent activation of hypoxia-inducible factor-1 induces late preconditioning in liver cells.
Hepatology (Baltimore, Md.) 20080701
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Adenosine receptor agonists attenuate the development of diazepam withdrawal-induced sensitization in mice.
European journal of pharmacology 20080624
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Expression of adenosine A 2A receptors in the rat lumbar spinal cord and implications in the modulation of N-methyl-d-aspartate receptor currents.
Anesthesia and analgesia 20080601
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Systemic administration of the adenosine A(2A) agonist CGS 21680 induces sedation at doses that suppress lever pressing and food intake.
Pharmacology, biochemistry, and behavior 20080501
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Gene expression in the rat brain during prostaglandin D2 and adenosinergically-induced sleep.
Journal of neurochemistry 20080501
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Enhancement of long-term potentiation by brain-derived neurotrophic factor requires adenosine A2A receptor activation by endogenous adenosine.
Neuropharmacology 20080501
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Up-regulation of A 2B adenosine receptor in A 2A adenosine receptor knockout mouse coronary artery.
Journal of molecular and cellular cardiology 20080501
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[Different effects of adenosine A2A receptors in the models of traumatic brain injury and peripheral tissue injury].
Sheng li xue bao : [Acta physiologica Sinica] 20080425
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Actions of adenosine A 2A receptors on synaptic connections of spiny projection neurons in the neostriatal inhibitory network.
Journal of neurophysiology 20080401
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Spinal adenosine A2a receptor activation elicits long-lasting phrenic motor facilitation.
The Journal of neuroscience : the official journal of the Society for Neuroscience 20080227
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Inhaled adenosine A(2A) receptor agonists for the treatment of chronic obstructive pulmonary disease.
Bioorganic & medicinal chemistry letters 20080215
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A1 and A2A receptor activation by endogenous adenosine is required for VIP enhancement of K+ -evoked [3H]-GABA release from rat hippocampal nerve terminals.
Neuroscience letters 20080117
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Adenosine A2A receptor agonists inhibit lipopolysaccharide-induced production of tumor necrosis factor-alpha by equine monocytes.
Veterinary immunology and immunopathology 20080115
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Adenosine A2A receptors are essential for long-term potentiation of NMDA-EPSCs at hippocampal mossy fiber synapses.
Neuron 20080110
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Fetal alcohol exposure alters cerebrovascular reactivity to vasoactive intestinal peptide in adult sheep.
Neonatology 20080101
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Effect of adenosine A2 receptor stimulation on platelet activation-aggregation: differences between canine and human models.
Thrombosis research 20080101
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Regulation of A(2A) adenosine receptor expression and functioning following permanent focal ischemia in rat brain.
Journal of neurochemistry 20080101
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Flow cytometry application for studies on adenosine A2A receptors expression.
Acta poloniae pharmaceutica 20080101
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Paradoxical effects of adenosine receptor ligands on hydroxyl radical generation by L-DOPA in the rat striatum.
Pharmacological reports : PR 20080101
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Effect of the pyridoindole SMe1EC2 and compounds affecting A(1) and A(2A) adenosine receptors in rat hippocampus under ischemia in vitro.
Pharmacological reports : PR 20080101
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Involvement of adenosine receptor agonists on the development of hypersensitivity to acute dose of morphine during morphine withdrawal period.
Pharmacological reports : PR 20080101
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The effect of caffeine to increase reaction time in the rat during a test of attention is mediated through antagonism of adenosine A2A receptors.
Behavioural brain research 20071211
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Adenosine A1 and A2A receptor effects on G-protein cycling in beta-adrenergic stimulated ventricular membranes.
Journal of cellular physiology 20071201
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Adenosine induces expression of glial cell line-derived neurotrophic factor (GDNF) in primary rat astrocytes.
Neuroscience research 20071201
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Protective roles of adenosine A1, A2A, and A3 receptors in skeletal muscle ischemia and reperfusion injury.
American journal of physiology. Heart and circulatory physiology 20071201
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Altering cAMP levels within a central pattern generator modifies or disrupts rhythmic motor output.
Journal of comparative physiology. A, Neuroethology, sensory, neural, and behavioral physiology 20071201
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Wound healing is impaired in MyD88-deficient mice: a role for MyD88 in the regulation of wound healing by adenosine A2A receptors.
The American journal of pathology 20071201
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Pharmacological characterization of a novel, potent adenosine A1 and A2A receptor dual antagonist, 5-[5-amino-3-(4-fluorophenyl)pyrazin-2-yl]-1-isopropylpyridine-2(1H)-one (ASP5854), in models of Parkinson's disease and cognition.
The Journal of pharmacology and experimental therapeutics 20071101
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Interaction of A2A adenosine and D2 dopamine receptors modulates corticostriatal glutamatergic transmission.
Neuropharmacology 20071101
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Transient inhibition of astrocytogenesis in developing mouse brain following postnatal caffeine exposure.
Pediatric research 20071101
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Adenosine receptor A2A-R contributes to motoneuron survival by transactivating the tyrosine kinase receptor TrkB.
Proceedings of the National Academy of Sciences of the United States of America 20071023
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Purinergic modulation of glutamate release under ischemic-like conditions in the hippocampus.
Neuroscience 20071012
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Activation of central adenosine A(2A) receptors enhances superior laryngeal nerve stimulation-induced apnea in piglets via a GABAergic pathway.
