-
Role of TRPA1 in acute cardiopulmonary toxicity of inhaled acrolein.
Toxicology and applied pharmacology 20170601
-
Gastroprotective and ulcer healing effects of hydroethanolic extract of leaves of Caryocar coriaceum: Mechanisms involved in the gastroprotective activity.
Chemico-biological interactions 20170105
-
Inhibition of interleukin-1β-induced endothelial tissue factor expression by the synthetic cannabinoid WIN 55,212-2.
Oncotarget 20160920
-
α,β-Unsaturated aldehyde pollutant acrolein suppresses cardiomyocyte contractile function: Role of TRPV1 and oxidative stress.
Environmental toxicology 20150101
-
Synthesis and pharmacological evaluation of novel N-aryl-3,4-dihydro-1'H-spiro[chromene-2,4'-piperidine]-1'-carboxamides as TRPM8 antagonists.
Bioorganic & medicinal chemistry 20131101
-
Peripheral antinociceptive action of mangiferin in mouse models of experimental pain: role of endogenous opioids, K(ATP)-channels and adenosine.
Pharmacology, biochemistry, and behavior 20130901
-
Study on TRPV1-mediated mechanism for the hypersecretion of mucus in respiratory inflammation.
Molecular immunology 20130101
-
Role of transient receptor potential ion channels and evoked levels of neuropeptides in a formaldehyde-induced model of asthma in BALB/c mice.
PloS one 20130101
-
Peripheral antinociceptive effect of anandamide and drugs that affect the endocannabinoid system on the formalin test in normal and streptozotocin-diabetic rats.
Neuropharmacology 20121201
-
Transient receptor potential vanilloid subtype 1 contributes to mesencephalic dopaminergic neuronal survival by inhibiting microglia-originated oxidative stress.
Brain research bulletin 20121101
-
Role of KATP channels and TRPV1 receptors in hydrogen sulfide-enhanced gastric emptying of liquid in awake mice.
European journal of pharmacology 20121015
-
Protection of ghrelin postconditioning on hypoxia/reoxygenation in gastric epithelial cells.
World journal of gastroenterology 20121014
-
Using novel in vitro NociOcular assay based on TRPV1 channel activation for prediction of eye sting potential of baby shampoos.
Toxicological sciences : an official journal of the Society of Toxicology 20121001
-
Acute myocardial infarction inhibits the neurogenic tachycardic and vasopressor response in rats via presynaptic cannabinoid type 1 receptor.
The Journal of pharmacology and experimental therapeutics 20121001
-
Endothelium-dependent mechanisms of the vasodilatory effect of the endocannabinoid, anandamide, in the rat pulmonary artery.
Pharmacological research 20120901
-
Proton-gated ion channels in mouse bone marrow stromal cells.
Stem cell research 20120901
-
Involvement of TRPV1 and TRPV4 channels in migration of rat pulmonary arterial smooth muscle cells.
Pflugers Archiv : European journal of physiology 20120901
-
N-arachidonoyl-serotonin in the basolateral amygdala increases anxiolytic behavior in the elevated plus maze.
Behavioural brain research 20120801
-
TRPV1-mediated calcium signal couples with cannabinoid receptors and sodium-calcium exchangers in rat odontoblasts.
Cell calcium 20120801
-
Disruption of TRPV1-mediated coupling of coronary blood flow to cardiac metabolism in diabetic mice: role of nitric oxide and BK channels.
American journal of physiology. Heart and circulatory physiology 20120715
-
Substance P release in response to cardiac ischemia from rat thoracic spinal dorsal horn is mediated by TRPV1.
Neuroscience 20120712
-
Capsaicin induces cycle arrest by inhibiting cyclin-dependent-kinase in bladder carcinoma cells.
International journal of urology : official journal of the Japanese Urological Association 20120701
-
Capacity of capsazepinoids to relax human small airways and inhibit TLR3-induced TSLP and IFNβ production in diseased bronchial epithelial cells.
International immunopharmacology 20120701
-
Extracellular matrix proteoglycan plays a pivotal role in sensitization by low pH of mechanosensitive currents in nociceptive sensory neurones.
The Journal of physiology 20120701
-
The transient receptor potential vanilloid receptor 1, TRPV1 (VR1) inhibits peristalsis in the mouse jejunum.
Archives of Iranian medicine 20120701
-
Characterization of a novel splice variant of δ ENaC subunit in human lungs.
American journal of physiology. Lung cellular and molecular physiology 20120615
-
A possible participation of transient receptor potential vanilloid type 1 channels in the antidepressant effect of fluoxetine.
European journal of pharmacology 20120615
-
Enhanced vasorelaxant effects of the endocannabinoid-like mediator, oleamide, in hypertension.
European journal of pharmacology 20120605
-
The investigation into indomethacin-induced potentiation of the contractile response to antigen in ovalbumin-sensitized guinea-pig tracheas.
Fundamental & clinical pharmacology 20120601
-
Calcium regulation by thermo- and osmosensing transient receptor potential vanilloid channels (TRPVs) in human conjunctival epithelial cells.
Histochemistry and cell biology 20120601
-
Involvement of transient receptor potential vanilloid type 1 channels in the pro-convulsant effect of anandamide in pentylenetetrazole-induced seizures.
Epilepsy research 20120601
-
Differential role of CB1 and TRPV1 receptors on anandamide modulation of defensive responses induced by nitric oxide in the dorsolateral periaqueductal gray.
Neuropharmacology 20120601
-
Ischemic neuroprotection by TRPV1 receptor-induced hypothermia.
Journal of cerebral blood flow and metabolism : official journal of the International Society of Cerebral Blood Flow and Metabolism 20120601
-
Transient receptor potential vanilloid type 1 channels contribute to reflex cutaneous vasodilation in humans.
Journal of applied physiology (Bethesda, Md. : 1985) 20120601
-
Presynaptic enhancement by eugenol of spontaneous excitatory transmission in rat spinal substantia gelatinosa neurons is mediated by transient receptor potential A1 channels.
Neuroscience 20120517
-
Acid and stretch, but not capsaicin, are effective stimuli for ATP release in the porcine bladder mucosa: Are ASIC and TRPV1 receptors involved?
European journal of pharmacology 20120515
-
Effects of hecogenin and its possible mechanism of action on experimental models of gastric ulcer in mice.
European journal of pharmacology 20120515
-
Confocal microscopy with double immunofluorescence staining reveals the functional transient receptor potential vanilloid subtype 1 expressed in myoepithelial cells of human submandibular glands.
Microscopy research and technique 20120501
-
Role of TRPV1 in consolidation of fear memories depends on the averseness of the conditioning procedure.
Neurobiology of learning and memory 20120501
-
Activation of transient receptor potential vanilloid subtype 1 increases expression and permeability of tight junction in normal and hyposecretory submandibular gland.
Laboratory investigation; a journal of technical methods and pathology 20120501
-
Transient receptor potential vanilloid 1 receptors mediate acid-induced mucin secretion via Ca2+ influx in human airway epithelial cells.
Journal of biochemical and molecular toxicology 20120501
-
20-Hydroxyeicosatetraenoic acid (20-HETE) is a novel activator of transient receptor potential vanilloid 1 (TRPV1) channel.
The Journal of biological chemistry 20120420
-
Vasorelaxation to capsaicin and its effects on calcium influx in arteries.
European journal of pharmacology 20120415
-
Cannabidiol inhibits lung cancer cell invasion and metastasis via intercellular adhesion molecule-1.
FASEB journal : official publication of the Federation of American Societies for Experimental Biology 20120401
-
Endocannabinoid analogues exacerbate marble-burying behavior in mice via TRPV1 receptor.