Journal of applied physiology (Bethesda, Md. : 1985) 20071001
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The neuronal Ca(2+) -binding protein 2 (NECAB2) interacts with the adenosine A(2A) receptor and modulates the cell surface expression and function of the receptor.
Molecular and cellular neurosciences 20070901
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Pharmacologic characterization of novel adenosine A2A receptor agonists in equine neutrophils.
American journal of veterinary research 20070901
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The role of adenosine A1 and A2A receptors of entorhinal cortex on piriform cortex kindled seizures in rats.
Pharmacological research 20070801
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Adenosine stimulates the basolateral 50 pS K channels in the thick ascending limb of the rat kidney.
American journal of physiology. Renal physiology 20070701
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Adenosine closes the K+ channel KCa3.1 in human lung mast cells and inhibits their migration via the adenosine A2A receptor.
European journal of immunology 20070601
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Anticonvulsant effect of A1 but not A2A adenosine receptors of piriform cortex in amygdala-kindled rats.
Canadian journal of physiology and pharmacology 20070601
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The adenosine A2A receptor agonist CGS 21680 fails to ameliorate the course of dextran sulphate-induced colitis in mice.
Inflammation research : official journal of the European Histamine Research Society ... [et al.] 20070501
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Opposite effects of the A2A receptor agonist CGS21680 in the striatum of Huntington's disease versus wild-type mice.
Neuroscience letters 20070424
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The adenosine A2A receptor agonist, CGS-21680, blocks excessive rearing, acquisition of wheel running, and increases nucleus accumbens CREB phosphorylation in chronically food-restricted rats.
Brain research 20070420
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Mitogen-activated protein kinase signaling is involved in suramin-induced neurite outgrowth in a neuronal cell line.
Biochemical and biophysical research communications 20070413
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Characterization of the potency, selectivity, and pharmacokinetic profile for six adenosine A2A receptor antagonists.
Naunyn-Schmiedeberg's archives of pharmacology 20070401
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Hyperalgesia, low-anxiety, and impairment of avoidance learning in neonatal caffeine-treated rats.
Psychopharmacology 20070301
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Attenuation of experimental subarachnoid hemorrhage--induced cerebral vasospasm by the adenosine A2A receptor agonist CGS 21680.
Journal of neurosurgery 20070301
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Stimulation of adenosine A1 and A2A receptors by AMP in the submucosal plexus of guinea pig small intestine.
American journal of physiology. Gastrointestinal and liver physiology 20070201
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Evaluation of neuronal phosphoproteins as effectors of caffeine and mediators of striatal adenosine A2A receptor signaling.
Brain research 20070119
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Contractile effects of adenosine, coronary flow and perfusion pressure in murine myocardium.
Pflugers Archiv : European journal of physiology 20070101
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Effects of adenosine on functions of polymorphonuclear leukocytes from patients with septic shock.
Shock (Augusta, Ga.) 20070101
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Protective effect of adenosine A2A receptor activation in small-for-size liver transplantation.
Transplant international : official journal of the European Society for Organ Transplantation 20070101
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Adenosine A2A receptor modulation of juvenile female rat skeletal muscle microvessel permeability.
American journal of physiology. Heart and circulatory physiology 20061201
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Protective effects of adenosine A2A agonist during hemorrhagic shock: a simple intervention may result in a complex response.
Critical care medicine 20061201
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The impact of adenosine and A(2B) receptors on glucose homoeostasis.
The Journal of pharmacy and pharmacology 20061201
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Expression of adenosine receptors in cardiac fibroblasts as a function of insulin and glucose level.
Archives of biochemistry and biophysics 20061101
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Adenosine A2A receptors are expressed in human atrial myocytes and modulate spontaneous sarcoplasmic reticulum calcium release.
Cardiovascular research 20061101
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Experimental studies and theoretical aspects on A2A/D2 receptor interactions in a model of Parkinson's disease. Relevance for L-dopa induced dyskinesias.
Journal of the neurological sciences 20061025
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Glial cell line-derived neurotrophic factor (GDNF) enhances dopamine release from striatal nerve endings in an adenosine A2A receptor-dependent manner.
Brain research 20061003
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Stimulation of adenosine receptors selectively activates gene expression in striatal enkephalinergic neurons.
Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology 20061001
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Corpus cavernosum from men with vasculogenic impotence is partially resistant to adenosine relaxation due to endothelial A(2B) receptor dysfunction.
The Journal of pharmacology and experimental therapeutics 20061001
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Evidence for both adenosine A1 and A2A receptors activating single vagal sensory C-fibres in guinea pig lungs.
The Journal of physiology 20060901
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A role for Fyn in Trk receptor transactivation by G-protein-coupled receptor signaling.
Molecular and cellular neurosciences 20060901
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Triggering of BDNF facilitatory action on neuromuscular transmission by adenosine A2A receptors.
Neuroscience letters 20060814
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Role of adenosine A1 receptors in the modulation of dopamine D1 and adenosine A2A receptor signaling in the neostriatum.
Neuroscience 20060811
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Activation of adenosine A2A receptors alters postsynaptic currents and depolarizes neurons of the supraoptic nucleus.
American journal of physiology. Regulatory, integrative and comparative physiology 20060801
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Adenosine is upregulated during peritonitis and is involved in downregulation of inflammation.
Kidney international 20060801
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Contribution of adenosine receptors in the control of arteriolar tone and adenosine-angiotensin II interaction.