Neuropharmacology 20120401
-
Gastroprotective potential of frutalin, a D-galactose binding lectin, against ethanol-induced gastric lesions.
Fitoterapia 20120401
-
Cardiac-specific knockout of ET(A) receptor mitigates low ambient temperature-induced cardiac hypertrophy and contractile dysfunction.
Journal of molecular cell biology 20120401
-
Heteromeric heat-sensitive transient receptor potential channels exhibit distinct temperature and chemical response.
The Journal of biological chemistry 20120302
-
TRPV1 agonist capsaicin attenuates lung ischemia-reperfusion injury in rabbits.
The Journal of surgical research 20120301
-
Gastroprotective effect of Byrsonima sericea DC leaf extract against ethanol-induced gastric injury and its possible mechanisms of action.
Anais da Academia Brasileira de Ciencias 20120301
-
[Effects of anandamide on IL-11 production through the TRPV1 of human periodontal ligament cells].
Kokubyo Gakkai zasshi. The Journal of the Stomatological Society, Japan 20120301
-
Influence of influenza A infection on capsaicin-induced responses in murine airways.
The Journal of pharmacology and experimental therapeutics 20120201
-
Transient receptor potential vanilloid-1 participates in the inhibitory effect of ginsenoside Rg1 on capsaicin-induced interleukin-8 and prostaglandin E2 production in HaCaT cells.
The Journal of pharmacy and pharmacology 20120201
-
Use and limitations of three TRPV-1 receptor antagonists on smooth muscles of animals and man: a vote for BCTC.
European journal of pharmacology 20120105
-
Beneficial effects of capsiate on ethanol-induced mucosal injury in rats are related to stimulation of calcitonin gene-related Peptide release.
Planta medica 20120101
-
Opposing roles for cannabinoid receptor type-1 (CB₁) and transient receptor potential vanilloid type-1 channel (TRPV1) on the modulation of panic-like responses in rats.
Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology 20120101
-
Thermo-sensitive transient receptor potential vanilloid channel-1 regulates intracellular calcium and triggers chromogranin A secretion in pancreatic neuroendocrine BON-1 tumor cells.
Cellular signalling 20120101
-
Small molecule positive allosteric modulation of TRPV1 activation by vanilloids and acidic pH.
The Journal of pharmacology and experimental therapeutics 20120101
-
Peripheral glutamate receptors are required for hyperalgesia induced by capsaicin.
Pain research and treatment 20120101
-
ASICs Do Not Play a Role in Maintaining Hyperalgesia Induced by Repeated Intramuscular Acid Injections.
Pain research and treatment 20120101
-
Dragon's blood inhibits chronic inflammatory and neuropathic pain responses by blocking the synthesis and release of substance P in rats.
Journal of pharmacological sciences 20120101
-
Activation of TRPV1 by capsaicin induces functional kinin B(1) receptor in rat spinal cord microglia.
Journal of neuroinflammation 20120101
-
L type Ca²+ channel blockers prevent oxaliplatin-induced cold hyperalgesia and TRPM8 overexpression in rats.
Molecular pain 20120101
-
Anandamide induces sperm release from oviductal epithelia through nitric oxide pathway in bovines.
PloS one 20120101
-
The association of N-palmitoylethanolamine with the FAAH inhibitor URB597 impairs melanoma growth through a supra-additive action.
BMC cancer 20120101
-
Anandamide induces endothelium-dependent vasoconstriction and CGRPergic nerve-mediated vasodilatation in the rat mesenteric vascular bed.
Journal of pharmacological sciences 20120101
-
Antioncogenic effects of transient receptor potential vanilloid 1 in the progression of transitional urothelial cancer of human bladder.
ISRN urology 20120101
-
Capsaicin, a TRPV1 Ligand, Suppresses Bone Resorption by Inhibiting the Prostaglandin E Production of Osteoblasts, and Attenuates the Inflammatory Bone Loss Induced by Lipopolysaccharide.
ISRN pharmacology 20120101
-
The Effectiveness of GECB Pastille in Reducing Complications of Dry Socket Syndrome.
International journal of dentistry 20120101
-
The cytochrome P450 inhibitor, ketoconazole, inhibits oxidized linoleic acid metabolite-mediated peripheral inflammatory pain.
Molecular pain 20120101
-
Aberrant TRPV1 expression in heat hyperalgesia associated with trigeminal neuropathic pain.
International journal of medical sciences 20120101
-
Antagonism of the TRPv1 receptor partially corrects muscle metaboreflex overactivity in spontaneously hypertensive rats.
The Journal of physiology 20111215
-
Cardiovascular effects of 1-nitro-2-phenylethane, the main constituent of the essential oil of Aniba canelilla, in spontaneously hypertensive rats.
Fundamental & clinical pharmacology 20111201
-
An investigation of the safety and pharmacokinetics of the novel TRPV1 antagonist XEN-D0501 in healthy subjects.
British journal of clinical pharmacology 20111201
-
TRPV1, TRPA1, and CB1 in the isolated vagus nerve--axonal chemosensitivity and control of neuropeptide release.
Neuropeptides 20111201
-
Activation of TRPV1 reduces vascular lipid accumulation and attenuates atherosclerosis.
Cardiovascular research 20111201
-
Neurotrophins in the lower urinary tract: becoming of age.
Current neuropharmacology 20111201
-
Transient receptor potential vanilloid 1 channels modulate the anxiolytic effect of diazepam.
Brain research 20111124
-
The anti-botulism triterpenoid toosendanin elicits calcium increase and exocytosis in rat sensory neurons.
Cellular and molecular neurobiology 20111101
-
Suppression of tumor necrosis factor-α-induced nuclear factor κB activation and aromatase activity by capsaicin and its analog capsazepine.
Journal of medicinal food 20111101
-
Hydrogen sulfide upregulates cyclooxygenase-2 and prostaglandin E metabolite in sepsis-evoked acute lung injury via transient receptor potential vanilloid type 1 channel activation.
Journal of immunology (Baltimore, Md. : 1950) 20111101
-
Proteinase-activated receptor 2 sensitizes transient receptor potential vanilloid 1, transient receptor potential vanilloid 4, and transient receptor potential ankyrin 1 in paclitaxel-induced neuropathic pain.
Neuroscience 20111013
-
Capsaicinoids regulate airway anion transporters through Rho kinase- and cyclic AMP-dependent mechanisms.
American journal of respiratory cell and molecular biology 20111001
-
Opposite effect of capsaicin and capsazepine on behavioral thermoregulation in insects.
Journal of comparative physiology. A, Neuroethology, sensory, neural, and behavioral physiology 20111001
-
Contribution of peripheral vanilloid receptor to the nociception induced by injection of spermine in mice.
Pharmacology, biochemistry, and behavior 20111001
-
Characterization of capsaicin induced responses in mice vas deferens: evidence of CGRP uptake.
European journal of pharmacology 20110930
-
The Ile585Val TRPV1 variant is involved in risk of painful knee osteoarthritis.
Annals of the rheumatic diseases 20110901
-
Vanillyl nonanoate protects rat gastric mucosa from ethanol-induced injury through a mechanism involving calcitonin gene-related peptide.
European journal of pharmacology 20110901
-
Sensitivity of bronchopulmonary receptors to cold and heat mediated by transient receptor potential cation channel subtypes in an ex vivo rat lung preparation.
Respiratory physiology & neurobiology 20110815
-
Cardioprotection by ischemic postconditioning is lost in isolated perfused heart from diabetic rats: Involvement of transient receptor potential vanilloid 1, calcitonin gene-related peptide and substance P.