Kidney international 20060801
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Adenosine2A receptor vasodilation of rat preglomerular microvessels is mediated by EETs that activate the cAMP/PKA pathway.
American journal of physiology. Renal physiology 20060701
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Adenosine A2a receptors induce heterologous desensitization of chemokine receptors.
Blood 20060701
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Adenosine A2A receptor mediated protective effect of 2-(6-cyano-1-hexyn-1-yl)adenosine on retinal ischaemia/reperfusion damage in rats.
The British journal of ophthalmology 20060701
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Adenosine A2A receptor stimulation decreases GAT-1-mediated GABA uptake in the globus pallidus of the rat.
Neuropharmacology 20060701
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Reduction of apoptosis in the amygdala by an A2A adenosine receptor agonist following myocardial infarction.
Apoptosis : an international journal on programmed cell death 20060701
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Expression pattern of FOS in orexin neurons during sleep induced by an adenosine A2A receptor agonist.
Behavioural brain research 20060630
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A novel cell-based assay for G-protein-coupled receptor-mediated cyclic adenosine monophosphate response element binding protein phosphorylation.
Journal of biomolecular screening 20060601
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Inhibition of platelet-activating factor biosynthesis by adenosine and histamine in human neutrophils: involvement of cPLA2alpha and reversal by lyso-PAF.
Journal of leukocyte biology 20060501
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Microsphere-based protease assays and screening application for lethal factor and factor Xa.
Cytometry. Part A : the journal of the International Society for Analytical Cytology 20060501
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The effect of A2A adenosine receptor agonist on composite tissue allotransplant survival: an in vivo preliminary study.
The Journal of surgical research 20060401
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Adenosine A2A receptor activation reduces lung injury in trauma/hemorrhagic shock.
Critical care medicine 20060401
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Differential expression of adenosine receptors in human neutrophils: up-regulation by specific Th1 cytokines and lipopolysaccharide.
Journal of leukocyte biology 20060301
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Adenosine receptor modelling. A1/A2a selectivity.
European journal of medicinal chemistry 20060301
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Dialysis delivery of an adenosine A2A agonist into the pontine reticular formation of C57BL/6J mouse increases pontine acetylcholine release and sleep.
Journal of neurochemistry 20060301
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A2a receptors mediate inhibitory effects of adenosine on colonic motility in the presence of experimental colitis.
Inflammatory bowel diseases 20060201
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Adenosine A2A receptors mediate GABAergic inhibition of respiration in immature rats.
Journal of applied physiology (Bethesda, Md. : 1985) 20060101
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Contractile effects of adenosine A1 and A2A receptors in isolated murine hearts.
American journal of physiology. Heart and circulatory physiology 20060101
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Adenosine A1 and A2A receptors of hippocampal CA1 region have opposite effects on piriform cortex kindled seizures in rats.
Seizure 20060101
-
Involvement of peripheral adenosine A2 receptors in adenosine A1 receptor-mediated recovery of respiratory motor function after upper cervical spinal cord hemisection.
The journal of spinal cord medicine 20060101
-
The role of adenosine A2a receptors in experimental acute pancreatitis.
Advances in medical sciences 20060101
-
Characterization of the effects of adenosine receptor agonists on cerebral blood flow in uninjured and traumatically injured rat brain using continuous arterial spin-labeled magnetic resonance imaging.
Journal of cerebral blood flow and metabolism : official journal of the International Society of Cerebral Blood Flow and Metabolism 20051201
-
Adenosine A1 receptors mediate inhibition of cAMP formation in vitro in the pontine, REM sleep induction zone.
Brain research 20051109
-
Adenosine A2A receptor stimulation potentiates nitric oxide release by activated microglia.
Journal of neurochemistry 20051101
-
Adenosine A2A receptors and metabotropic glutamate 5 receptors are co-localized and functionally interact in the hippocampus: a possible key mechanism in the modulation of N-methyl-D-aspartate effects.
Journal of neurochemistry 20051101
-
Influence of adenosine receptor agonists on benzodiazepine withdrawal signs in mice.
European journal of pharmacology 20051031
-
Effect of adenosine A2A receptor agonist (CGS) on ischemia/reperfusion injury in isolated rat liver.
Apoptosis : an international journal on programmed cell death 20051001
-
Persistent upregulation of mu-opioid, but not adenosine, receptors in brains of long-term withdrawn escalating dose 'binge' cocaine-treated rats.
Synapse (New York, N.Y.) 20050901
-
Adenosine triggers preconditioning through MEK/ERK1/2 signalling pathway during hypoxia/reoxygenation in neonatal rat cardiomyocytes.
Journal of molecular and cellular cardiology 20050901
-
2-(1-Hexyn-1-yl)adenosine-induced intraocular hypertension is mediated via K+ channel opening through adenosine A2A receptor in rabbits.
European journal of pharmacology 20050822
-
Adenosine inhibits the release of interleukin-1beta in activated human peripheral mononuclear cells.
Cytokine 20050821
-
Exaggerated response to adenosine in kidneys from high salt-fed rats: role of epoxyeicosatrienoic acids.
American journal of physiology. Renal physiology 20050801
-
Activation of Th1 and Tc1 cell adenosine A2A receptors directly inhibits IL-2 secretion in vitro and IL-2-driven expansion in vivo.
Blood 20050615
-
Requisite roles of A2A receptors, nitric oxide, and KATP channels in retinal arteriolar dilation in response to adenosine.
Investigative ophthalmology & visual science 20050601
-
Adenosine A2A receptor stimulation increases angiogenesis by down-regulating production of the antiangiogenic matrix protein thrombospondin 1.
Molecular pharmacology 20050501
-
Activation of adenosine receptors in the posterior cingulate cortex impairs memory retrieval in the rat.
Neurobiology of learning and memory 20050501
-
Sustained cardioprotection afforded by A2A adenosine receptor stimulation after 72 hours of myocardial reperfusion.
Journal of cardiovascular pharmacology 20050501
-
CGS21680 attenuates symptoms of Huntington's disease in a transgenic mouse model.
Journal of neurochemistry 20050401
-
The role of adenosine A2A and A2B receptors in the regulation of TNF-alpha production by human monocytes.
Biochemical pharmacology 20050315
-
Role of central and peripheral adenosine receptors in the cardiovascular responses to intraperitoneal injections of adenosine A1 and A2A subtype receptor agonists.
British journal of pharmacology 20050301
-
An adenosine A receptor agonist induces sleep by increasing GABA release in the tuberomammillary nucleus to inhibit histaminergic systems in rats.
Journal of neurochemistry 20050301
-
Kinetic and functional properties of [3H]ZM241385, a high affinity antagonist for adenosine A2A receptors.
Life sciences 20050211
-
Adenosine A2A receptor and dopamine D3 receptor interactions: evidence of functional A2A/D3 heteromeric complexes.
Molecular pharmacology 20050201
-
Co-localization and functional interaction between adenosine A(2A) and metabotropic group 5 receptors in glutamatergic nerve terminals of the rat striatum.
Journal of neurochemistry 20050201
-
Upregulation of A2A adenosine receptor expression by TNF-alpha in PBMC of patients with CHF: a regulatory mechanism of inflammation.
Journal of cardiac failure 20050201
-
Functional expression of single-chain heterodimeric G-protein-coupled receptors for adenosine and dopamine.
Cell structure and function 20050201
-
In vitro platelet responsiveness to adenosine-mediated 'preconditioning' is age-dependent.
Journal of thrombosis and thrombolysis 20050201
-
Inhibition of phenylephrine-induced cardiomyocyte hypertrophy by activation of multiple adenosine receptor subtypes.
The Journal of pharmacology and experimental therapeutics 20050101
-
Hypoxia induces neurite outgrowth in PC12 cells that is mediated through adenosine A2A receptors.
Neuroscience 20050101
-
A2B adenosine receptor activity is reduced in neutrophils from patients with systemic sclerosis.
Arthritis research & therapy 20050101
-
Trafficking of adenosine A2A and dopamine D2 receptors.
Journal of molecular neuroscience : MN 20050101
-
Effects of adenosine and adenosine A2A receptor agonist on motor nerve conduction velocity and nerve blood flow in experimental diabetic neuropathy.
Neurological research 20050101
-
Distinctive and synergistic signaling of human adenosine A2a and dopamine D2L receptors in CHO cells.
Journal of receptor and signal transduction research 20050101
-
Small conductance calcium-activated K+ channels, SkCa, but not voltage-gated K+ (Kv) channels, are implicated in the antinociception induced by CGS21680, a A2A adenosine receptor agonist.
Life sciences 20041210
-
Regulation of A2B adenosine receptor functioning by tumour necrosis factor a in human astroglial cells.
Journal of neurochemistry 20041201
-
Autoinhibition of transmitter release from PC12 cells and sympathetic neurons through a P2Y receptor-mediated inhibition of voltage-gated Ca2+ channels.
The European journal of neuroscience 20041201
-
Adenosine A2A receptor facilitates calcium-dependent protein secretion through the activation of protein kinase A and phosphatidylinositol-3 kinase in PC12 cells.
Cell structure and function 20041201
-
Dietary K intake regulates the response of apical K channels to adenosine in the thick ascending limb.
American journal of physiology. Renal physiology 20041101
-
Effects of adenosine on optic nerve head circulation in rabbits.
Experimental eye research 20041101
-
Adenosine receptor-mediated modulation of dopamine release in the nucleus accumbens depends on glutamate neurotransmission and N-methyl-D-aspartate receptor stimulation.
Journal of neurochemistry 20041101
-
Effect of omeprazole on gastric adenosine A1 and A2A receptor gene expression and function.
The Journal of pharmacology and experimental therapeutics 20041001
-
Adenosine receptors control HIV-1 Tat-induced inflammatory responses through protein phosphatase.
Virology 20041001
-
Binding of adenosine receptor ligands to brain of adenosine receptor knock-out mice: evidence that CGS 21680 binds to A1 receptors in hippocampus.
Naunyn-Schmiedeberg's archives of pharmacology 20041001
-
Hypoxanthine effects on cyclic AMP levels in human lymphocytes.
Nucleosides, nucleotides & nucleic acids 20041001
-
Adenosine A2A receptor occupancy stimulates expression of proteins involved in reverse cholesterol transport and inhibits foam cell formation in macrophages.
Journal of leukocyte biology 20040901
-
Facilitation of noradrenaline release by activation of adenosine A(2A) receptors triggers both phospholipase C and adenylate cyclase pathways in rat tail artery.
Cardiovascular research 20040901
-
Permissive role of adenosine A2A receptors on metabotropic glutamate receptor 5 (mGluR5)-mediated effects in the striatum.