Regulatory peptides 20110808
-
Molecular mechanisms of activation of endothelial nitric oxide synthase mediated by transient receptor potential vanilloid type 1.
Cardiovascular research 20110801
-
Cannabinoid receptor agonists potentiate action potential-independent release of GABA in the dentate gyrus through a CB1 receptor-independent mechanism.
The Journal of physiology 20110801
-
TRPV1 agonist piperine but not olvanil enhances glutamatergic spontaneous excitatory transmission in rat spinal substantia gelatinosa neurons.
Biochemical and biophysical research communications 20110715
-
Transient receptor potential (TRP) channels as drug targets for diseases of the digestive system.
Pharmacology & therapeutics 20110701
-
Desensitization of transient receptor potential ankyrin 1 (TRPA1) by the TRP vanilloid 1-selective cannabinoid arachidonoyl-2 chloroethanolamine.
Molecular pharmacology 20110701
-
Oxaliplatin elicits mechanical and cold allodynia in rodents via TRPA1 receptor stimulation.
Pain 20110701
-
Thermosensitive transient receptor potential channels in human corneal epithelial cells.
Journal of cellular physiology 20110701
-
Leukotriene B4 mediates inflammation via TRPV1 in duct obstruction-induced pancreatitis in rats.
Pancreas 20110701
-
Characterization of skin inflammation induced by repeated exposure of toluene, xylene, and formaldehyde in mice.
Environmental toxicology 20110601
-
TRPM8 in mouse sperm detects temperature changes and may influence the acrosome reaction.
Journal of cellular physiology 20110601
-
TRPV1 receptors modulate retinal development.
International journal of developmental neuroscience : the official journal of the International Society for Developmental Neuroscience 20110601
-
The vanilloid capsaicin induces IL-6 secretion in prostate PC-3 cancer cells.
Cytokine 20110601
-
The quaternary lidocaine derivative, QX-314, exerts biphasic effects on transient receptor potential vanilloid subtype 1 channels in vitro.
Anesthesiology 20110601
-
Lafutidine, a unique histamine H2-receptor antagonist, inhibits distention-induced gastric acid secretion through an H2 receptor-independent mechanism.
European journal of pharmacology 20110511
-
The polymodal ion channel transient receptor potential vanilloid 4 modulates calcium flux, spiking rate, and apoptosis of mouse retinal ganglion cells.
The Journal of neuroscience : the official journal of the Society for Neuroscience 20110511
-
Post-ictal analgesia in genetically epilepsy-prone rats is induced by audiogenic seizures and involves cannabinoid receptors in the periaqueductal gray.
Brain research 20110510
-
Acteoside inhibits PMA-induced matrix metalloproteinase-9 expression via CaMK/ERK- and JNK/NF-κB-dependent signaling.
Molecular nutrition & food research 20110501
-
Disruption of the transient receptor potential vanilloid 1 can affect survival, bacterial clearance, and cytokine gene expression during murine sepsis.
Anesthesiology 20110501
-
Characterization of TRPM8-like channels activated by the cooling agent icilin in the macrophage cell line RAW 264.7.
The Journal of membrane biology 20110501
-
Cannabinoid potentiation of glycine receptors contributes to cannabis-induced analgesia.
Nature chemical biology 20110501
-
TRPA1 is required for histamine-independent, Mas-related G protein-coupled receptor-mediated itch.
Nature neuroscience 20110501
-
The hypothermic response to bacterial lipopolysaccharide critically depends on brain CB1, but not CB2 or TRPV1, receptors.
The Journal of physiology 20110501
-
Mechanisms underlying the protective effect of eugenol in rats with acute doxorubicin cardiotoxicity.
Archives of pharmacal research 20110501
-
Melittin activates TRPV1 receptors in primary nociceptive sensory neurons via the phospholipase A2 cascade pathways.
Biochemical and biophysical research communications 20110429
-
Role of transient receptor potential ankyrin subfamily member 1 in pruritus induced by endothelin-1.
Neuroscience letters 20110404
-
Characterization of in vitro metabolism of capsazepine, a vanilloid transient receptor potential channel antagonist, by liquid chromatography quadrupole ion trap mass spectrometry.
Biomedical chromatography : BMC 20110401
-
Inhibitory effect of standardized cannabis sativa extract and its ingredient cannabidiol on rat and human bladder contractility.
Urology 20110401
-
Increased transient receptor potential vanilloid type 1 (TRPV1) signaling in idiopathic overactive bladder urothelial cells.
Neurourology and urodynamics 20110401
-
Human dental pulp fibroblasts express the 'cold-sensing' transient receptor potential channels TRPA1 and TRPM8.
Journal of endodontics 20110401
-
Endocannabinoid 2-arachidonoylglycerol protects neurons against β-amyloid insults.
Neuroscience 20110331
-
NOX3 NADPH oxidase couples transient receptor potential vanilloid 1 to signal transducer and activator of transcription 1-mediated inflammation and hearing loss.
Antioxidants & redox signaling 20110315
-
Atomic force microscopy of microvillous cell surface dynamics at fixed and living alveolar type II cells.
Analytical and bioanalytical chemistry 20110301
-
[Apoptosis inhibition of capsaicin on myocardial ischemia-reperfusion injury in rats].
Sichuan da xue xue bao. Yi xue ban = Journal of Sichuan University. Medical science edition 20110301
-
Effects of acetazolamide on transient K+ currents and action potentials in nodose ganglion neurons of adult rats.
CNS neuroscience & therapeutics 20110201
-
dsRNA-induced expression of thymic stromal lymphopoietin (TSLP) in asthmatic epithelial cells is inhibited by a small airway relaxant.
Pulmonary pharmacology & therapeutics 20110201
-
Hesperidin produces antinociceptive response and synergistic interaction with ketorolac in an arthritic gout-type pain in rats.
Pharmacology, biochemistry, and behavior 20110201
-
Diabetic rats show reduced cardiac-somatic reflex evoked by intrapericardial capsaicin.
European journal of pharmacology 20110125
-
TRPV1 activation is required for hypertonicity-stimulated inflammatory cytokine release in human corneal epithelial cells.
Investigative ophthalmology & visual science 20110101
-
Inhibitory effects of zingerone, a pungent component of Zingiber officinale Roscoe, on colonic motility in rats.
Journal of natural medicines 20110101
-
TRPA1 receptors mediate environmental irritant-induced meningeal vasodilatation.
Pain 20110101
-
TRPV channel expression in human skin and possible role in thermally induced cell death.
Journal of burn care & research : official publication of the American Burn Association 20110101
-
Capsaicin-induced changes in LTP in the lateral amygdala are mediated by TRPV1.
PloS one 20110101
-
Antinociception produced by Thalassia testudinum extract BM-21 is mediated by the inhibition of acid sensing ionic channels by the phenolic compound thalassiolin B.
Molecular pain 20110101
-
Anti-inflammatory and anti-infectious effects of Evodia rutaecarpa (Wuzhuyu) and its major bioactive components.
Chinese medicine 20110101
-
Anandamide capacitates bull spermatozoa through CB1 and TRPV1 activation.
PloS one 20110101
-
Intestinal epithelial stem/progenitor cells are controlled by mucosal afferent nerves.
PloS one 20110101
-
Multimodal assessment of painful peripheral neuropathy induced by chronic oxaliplatin-based chemotherapy in mice.
Molecular pain 20110101
-
Nateglinide stimulates glucagon-like peptide-1 release by human intestinal L cells via a K(ATP) channel-independent mechanism.
Biological & pharmaceutical bulletin 20110101
-
The role of cannabinoids in modulating emotional and non-emotional memory processes in the hippocampus.