Journal of neurochemistry 20040901
-
Neuroprotective effect of L-DOPA co-administered with the adenosine A2A receptor agonist CGS 21680 in an animal model of Parkinson's disease.
Brain research bulletin 20040830
-
Role of adenosine A1 receptor in the regulation of gastrin release.
The Journal of pharmacology and experimental therapeutics 20040801
-
The synergistic effect of adenosine A2A receptors agonist, type IV phosphodiestease inhibitor and ATP-sensitive K channels activation on free radicals production and aggregation of human polymorphoneuclear leukocytes.
Pharmacological research 20040801
-
Neuronal A1 receptors mediate increase in extracellular kynurenic acid after local intrastriatal adenosine infusion.
Journal of neurochemistry 20040801
-
Transactivation of Trk neurotrophin receptors by G-protein-coupled receptor ligands occurs on intracellular membranes.
The Journal of neuroscience : the official journal of the Society for Neuroscience 20040728
-
Adenosine A2A receptors interact with GABAergic pathways to modulate respiration in neonatal piglets.
Respiratory physiology & neurobiology 20040720
-
Activation of adenosine A2A receptor protects sympathetic neurons against nerve growth factor withdrawal.
Journal of neuroscience research 20040715
-
Adenosine A2A receptor blockade differentially influences excitotoxic mechanisms at pre- and postsynaptic sites in the rat striatum.
Journal of neuroscience research 20040701
-
Adenosine A2A receptor-induced inhibition of NMDA and GABAA receptor-mediated synaptic currents in a subpopulation of rat striatal neurons.
Neuropharmacology 20040601
-
Adenosine A(2A) receptor activation promotes wound neovascularization by stimulating angiogenesis and vasculogenesis.
The American journal of pathology 20040601
-
An IgM class anti-neutrophil cytoplasm antibody inhibits neutrophil adhesion and apoptosis via a Syk dependent signaling cascade.
Molecular immunology 20040601
-
Role of adenosine A2A receptor in the regulation of gastric somatostatin release.
The Journal of pharmacology and experimental therapeutics 20040501
-
Protection against cisplatin ototoxicity by adenosine agonists.
Biochemical pharmacology 20040501
-
Direct interaction of adenosine with the TRPV1 channel protein.
The Journal of neuroscience : the official journal of the Society for Neuroscience 20040407
-
[Role of adenosine in intraocular pressure].
Nihon yakurigaku zasshi. Folia pharmacologica Japonica 20040401
-
Activation of adenosine A2A receptor facilitates brain-derived neurotrophic factor modulation of synaptic transmission in hippocampal slices.
The Journal of neuroscience : the official journal of the Society for Neuroscience 20040324
-
Binding of the prototypical adenosine A(2A) receptor agonist CGS 21680 to the cerebral cortex of adenosine A(1) and A(2A) receptor knockout mice.
British journal of pharmacology 20040301
-
Post-ischemic cardioprotection by A2A adenosine receptors: dependent of phosphatidylinositol 3-kinase pathway.
Journal of cardiovascular pharmacology 20040301
-
Down-regulation of rat brain adenosine A1 receptors at the end of pregnancy.
Journal of neurochemistry 20040201
-
Lack of adenosine A1 and dopamine D2 receptor-mediated modulation of the cardiovascular effects of the adenosine A2A receptor agonist CGS 21680.
European journal of pharmacology 20040126
-
Input-specific modulation of neurotransmitter release in the lateral horn of the spinal cord via adenosine receptors.
The Journal of neuroscience : the official journal of the Society for Neuroscience 20040107
-
Stimulation of adenosine A2A receptors elicits zif/268 and NMDA epsilon2 subunit mRNA expression in cortex and striatum of the 'weaver' mutant mouse, a genetic model of nigrostriatal dopamine deficiency.
Neuroscience 20040101
-
Synthesis and structure-activity relationships of 4-cycloalkylamino-1, 2, 4-triazolo[4, 3-a]quinoxalin-1- one derivatives as A1 and A3 adenosine receptor antagonists.
Archiv der Pharmazie 20040101
-
Effects of stable adenosine receptor agonists on bone marrow hematopoietic cells as inferred from the cytotoxic action of 5-fluorouracil.
Physiological research 20040101
-
Barium, glibenclamide and CGS21680 prevent adenosine A1 receptor changes of ES coupling and spike threshold.
Neuro-Signals 20040101
-
Changes in intracellular cyclic AMP formation mask opposing modulation of kainate-enhanced glutamate release in the striatum.
Proceedings of the Western Pharmacology Society 20040101
-
Modulation of GABAergic transmission in the striatopallidal system by adenosine A2A receptors: a potential mechanism for the antiparkinsonian effects of A2A antagonists.
Neurology 20031209
-
Sleep regulation in adenosine A2A receptor-deficient mice.
Neurology 20031209
-
Adenosine modulation of [Ca2+]i in cerebellar granular cells: multiple adenosine receptors involved.
Brain research 20031205
-
Involvement of adenosine A1 and A2A receptors in the adenosinergic modulation of the discriminative-stimulus effects of cocaine and methamphetamine in rats.
The Journal of pharmacology and experimental therapeutics 20031201
-
Th1 cytokines regulate adenosine receptors and their downstream signaling elements in human microvascular endothelial cells.
Journal of immunology (Baltimore, Md. : 1950) 20031015
-
Blockade of A2A adenosine receptors prevents basic fibroblast growth factor-induced reactive astrogliosis in rat striatal primary astrocytes.
Glia 20030801
-
Adenosine inhibits activation-induced T cell expression of CD2 and CD28 co-stimulatory molecules: role of interleukin-2 and cyclic AMP signaling pathways.
Journal of cellular biochemistry 20030801
-
Enhanced adenosine A2A receptor facilitation of synaptic transmission in the hippocampus of aged rats.
Journal of neurophysiology 20030801
-
Adenosine A 2B receptors modulate cAMP levels and induce CREB but not ERK1/2 and p38 phosphorylation in rat skeletal muscle cells.
Biochemical and biophysical research communications 20030718
-
Influence of CGS 21680, a selective adenosine A(2A) agonist, on the phencyclidine-induced sensorimotor gating deficit and motor behaviour in rats.
Psychopharmacology 20030701
-
Involvement of adenosine A1 and A2A receptors in the motor effects of caffeine after its acute and chronic administration.
Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology 20030701
-
The human D2 dopamine receptor synergizes with the A2A adenosine receptor to stimulate adenylyl cyclase in PC12 cells.
Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology 20030701
-
Enabling role of adenosine A1 receptors in adenosine A2A receptor-mediated striatal expression of c-fos.
The European journal of neuroscience 20030701
-
A dual role of adenosine A2A receptors in 3-nitropropionic acid-induced striatal lesions: implications for the neuroprotective potential of A2A antagonists.
The Journal of neuroscience : the official journal of the Society for Neuroscience 20030615
-
Characterization of adenosine receptor(s) involved in adenosine-induced bronchoconstriction in an allergic mouse model.
American journal of physiology. Lung cellular and molecular physiology 20030601
-
Adenosine-mediated early preconditioning in mouse: protective signaling and concentration dependent effects.
Cardiovascular research 20030601
-
Adenosine A2A receptor-mediated facilitation of noradrenaline release involves protein kinase C activation and attenuation of presynaptic inhibitory receptor-mediated effects in the rat vas deferens.
Journal of neurochemistry 20030501
-
Binding of HTLV-1 virions to T cells occurs by a temperature and calcium-dependent process and is blocked by certain type 2 adenosine receptor antagonists.
Virus research 20030501
-
Up-regulation of striatal adenosine A(2A) receptors in schizophrenia.
Neuroreport 20030303
-
Differential allosteric modulation by amiloride analogues of agonist and antagonist binding at A(1) and A(3) adenosine receptors.
Biochemical pharmacology 20030215
-
Regional differences in the adenosine A(2) receptor-mediated modulation of contractions in rat vas deferens.
European journal of pharmacology 20030124
-
Positive coupling of atypical adenosine A3 receptors on human eosinophils to adenylyl cyclase.
Biochemical and biophysical research communications 20030117
-
Sole activation of three luminal adenosine receptor subtypes in different parts of coronary vasculature.
American journal of physiology. Heart and circulatory physiology 20030101
-
A role for histamine in cytokine modulation by the adenosine A(3) receptor agonist, 2-Cl-IB-MECA.
European journal of pharmacology 20021213
-
Basolateral and apical A1 adenosine receptors mediate sodium transport in cultured renal epithelial (A6) cells.
American journal of physiology. Renal physiology 20021201
-
The adenosine A2A receptor agonist CGS 21680 exhibits antipsychotic-like activity in Cebus apella monkeys.
Behavioural pharmacology 20021201
-
Formalin-induced pain and mu-opioid receptor density in brain and spinal cord are modulated by A1 and A2a adenosine agonists in mice.
Brain research 20021129
-
The A2A receptor mediates an endogenous regulatory pathway of cytokine expression in THP-1 cells.
Journal of leukocyte biology 20021101
-
Actions of specific adenosine receptor A1 and A2 agonists and antagonists in recovery of phrenic motor output following upper cervical spinal cord injury in adult rats.
Clinical and experimental pharmacology & physiology 20021001
-
Early activation of the p42/p44MAPK pathway mediates adenosine-induced nitric oxide production in human endothelial cells: a novel calcium-insensitive mechanism.
FASEB journal : official publication of the Federation of American Societies for Experimental Biology 20021001
-
Presynaptic adenosine A1 receptors regulate retinohypothalamic neurotransmission in the hamster suprachiasmatic nucleus.
Journal of neurobiology 20020905
-
Involvement of DARPP-32 phosphorylation in the stimulant action of caffeine.
Nature 20020815
-
Suppression of adenosine A(3) receptor-mediated hypotension and mast cell degranulation in the rat by dexamethasone.
The Journal of pharmacology and experimental therapeutics 20020801
-
Chronic caffeine treatment causes changes in cardiac adenosine receptor function in rats.
Pharmacology 20020701
-
Coronary function and adenosine receptor-mediated responses in ischemic-reperfused mouse heart.
Cardiovascular research 20020701
-
Selective allosteric enhancement of agonist binding and function at human A3 adenosine receptors by a series of imidazoquinoline derivatives.
Molecular pharmacology 20020701
-
[Role of G-protein-coupled adenosine receptors in downregulation of inflammation and protection from tissue damage].
Zeitschrift fur Gastroenterologie 20020701
-
Targeted deletion of adenosine A(3) receptors augments adenosine-induced coronary flow in isolated mouse heart.