Frontiers in behavioral neuroscience 20110101
-
Differential effects of TRPV1 receptor ligands against nicotine-induced depression-like behaviors.
BMC pharmacology 20110101
-
Osmosensitivity of transient receptor potential vanilloid 1 is synergistically enhanced by distinct activating stimuli such as temperature and protons.
PloS one 20110101
-
Capsaicin induces reflex scratching in inflamed skin.
Pharmacology 20110101
-
Anandamide inhibits Theiler's virus induced VCAM-1 in brain endothelial cells and reduces leukocyte transmigration in a model of blood brain barrier by activation of CB(1) receptors.
Journal of neuroinflammation 20110101
-
Hydrogen sulfide and neurogenic inflammation in polymicrobial sepsis: involvement of substance P and ERK-NF-κB signaling.
PloS one 20110101
-
Pharmacological blockade of TRPM8 ion channels alters cold and cold pain responses in mice.
PloS one 20110101
-
Endocannabinoid system and psychiatry: in search of a neurobiological basis for detrimental and potential therapeutic effects.
Frontiers in behavioral neuroscience 20110101
-
Increasing antiproliferative properties of endocannabinoids in N1E-115 neuroblastoma cells through inhibition of their metabolism.
PloS one 20110101
-
Role of the transient receptor potential vanilloid 1 in inflammation and sepsis.
Journal of inflammation research 20110101
-
NF-κB feedback control of JNK1 activation modulates TRPV1-induced increases in IL-6 and IL-8 release by human corneal epithelial cells.
Molecular vision 20110101
-
Acute myocardial ischemia enhances the vanilloid TRPV1 and serotonin 5-HT3 receptor-mediated Bezold-Jarisch reflex in rats.
Pharmacological reports : PR 20110101
-
Evidence for CGRP re-uptake in rat dura mater encephali.
British journal of pharmacology 20101201
-
The proteinase/proteinase-activated receptor-2/transient receptor potential vanilloid-1 cascade impacts pancreatic pain in mice.
Life sciences 20101120
-
The protective effect of capsaicin receptor-mediated genistein postconditioning on gastric ischemia-reperfusion injury in rats.
Digestive diseases and sciences 20101101
-
Mechanosensitive transient receptor potential vanilloid type 1 channels contribute to vascular remodeling of rat fistula veins.
Journal of vascular surgery 20101101
-
Signaling mechanisms involved in the intestinal pro-secretory actions of hydrogen sulfide.
Neurogastroenterology and motility : the official journal of the European Gastrointestinal Motility Society 20101101
-
Effects of capsazepine, a transient receptor potential vanilloid type 1 antagonist, on morphine-induced antinociception, tolerance, and dependence in mice.
British journal of anaesthesia 20101101
-
Phosphorylation of ERK in the spinal dorsal horn following pancreatic pronociceptive stimuli with proteinase-activated receptor-2 agonists and hydrogen sulfide in rats: evidence for involvement of distinct mechanisms.
Journal of neuroscience research 20101101
-
Transient receptor potential vanilloid type-1 (TRPV-1) channels contribute to cutaneous thermal hyperaemia in humans.
The Journal of physiology 20101101
-
TRPV1 receptors are involved in protein nitration and Müller cell reaction in the acutely axotomized rat retina.
Experimental eye research 20101101
-
Calcitonin gene-related peptide inhibits angiotensin II-induced endothelial progenitor cells senescence through up-regulation of klotho expression.
Atherosclerosis 20101101
-
Synthesis and SAR studies of 1,4-benzoxazine MenB inhibitors: novel antibacterial agents against Mycobacterium tuberculosis.
Bioorganic & medicinal chemistry letters 20101101
-
Endocannabinoid-dependent LTD in a nociceptive synapse requires activation of a presynaptic TRPV-like receptor.
Journal of neurophysiology 20101101
-
Bring on the heat: transient receptor potential vanilloid type-1 (TRPV-1) channels as a sensory link for local thermal hyperaemia.
The Journal of physiology 20101101
-
Mechanisms involved in the gastroprotective activity of esculin on acute gastric lesions in mice.
Chemico-biological interactions 20101006
-
Ginsenoside Rb1 and paeoniflorin inhibit transient receptor potential vanilloid-1-activated IL-8 and PGE₂ production in a human keratinocyte cell line HaCaT.
International immunopharmacology 20101001
-
Modulation of single-channel properties of TRPV1 by phosphorylation.
The Journal of physiology 20101001
-
Cardio-respiratory reflexes evoked by phenylbiguanide in rats involve vagal afferents which are not sensitive to capsaicin.
Acta physiologica (Oxford, England) 20100901
-
Existence and distinction of acid-evoked currents in rat astrocytes.
Glia 20100901
-
Epidermal growth factor receptor transactivation by the cannabinoid receptor (CB1) and transient receptor potential vanilloid 1 (TRPV1) induces differential responses in corneal epithelial cells.
Experimental eye research 20100901
-
Potentiation of the glutamatergic synaptic input to rat locus coeruleus neurons by P2X7 receptors.
Purinergic signalling 20100901
-
Cannabinoid receptors as target for treatment of osteoporosis: a tale of two therapies.
Current neuropharmacology 20100901
-
Axon reflexes evoked by transient receptor potential vanilloid 1 activation are mediated by tetrodotoxin-resistant voltage-gated Na+ channels in intestinal afferent nerves.
The Journal of pharmacology and experimental therapeutics 20100801
-
Role of TRPV1 channels in boar spermatozoa acquisition of fertilizing ability.
Molecular and cellular endocrinology 20100729
-
1-Nitro-2-phenylethane, the main constituent of the essential oil of Aniba canelilla, elicits a vago-vagal bradycardiac and depressor reflex in normotensive rats.
European journal of pharmacology 20100725
-
Screening of OATP1B1/3 and OCT1 inhibitors in cryopreserved hepatocytes in suspension.
European journal of pharmaceutical sciences : official journal of the European Federation for Pharmaceutical Sciences 20100711
-
Activation of phosphatidylinositol-linked D1-like receptors increases spontaneous glutamate release in rat somatosensory cortical neurons in vitro.
Brain research 20100709
-
Functional vanilloid receptor-1 in human submandibular glands.
Journal of dental research 20100701
-
Regulation of inflammatory pain by inhibition of fatty acid amide hydrolase.
The Journal of pharmacology and experimental therapeutics 20100701
-
The role of capsaicin in spontaneous pacemaking activity in gastrointestinal tract.
Journal of neurogastroenterology and motility 20100701
-
Capsaicin inhibits the spontaneous pacemaker activity in interstitial cells of cajal from the small intestine of mouse.
Journal of neurogastroenterology and motility 20100701
-
17-Beta-estradiol enhanced allodynia of inflammatory temporomandibular joint through upregulation of hippocampal TRPV1 in ovariectomized rats.
The Journal of neuroscience : the official journal of the Society for Neuroscience 20100630
-
Role of sensory C fibers in hypoxia/reoxygenation-impaired myogenic constriction of cerebral arteries.
Neurological research 20100601
-
The dual fatty acid amide hydrolase/TRPV1 blocker, N-arachidonoyl-serotonin, relieves carrageenan-induced inflammation and hyperalgesia in mice.
Pharmacological research 20100601
-
Effects of TRPV1 activation on synaptic excitation in the dentate gyrus of a mouse model of temporal lobe epilepsy.
Experimental neurology 20100601
-
Implementation of a fluorescence-based screening assay identifies histamine H3 receptor antagonists clobenpropit and iodophenpropit as subunit-selective N-methyl-D-aspartate receptor antagonists.
The Journal of pharmacology and experimental therapeutics 20100601
-
Functional roles of TRPV1 channels in lower urinary tract irritated by acetic acid: in vivo evaluations of the sex difference in decerebrate unanesthetized mice.
American journal of physiology. Renal physiology 20100601
-
Nitro-oleic acid inhibits firing and activates TRPV1- and TRPA1-mediated inward currents in dorsal root ganglion neurons from adult male rats.
The Journal of pharmacology and experimental therapeutics 20100601
-
TRPV channels mediate temperature-sensing in human corneal endothelial cells.
Experimental eye research 20100601
-
The nociception induced by glutamate in mice is potentiated by protons released into the solution.
The journal of pain : official journal of the American Pain Society 20100601
-
TRPA1 receptor induced relaxation of the human urethra involves TRPV1 and cannabinoid receptor mediated signals, and cyclooxygenase activation.
The Journal of urology 20100501
-
Accelerated senescence of endothelial progenitor cells in hypertension is related to the reduction of calcitonin gene-related peptide.
Journal of hypertension 20100501
-
In vitro TRPV1 activity of piperine derived amides.
Bioorganic & medicinal chemistry 20100501
-
Resolvins RvE1 and RvD1 attenuate inflammatory pain via central and peripheral actions.
Nature medicine 20100501
-
Opposing effects of cannabinoids and vanilloids on evoked quantal release at the frog neuromuscular junction.
Neuroscience letters 20100405
-
Dietary capsaicin reduces obesity-induced insulin resistance and hepatic steatosis in obese mice fed a high-fat diet.
Obesity (Silver Spring, Md.) 20100401
-
Neuroprotection induced by vitamin E against oxidative stress in hippocampal neurons: involvement of TRPV1 channels.
Molecular nutrition & food research 20100401
-
The TRPV1 ion channel antagonist capsazepine inhibits osteoclast and osteoblast differentiation in vitro and ovariectomy induced bone loss in vivo.
Bone 20100401
-
Direct activation of transient receptor potential V1 by nickel ions.
Pflugers Archiv : European journal of physiology 20100401
-
The TRPv1 receptor is a mediator of the exercise pressor reflex in rats.
The Journal of physiology 20100401
-
Pharmacological characterization of cannabinoid receptor activity in the rat-isolated ileum myenteric plexus-longitudinal muscle preparation.
British journal of pharmacology 20100401
-
Capsaicin mediates cell death in bladder cancer T24 cells through reactive oxygen species production and mitochondrial depolarization.
Urology 20100301
-
Anandamide potentiation of miniature spontaneous excitatory synaptic transmission is mediated via IP3 pathway.
Neurochemistry international 20100301
-
Mechanisms of action of hydrogen sulfide in relaxation of mouse distal colonic smooth muscle.
European journal of pharmacology 20100225
-
[The protective mechanism of N-acetylcysteine against ischemia/reperfusion induced gastric injury in rats].
Sheng li xue bao : [Acta physiologica Sinica] 20100225
-
Behavioral assessment and identification of a molecular marker in a salicylate-induced tinnitus in rats.
Neuroscience 20100217
-
Gastroprotective effect of barbatusin and 3-beta-hydroxy-3-deoxibarbatusin, quinonoid diterpenes isolated from Plectranthus grandis, in ethanol-induced gastric lesions in mice.
Journal of ethnopharmacology 20100217
-
Hydrogen sulfide promotes transient receptor potential vanilloid 1-mediated neurogenic inflammation in polymicrobial sepsis.
Critical care medicine 20100201
-
Pharmacologic antagonism of the oral aversive taste-directed response to capsaicin in a mouse brief access taste aversion assay.
The Journal of pharmacology and experimental therapeutics 20100201
-
Glycolic acid induces keratinocyte proliferation in a skin equivalent model via TRPV1 activation.
Journal of dermatological science 20100201
-
Influence of capsicum extract and capsaicin on endothelial health.
Journal of the Medical Association of Thailand = Chotmaihet thangphaet 20100201
-
TRPV1 gene deficiency attenuates miniature EPSC potentiation induced by mannitol and angiotensin II in supraoptic magnocellular neurons.
The Journal of neuroscience : the official journal of the Society for Neuroscience 20100120
-
Protective effect of anacardic acids from cashew (Anacardium occidentale) on ethanol-induced gastric damage in mice.
Chemico-biological interactions 20100105
-
Amiloride-sensitive channels are a major contributor to mechanotransduction in mammalian muscle spindles.
The Journal of physiology 20100101
-
2-APB and capsazepine-induced Ca2+ influx stimulates clathrin-dependent endocytosis in alveolar epithelial cells.
Cellular physiology and biochemistry : international journal of experimental cellular physiology, biochemistry, and pharmacology 20100101
-
Antinociceptive effect of geranylgeraniol and 6alpha,7beta-dihydroxyvouacapan-17beta-oate methyl ester isolated from Pterodon pubescens Benth.
BMC pharmacology 20100101
-
Anandamide suppresses proliferation and cytokine release from primary human T-lymphocytes mainly via CB2 receptors.
PloS one 20100101
-
Transient Receptor Potential Vanilloid 1 is essential for cisplatin-induced heat hyperalgesia in mice.
Molecular pain 20100101
-
Effects of topical application of alpha-D-glucosylglycerol on dermal levels of insulin-like growth factor-i in mice and on facial skin elasticity in humans.
Bioscience, biotechnology, and biochemistry 20100101
-
'TRPing' synaptic ribbon function in the rat pineal gland: neuroendocrine regulation involves the capsaicin receptor TRPV1.
Neuroendocrinology 20100101
-
Tumor tissue-derived formaldehyde and acidic microenvironment synergistically induce bone cancer pain.
PloS one 20100101
-
Emodin down-regulates expression of TRPV1 mRNA and its function in DRG neurons in vitro.
The American journal of Chinese medicine 20100101
-
Impact of central and peripheral TRPV1 and ROS levels on proinflammatory mediators and nociceptive behavior.
Molecular pain 20100101
-
TRPV1 in brain is involved in acetaminophen-induced antinociception.
PloS one 20100101
-
Moving towards supraspinal TRPV1 receptors for chronic pain relief.
Molecular pain 20100101
-
The M-channel blocker linopirdine is an agonist of the capsaicin receptor TRPV1.
Journal of pharmacological sciences 20100101
-
Involvement of lysophosphatidic acid in bone cancer pain by potentiation of TRPV1 via PKCε pathway in dorsal root ganglion neurons.
Molecular pain 20100101
-
Blocking spinal CCR2 with AZ889 reversed hyperalgesia in a model of neuropathic pain.
Molecular pain 20100101
-
A non-anesthetized mouse model for recording sensory urinary bladder activity.
Frontiers in neurology 20100101
-
Effect of resiniferatoxin on glutamatergic spontaneous excitatory synaptic transmission in substantia gelatinosa neurons of the adult rat spinal cord.
Neuroscience 20091229
-
Characterization of an AM404 analogue, N-(3-hydroxyphenyl)arachidonoylamide, as a substrate and inactivator of prostaglandin endoperoxide synthase.
Biochemistry 20091229
-
Up-regulation of CYP1A1 by rutaecarpine is dependent on aryl hydrocarbon receptor and calcium.
Toxicology 20091221
-
Sex differences in the expression profile of acid-sensing ion channels in the mouse urinary bladder: a possible involvement in irritative bladder symptoms.
BJU international 20091201
-
Anionic linear aliphatic surfactants activate TRPV1: a possible endpoint for estimation of detergent induced eye nociception?