American journal of physiology. Heart and circulatory physiology 20020601
-
Effects of adenosine A1 and A2A receptor activation on the evoked release of glutamate from rat cerebrocortical synaptosomes.
British journal of pharmacology 20020601
-
Adenosine promotes wound healing and mediates angiogenesis in response to tissue injury via occupancy of A(2A) receptors.
The American journal of pathology 20020601
-
Synergistic up-regulation of vascular endothelial growth factor expression in murine macrophages by adenosine A(2A) receptor agonists and endotoxin.
The American journal of pathology 20020601
-
Effects of adenosine receptor agonists on guinea-pig isolated working hearts and the role of endothelium and NO.
The Journal of pharmacy and pharmacology 20020601
-
Metabotropic glutamate mGlu5 receptor-mediated modulation of the ventral striopallidal GABA pathway in rats. Interactions with adenosine A(2A) and dopamine D(2) receptors.
Neuroscience letters 20020517
-
Dissociation of the PAF-receptor from NADPH oxidase and adenylate cyclase in human neutrophils results in accelerated influx and delayed clearance of cytosolic calcium.
British journal of pharmacology 20020501
-
Adenosine receptor-mediated control of in vitro release of pain-related neuropeptides from the rat spinal cord.
European journal of pharmacology 20020419
-
Effects of CGS 21680, a selective adenosine A2A receptor agonist, on allergic airways inflammation in the rat.
European journal of pharmacology 20020308
-
Cardiac myocyte adenosine A2a receptor activation fails to alter cAMP or contractility: role of receptor localization.
American journal of physiology. Heart and circulatory physiology 20020301
-
Regulation of glycogen metabolism in hepatocytes through adenosine receptors. Role of Ca2+ and cAMP.
European journal of pharmacology 20020222
-
Cardiac effects of adenosine in A(2A) receptor knockout hearts: uncovering A(2B) receptors.
American journal of physiology. Heart and circulatory physiology 20020201
-
Effects of adenosine agonists on consumptive behaviour and body temperature.
The Journal of pharmacy and pharmacology 20020201
-
Adenosine A2A receptor agonists promote more rapid wound healing than recombinant human platelet-derived growth factor (Becaplermin gel).
Inflammation 20020201
-
Activation of adenosine A2a receptor pathway reduces leukocyte infiltration but enhances edema formation in rat caerulein pancreatitis.
Pancreas 20020101
-
Effects of A(3) adenosine receptor activation and gene knock-out in ischemic-reperfused mouse heart.
Cardiovascular research 20020101
-
Comparison of the vascular effects of adenosine in isolated mouse heart and aorta.
American journal of physiology. Heart and circulatory physiology 20020101
-
Adenosine A(2A) receptor facilitation of hippocampal synaptic transmission is dependent on tonic A(1) receptor inhibition.
Neuroscience 20020101
-
Lipopolysaccharide binds to and activates A(1) adenosine receptors on human pulmonary artery endothelial cells.
Journal of endotoxin research 20020101
-
Adenosine A2A, 5-HT1A and 5-HT7 receptor in neonatally pregnenolone-treated rats.
Neuroreport 20011204
-
Adenosine inhibits excitatory transmission to substantia gelatinosa neurons of the adult rat spinal cord through the activation of presynaptic A(1) adenosine receptor.
Pain 20011201
-
Solubilisation and immunoprecipitation of rat striatal adenosine A(2A) receptors.
European journal of pharmacology 20011116
-
Adenosine A(2A) and A(2B) receptor activation of erythropoietin production.
American journal of physiology. Renal physiology 20011101
-
In vivo effects of adenosine A(2) receptor agonist and antagonist on neuronal and astrocytic intermediary metabolism studied with ex vivo (13)C MR spectroscopy.
Journal of neurochemistry 20011101
-
Inflammatory cytokines regulate function and expression of adenosine A(2A) receptors in human monocytic THP-1 cells.
Journal of immunology (Baltimore, Md. : 1950) 20011001
-
Adenosine-mediated hypotension in in vivo guinea-pig: receptors involved and role of NO.
British journal of pharmacology 20011001
-
Suppression of presynaptic responses to adenosine by activation of NMDA receptors.
European journal of pharmacology 20010907
-
Effects of adenosine receptor agonists and antagonists in a genetic animal model of primary paroxysmal dystonia.
British journal of pharmacology 20010901
-
Synergism between A(2A)-adenosine receptor activation and vasoactive intestinal peptide to facilitate [3H]-acetylcholine release from the rat motor nerve terminals.
Neuroscience letters 20010824
-
Adenosine A(1) receptors mediate plasma exudation from the oral mucosa.
Journal of applied physiology (Bethesda, Md. : 1985) 20010801
-
Functional characterization of coronary vascular adenosine receptors in the mouse.
British journal of pharmacology 20010801
-
Adenosine A2A agonist CGS 21680 decreases the affinity of dopamine D2 receptors for dopamine in human striatum.
Neuroreport 20010703
-
Novel short-acting A2A adenosine receptor agonists for coronary vasodilation: inverse relationship between affinity and duration of action of A2A agonists.
The Journal of pharmacology and experimental therapeutics 20010701
-
Modulation of ethanol-induced motor incoordination by mouse striatal A(1) adenosinergic receptor.
Brain research bulletin 20010701
-
The adenosine A2A agonist CGS 21680 reverses the reduction in prepulse inhibition of the acoustic startle response induced by phencyclidine, but not by apomorphine and amphetamine.
Psychopharmacology 20010701
-
Adenosine A(1) receptor-mediated inhibition of protein kinase A-induced calcitonin gene-related peptide release from rat trigeminal neurons.
Molecular pharmacology 20010601
-
Adenosine A2A receptor activation reduces proinflammatory events and decreases cell death following intracerebral hemorrhage.
Annals of neurology 20010601
-
Receptor subtypes mediating adenosine-induced dilation of cerebral arterioles.
American journal of physiology. Heart and circulatory physiology 20010501
-
Role of adenosine receptors in neuroprotective effect during global cerebral ischemia.
Bulletin of experimental biology and medicine 20010501
-
Activation of protein kinase A and atypical protein kinase C by A(2A) adenosine receptors antagonizes apoptosis due to serum deprivation in PC12 cells.
The Journal of biological chemistry 20010427
-
Beneficial effects of adenosine A(2a) agonist CGS-21680 in infarcted and stunned porcine myocardium.
American journal of physiology. Heart and circulatory physiology 20010401
-
Examination of the involvement of protein kinase A in D2 dopamine receptor antagonist-induced immediate early gene expression.
Journal of neurochemistry 20010401
-
Adenosine inhibits neutrophil vascular endothelial growth factor release and transendothelial migration via A2B receptor activation.
Shock (Augusta, Ga.) 20010401
-
Blunted adenosine A2a receptor function in platelets in patients with major depression.
European neuropsychopharmacology : the journal of the European College of Neuropsychopharmacology 20010401
-
Subchronic treatment with methamphetamine and phencyclidine differentially alters the adenosine A1 and A2A receptors in the prefrontal cortex, hippocampus, and striatum of the rat.
Neurochemical research 20010401
-
Adenosine agonists CGS 21680 and NECA inhibit the initiation of cocaine self-administration.
Pharmacology, biochemistry, and behavior 20010401
-
A(1) or A(3) adenosine receptors induce late preconditioning against infarction in conscious rabbits by different mechanisms.
Circulation research 20010316
-
Stimulation of p38 MAP kinase reduces acidosis and Na(+) overload in preconditioned hepatocytes.
FEBS letters 20010302
-
Adenosine inhibits norepinephrine release in the postischemic rat heart: the mechanism of neuronal stunning.
Cardiovascular research 20010301
-
Galpha(olf) is necessary for coupling D1 and A2a receptors to adenylyl cyclase in the striatum.
Journal of neurochemistry 20010301
-
The influence of tumour necrosis factor-alpha on the cardiovascular system of anaesthetized rats.
Naunyn-Schmiedeberg's archives of pharmacology 20010301
-
The role of the D(2) dopamine receptor (D(2)R) in A(2A) adenosine receptor (A(2A)R)-mediated behavioral and cellular responses as revealed by A(2A) and D(2) receptor knockout mice.
Proceedings of the National Academy of Sciences of the United States of America 20010213
-
Adenosine enhances glial glutamate efflux via A2a adenosine receptors.
Life sciences 20010209
-
Functional and molecular characterization of receptor subtypes mediating coronary microvascular dilation to adenosine.
Journal of molecular and cellular cardiology 20010201
-
Adenosine A(2A) receptors mediate cardiovascular responses to hypoxia in fetal sheep.
American journal of physiology. Heart and circulatory physiology 20010101
-
Adenosine attenuates reperfusion-induced apoptotic cell death by modulating expression of Bcl-2 and Bax proteins.
Journal of molecular and cellular cardiology 20010101
-
An adenosine A2a agonist increases sleep and induces Fos in ventrolateral preoptic neurons.
Neuroscience 20010101
-
Role of endothelium in ischaemia-induced myocardial dysfunction of isolated working hearts: cardioprotection by activation of adenosine A(2A) receptors.
Journal of autonomic pharmacology 20010101
-
N-cycloalkyl derivatives of adenosine and 1-deazaadenosine as agonists and partial agonists of the A(1) adenosine receptor.
Journal of medicinal chemistry 20000127
-
Actions of adenosine A2A receptor antagonist KW-6002 on drug-induced catalepsy and hypokinesia caused by reserpine or MPTP.
Psychopharmacology 19991101
-
Differences in the order of potency for agonists but not antagonists at human and rat adenosine A2A receptors.
Biochemical pharmacology 19990101
-
Comparative pharmacology of human adenosine receptor subtypes - characterization of stably transfected receptors in CHO cells.
Naunyn-Schmiedeberg's archives of pharmacology 19980101
-
Mechanism and pressor relevance of the short-term cardiovascular and renin excitatory actions of the selective A2A-adenosine receptor agonists.
Journal of cardiovascular pharmacology 19970901
-
Evidence against a major role of adenosine in oxygen-dependent regulation of erythropoietin in rats.
Kidney international 19970801
-
KF17837: a novel selective adenosine A2A receptor antagonist with anticataleptic activity.
European journal of pharmacology 19940502
-
Structure-activity relationships of 8-styrylxanthines as A2-selective adenosine antagonists.
Journal of medicinal chemistry 19930514
-
Binding of the adenosine A2 receptor ligand [3H]CGS 21680 to human and rat brain: evidence for multiple affinity sites.
Journal of neurochemistry 19901101
-
[3H]CGS 21680, a selective A2 adenosine receptor agonist directly labels A2 receptors in rat brain.
The Journal of pharmacology and experimental therapeutics 19891201