Toxicology in vitro : an international journal published in association with BIBRA 20091201
-
Release of ATP from rat urinary bladder mucosa: role of acid, vanilloids and stretch.
British journal of pharmacology 20091201
-
The cannabinoid R+ methanandamide induces IL-6 secretion by prostate cancer PC3 cells.
Journal of immunotoxicology 20091201
-
Effects of transient receptor potential (TRP) channel agonists and antagonists on slowly adapting type II mechanoreceptors in the rat sinus hair follicle.
Journal of the peripheral nervous system : JPNS 20091201
-
Characterization of a calcitonin gene-related peptide release assay in rat isolated distal colon.
Archives of pharmacal research 20091201
-
Importance of the non-selective cation channel TRPV1 for microglial reactive oxygen species generation.
Journal of neuroimmunology 20091130
-
Evodiamine inhibits adipogenesis via the EGFR-PKCalpha-ERK signaling pathway.
FEBS letters 20091119
-
Evidence for a potential role for TRPV1 receptors in the dorsolateral periaqueductal gray in the attenuation of the anxiolytic effects of cannabinoids.
Progress in neuro-psychopharmacology & biological psychiatry 20091113
-
Non-selective cation channel activity is required for lysophosphatidylcholine-induced monocyte migration.
Journal of cellular physiology 20091101
-
Capsaicin protects mouse neuromuscular junctions from the neuroparalytic effects of botulinum neurotoxin a.
The Journal of pharmacology and experimental therapeutics 20091101
-
Endogenous expression of TRPV1 channel in cultured human melanocytes.
Journal of dermatological science 20091101
-
Do distinct populations of dorsal root ganglion neurons account for the sensory peptidergic innervation of the kidney?
American journal of physiology. Renal physiology 20091101
-
Electrophysiological and morphological properties of neurons in the substantia gelatinosa of the mouse trigeminal subnucleus caudalis.
Pain 20091101
-
Acid-evoked Ca2+ signalling in rat sensory neurones: effects of anoxia and aglycaemia.
Pflugers Archiv : European journal of physiology 20091101
-
Transient receptor potential ankyrin receptor 1 is a novel target for pro-tussive agents.
British journal of pharmacology 20091101
-
Evidence of TRPV1 receptor and PKC signaling pathway in the antinociceptive effect of amyrin octanoate.
Brain research 20091027
-
Mediating roles of the vanilloid receptor TRPV1 in activation of rat primary afferent nociceptive neurons by formaldehyde.
Sheng li xue bao : [Acta physiologica Sinica] 20091025
-
Essential role for TRPV1 in stress-induced (mast cell-dependent) colonic hypersensitivity in maternally separated rats.
Neurogastroenterology and motility : the official journal of the European Gastrointestinal Motility Society 20091001
-
Characterization of the endocannabinoid system in human spermatozoa and involvement of transient receptor potential vanilloid 1 receptor in their fertilizing ability.
Endocrinology 20091001
-
Genetic mapping of targets mediating differential chemical phenotypes in Plasmodium falciparum.
Nature chemical biology 20091001
-
Capsaicin affects brain function in a model of hepatic encephalopathy associated with fulminant hepatic failure in mice.
British journal of pharmacology 20091001
-
Proton acts as a neurotransmitter for nicotine-induced adrenergic and calcitonin gene-related peptide-containing nerve-mediated vasodilation in the rat mesenteric artery.
The Journal of pharmacology and experimental therapeutics 20090901
-
Hydrogen sulfide prevents ethanol-induced gastric damage in mice: role of ATP-sensitive potassium channels and capsaicin-sensitive primary afferent neurons.
The Journal of pharmacology and experimental therapeutics 20090901
-
Blockade of endocannabinoid-degrading enzymes attenuates neuropathic pain.
The Journal of pharmacology and experimental therapeutics 20090901
-
AT(1) receptor blockers increase insulin-like growth factor-I production by stimulating sensory neurons in spontaneously hypertensive rats.
Translational research : the journal of laboratory and clinical medicine 20090901
-
Possible role for TRPV1 in neomycin-induced inhibition of visceral hypersensitivity in rat.
Neurogastroenterology and motility : the official journal of the European Gastrointestinal Motility Society 20090801
-
Anxiolytic-like effects induced by blockade of transient receptor potential vanilloid type 1 (TRPV1) channels in the medial prefrontal cortex of rats.
Psychopharmacology 20090801
-
Activation of TRPV1 and TRPA1 leads to muscle nociception and mechanical hyperalgesia.
Pain 20090801
-
Triggering of transient receptor potential vanilloid type 1 (TRPV1) by capsaicin induces Fas/CD95-mediated apoptosis of urothelial cancer cells in an ATM-dependent manner.
Carcinogenesis 20090801
-
N-arachidonyl dopamine sensitizes rat capsaicin-sensitive lung vagal afferents via activation of TRPV1 receptors.
Respiratory physiology & neurobiology 20090731
-
Involvement of increased expression of transient receptor potential melastatin 8 in oxaliplatin-induced cold allodynia in mice.
Neuroscience letters 20090717
-
Mechanotransduction and chemosensitivity of two major classes of bladder afferents with endings in the vicinity to the urothelium.
The Journal of physiology 20090715
-
Role of ET(A) and ET(B) endothelin receptors on endothelin-1-induced potentiation of nociceptive and thermal hyperalgesic responses evoked by capsaicin in rats.
Neuroscience letters 20090703
-
(Endo)cannabinoids mediate different Ca2+ entry mechanisms in human bronchial epithelial cells.
Naunyn-Schmiedeberg's archives of pharmacology 20090701
-
QX-314 produces long-lasting local anesthesia modulated by transient receptor potential vanilloid receptors in mice.
Anesthesiology 20090701
-
Exposure to concentrated coarse air pollution particles causes mild cardiopulmonary effects in healthy young adults.
Environmental health perspectives 20090701
-
Ethanol aggravates itch-related scratching in hairless mice developing atopic dermatitis.
European journal of pharmacology 20090602
-
A novel role for the TRPV1 channel in UV-induced matrix metalloproteinase (MMP)-1 expression in HaCaT cells.
Journal of cellular physiology 20090601
-
Bronchoconstriction induced by hyperventilation with humidified hot air: role of TRPV1-expressing airway afferents.
Journal of applied physiology (Bethesda, Md. : 1985) 20090601
-
Depolarization-induced release of endocannabinoids by murine dorsal motor nucleus of the vagus nerve neurons differentially regulates inhibitory and excitatory neurotransmission.
Neuropharmacology 20090601
-
Transient receptor potential melastatin 8 channel involvement in the regulation of vascular tone.
American journal of physiology. Heart and circulatory physiology 20090601
-
Enhancement of the hypotensive effects of intrathecally injected endocannabinoids by the entourage compound palmitoylethanolamide.
European journal of pharmacology 20090521
-
A transient receptor potential-like channel mediates synaptic transmission in rod bipolar cells.
The Journal of neuroscience : the official journal of the Society for Neuroscience 20090513
-
Transient receptor potential vanilloid type 1 receptor regulates glutamatergic synaptic inputs to the spinothalamic tract neurons of the spinal cord deep dorsal horn.
Neuroscience 20090505
-
Excitation of cutaneous C nociceptors by intraplantar administration of anandamide.
Brain research 20090501
-
Anandamide-induced behavioral disruption through a vanilloid-dependent mechanism in rats.
Psychopharmacology 20090401
-
Sensitization of capsaicin-sensitive lung vagal afferents by anandamide in rats: role of transient receptor potential vanilloid 1 receptors.
Journal of applied physiology (Bethesda, Md. : 1985) 20090401
-
Functional TRP and ASIC-like channels in cultured urothelial cells from the rat.
American journal of physiology. Renal physiology 20090401
-
Mechanisms involved in oleamide-induced vasorelaxation in rat mesenteric resistance arteries.
European journal of pharmacology 20090401
-
Functional type I vanilloid receptor expression by substantia gelatinosa neurons of trigeminal subnucleus caudalis in mice.
Neuroscience letters 20090320
-
Myosin light chain phosphatase activation is involved in the hydrogen sulfide-induced relaxation in mouse gastric fundus.
European journal of pharmacology 20090315
-
Modulation of anxiety-like behaviour by Transient Receptor Potential Vanilloid Type 1 (TRPV1) channels located in the dorsolateral periaqueductal gray.
European neuropsychopharmacology : the journal of the European College of Neuropsychopharmacology 20090301
-
N-acyldopamines control striatal input terminals via novel ligand-gated cation channels.
Neuropharmacology 20090301
-
Functional characterization of nonadrenergic noncholinergic neurotransmitter release via endocannabinoids: an in vitro study in rabbit corpus cavernosum.
The journal of sexual medicine 20090301
-
Deletion of vanilloid receptor (TRPV1) in mice alters behavioral effects of ethanol.
Neuropharmacology 20090301
-
Nociceptive vascular reflexes evoked by scorpion venom modulate cardiorespiratory parameters involving vanilloid receptor 1 in anaesthetised rats.
Neuroscience letters 20090227
-
TRPA1 activation by lidocaine in nerve terminals results in glutamate release increase.
Biochemical and biophysical research communications 20090220
-
Excitatory and inhibitory urinary bladder reflexes induced by stimulation of cervicovaginal capsaicin-sensitive sensory fibers in rats.
Naunyn-Schmiedeberg's archives of pharmacology 20090201
-
Reciprocal changes in vanilloid (TRPV1) and endocannabinoid (CB1) receptors contribute to visceral hyperalgesia in the water avoidance stressed rat.
Gut 20090201
-
Salt intake augments hypotensive effects of transient receptor potential vanilloid 4: functional significance and implication.
Hypertension (Dallas, Tex. : 1979) 20090201
-
Activation of sensory neurons reduces ischemia/reperfusion-induced acute renal injury in rats.
Anesthesiology 20090201
-
Capsaicin-induced glutamate release is implicated in nociceptive processing through activation of ionotropic glutamate receptors and group I metabotropic glutamate receptor in primary afferent fibers.
Journal of pharmacological sciences 20090201
-
Interaction with phosphoinositides confers adaptation onto the TRPV1 pain receptor.
PLoS biology 20090201
-
Differential effects of topically applied formalin and aromatic compounds on neurogenic-mediated microvascular leakage in rat skin.
Toxicology 20090108
-
Capsaicin, a component of red peppers, induces expression of androgen receptor via PI3K and MAPK pathways in prostate LNCaP cells.
FEBS letters 20090105
-
TRPV1 channels facilitate glutamate transmission in the striatum.
Molecular and cellular neurosciences 20090101
-
Divergent effects of anandamide transporter inhibitors with different target selectivity on social play behavior in adolescent rats.
The Journal of pharmacology and experimental therapeutics 20090101
-
Contribution of transient receptor potential vanilloid subtype 1 to the analgesic and antihyperalgesic activity of nefopam in rodents.
Pharmacology 20090101
-
Antiaversive effects of cannabinoids: is the periaqueductal gray involved?
Neural plasticity 20090101
-
Vanilloid receptor antagonists: emerging class of novel anti-inflammatory agents for pain management.
Current pharmaceutical design 20090101
-
Reactive oxygen species mediate TNFR1 increase after TRPV1 activation in mouse DRG neurons.
Molecular pain 20090101
-
TRPM8, a versatile channel in human sperm.
PloS one 20090101
-
Tumor necrosis factor-alpha (TNF-alpha) enhances functional thermal and chemical responses of TRP cation channels in human synoviocytes.
Molecular pain 20090101
-
Selective targeting of TRPV1 expressing sensory nerve terminals in the spinal cord for long lasting analgesia.
PloS one 20090101
-
NMDA receptor subunit expression and PAR2 receptor activation in colospinal afferent neurons (CANs) during inflammation induced visceral hypersensitivity.
Molecular pain 20090101
-
Dynamic regulation of the endocannabinoid system: implications for analgesia.
Molecular pain 20090101
-
Differential role of the menthol-binding residue Y745 in the antagonism of thermally gated TRPM8 channels.
Molecular pain 20090101
-
Polymorphisms in gene encoding TRPV1-receptor involved in pain perception are unrelated to chronic pancreatitis.
BMC gastroenterology 20090101
-
[Modulation of the smooth muscle contractions of the rat vas deferens by TRPM8 channel agonist menthol].
Fiziolohichnyi zhurnal (Kiev, Ukraine : 1994) 20090101
-
TRPV1 stimulation triggers apoptotic cell death of rat cortical neurons.
Biochemical and biophysical research communications 20081226
-
Short interfering RNA against transient receptor potential vanilloid 1 attenuates cisplatin-induced hearing loss in the rat.
The Journal of neuroscience : the official journal of the Society for Neuroscience 20081203
-
CO2 chemosensing in rat oesophagus.
Gut 20081201
-
Facilitation of contextual fear memory extinction and anti-anxiogenic effects of AM404 and cannabidiol in conditioned rats.
European neuropsychopharmacology : the journal of the European College of Neuropsychopharmacology 20081201
-
Virodhamine relaxes the human pulmonary artery through the endothelial cannabinoid receptor and indirectly through a COX product.
British journal of pharmacology 20081201
-
Phosphorylation of TRPV1 by neurokinin-1 receptor agonist exaggerates the capsaicin-mediated substance P release from cultured rat dorsal root ganglion neurons.
Neuropharmacology 20081201
-
Rutaecarpine inhibits hypoxia/reoxygenation-induced apoptosis in rat hippocampal neurons.
Neuropharmacology 20081201
-
Cannabinoids and capsaicin improve liver function following thioacetamide-induced acute injury in mice.
The American journal of gastroenterology 20081201
-
Extracellular signal-regulated kinases mediate melittin-induced hypersensitivity of spinal neurons to chemical and thermal but not mechanical stimuli.
Brain research bulletin 20081125
-
TRPV1 mediates the uterine capsaicin-induced NMDA NR2B-dependent cross-organ reflex sensitization in anesthetized rats.
American journal of physiology. Renal physiology 20081101
-
Characterization of A-425619 at native TRPV1 receptors: a comparison between dorsal root ganglia and trigeminal ganglia.
European journal of pharmacology 20081031
-
Transient receptor potential vanilloid 1-mediated expression and secretion of endothelial cell-derived calcitonin gene-related peptide.
Regulatory peptides 20081009
-
Dependence of regulatory volume decrease on transient receptor potential vanilloid 4 (TRPV4) expression in human corneal epithelial cells.
Cell calcium 20081001
-
Heat-induced MMP-1 expression is mediated by TRPV1 through PKCalpha signaling in HaCaT cells.
Experimental dermatology 20081001
-
Behavioral and electrophysiological evidence for the differential functions of TRPV1 at early and late stages of chronic inflammatory nociception in rats.
Neurochemical research 20081001
-
Calcitonin gene-related peptide-mediated antihypertensive and anti-platelet effects by rutaecarpine in spontaneously hypertensive rats.
Peptides 20081001
-
Transient receptor potential vanilloid subtype 1 channel mediated neuropeptide secretion and depressor effects: role of endoplasmic reticulum associated Ca2+ release receptors in rat dorsal root ganglion neurons.
Journal of hypertension 20081001
-
A TRPV channel modulates C. elegans neurosecretion, larval starvation survival, and adult lifespan.
PLoS genetics 20081001
-
Capsaicin inhibits the in vitro binding of peptides selective for mu- and kappa-opioid, and nociceptin-receptors.
Brain research bulletin 20080930
-
Dorsal root ganglion neurons innervating skeletal muscle respond to physiological combinations of protons, ATP, and lactate mediated by ASIC, P2X, and TRPV1.
Journal of neurophysiology 20080901
-
Estrous cycle variation of TRPV1-mediated cross-organ sensitization between uterus and NMDA-dependent pelvic-urethra reflex activity.
American journal of physiology. Endocrinology and metabolism 20080901
-
Elevated temperatures alter TRPV1 agonist-evoked excitability of dorsal root ganglion neurons.
Inflammation research : official journal of the European Histamine Research Society ... [et al.] 20080901
-
Antistress effect of TRPV1 channel on synaptic plasticity and spatial memory.
Biological psychiatry 20080815
-
A subpopulation of capsaicin-sensitive porcine dorsal root ganglion neurons is lacking hyperpolarization-activated cyclic nucleotide-gated channels.
European journal of pain (London, England) 20080801
-
Effect of topical application of raspberry ketone on dermal production of insulin-like growth factor-I in mice and on hair growth and skin elasticity in humans.
Growth hormone & IGF research : official journal of the Growth Hormone Research Society and the International IGF Research Society 20080801
-
Role of TRPV1 channels in renal haemodynamics and function in Dahl salt-sensitive hypertensive rats.
Experimental physiology 20080801
-
Involvement of TRPV1 in nociceptive behavior in a rat model of cancer pain.
The journal of pain : official journal of the American Pain Society 20080801
-
Dual effect of anandamide on rat placenta nitric oxide synthesis.
Placenta 20080801
-
SA13353 (1-[2-(1-Adamantyl)ethyl]-1-pentyl-3-[3-(4-pyridyl)propyl]urea) inhibits TNF-alpha production through the activation of capsaicin-sensitive afferent neurons mediated via transient receptor potential vanilloid 1 in vivo.
European journal of pharmacology 20080707
-
Sustained increase of Ca+2 oscillations after chronic TRPV1 receptor activation with capsaicin in cultured spinal neurons.
Brain research 20080707
-
Therapeutic potential of 1-methylnicotinamide against acute gastric lesions induced by stress: role of endogenous prostacyclin and sensory nerves.
The Journal of pharmacology and experimental therapeutics 20080701
-
In vivo pharmacological evaluation of compound 48/80-induced airways oedema by MRI.
British journal of pharmacology 20080701
-
Cigarette smoke-induced neurogenic inflammation is mediated by alpha,beta-unsaturated aldehydes and the TRPA1 receptor in rodents.
The Journal of clinical investigation 20080701
-
Gastroprotective mechanisms of centipedic acid, a natural diterpene from Egletes viscosa LESS.
Biological & pharmaceutical bulletin 20080701
-
Attenuation of anxiety-related behaviour after the antagonism of transient receptor potential vanilloid type 1 channels in the rat ventral hippocampus.
Behavioural pharmacology 20080701
-
[Protective effect of capsaicin on against myocardial ischemia-reperfusion injury of rat in vivo].
Sichuan da xue xue bao. Yi xue ban = Journal of Sichuan University. Medical science edition 20080701
-
Gastroprotective action of orexin-A against stress-induced gastric damage is mediated by endogenous prostaglandins, sensory afferent neuropeptides and nitric oxide.
Regulatory peptides 20080605
-
The activation of transient receptor potential vanilloid receptor subtype 1 by capsaicin without extracellular Ca2+ is involved in the mechanism of distinct substance P release in cultured rat dorsal root ganglion neurons.
Naunyn-Schmiedeberg's archives of pharmacology 20080601
-
Interdependent regulation of afferent renal nerve activity and renal function: role of transient receptor potential vanilloid type 1, neurokinin 1, and calcitonin gene-related peptide receptors.
The Journal of pharmacology and experimental therapeutics 20080601
-
Impaired capsaicin-induced relaxation of coronary arteries in a porcine model of the metabolic syndrome.
American journal of physiology. Heart and circulatory physiology 20080601
-
Monoacylglycerols activate capsaicin receptor, TRPV1.
Lipids 20080601
-
The analgesic drug, tramadol, acts as an agonist of the transient receptor potential vanilloid-1.
Anesthesia and analgesia 20080601
-
Inflammation reduces mechanical thresholds in a population of transient receptor potential channel A1-expressing nociceptors in the rat.
The European journal of neuroscience 20080601
-
Functional expression of transient receptor potential vanilloid-related channels in chronically hypoxic human pulmonary arterial smooth muscle cells.
The Journal of membrane biology 20080601
-
TRPV1: a target for next generation analgesics.
Current neuropharmacology 20080601
-
TRPV1 mediates cell death in rat synovial fibroblasts through calcium entry-dependent ROS production and mitochondrial depolarization.
Biochemical and biophysical research communications 20080516
-
Quebrachitol-induced gastroprotection against acute gastric lesions: role of prostaglandins, nitric oxide and K+ ATP channels.
Phytomedicine : international journal of phytotherapy and phytopharmacology 20080501
-
The TRPV1 receptor is associated with preferential stress in large dorsal root ganglion neurons in early diabetic sensory neuropathy.
Journal of neurochemistry 20080501
-
Functional study on TRPV1-mediated signalling in the mouse small intestine: involvement of tachykinin receptors.
Neurogastroenterology and motility : the official journal of the European Gastrointestinal Motility Society 20080501
-
TRPV1-mediated protection against endotoxin-induced hypotension and mortality in rats.
American journal of physiology. Regulatory, integrative and comparative physiology 20080501
-
Segmental regulation of sodium and water excretion by TRPV1 activation in the kidney.
Journal of cardiovascular pharmacology 20080501
-
A saturated N-acylethanolamine other than N-palmitoyl ethanolamine with anti-inflammatory properties: a neglected story..
Journal of neuroendocrinology 20080501
-
Novel gating and sensitizing mechanism of capsaicin receptor (TRPV1): tonic inhibitory regulation of extracellular sodium through the external protonation sites on TRPV1.
The Journal of biological chemistry 20080404
-
Cardiac oxidative stress and electrophysiological changes in rats exposed to concentrated ambient particles are mediated by TRP-dependent pulmonary reflexes.
Toxicological sciences : an official journal of the Society of Toxicology 20080401
-
Pronociceptive response elicited by TRPA1 receptor activation in mice.
Neuroscience 20080318
-
SAR studies of capsazepinoid bronchodilators. Part 2: Chlorination and catechol replacement in the A-ring.
Bioorganic & medicinal chemistry 20080301
-
SAR studies of capsazepinoid bronchodilators. Part 1: The importance of the catechol moiety and aspects of the B-ring structure.
Bioorganic & medicinal chemistry 20080301
-
Effect of increasing temperature on TRPV1-mediated responses in isolated rat pulmonary sensory neurons.
American journal of physiology. Lung cellular and molecular physiology 20080301
-
SAR studies of capsazepinoid bronchodilators 3: The thiourea part (coupling region) and the 2-(4-chlorophenyl)ethyl moiety (C-region).
Bioorganic & medicinal chemistry 20080301
-
Gastroprotective effect of a flavone from Lonchocarpus araripensis Benth. (Leguminosae) and the possible mechanism.
The Journal of pharmacy and pharmacology 20080301
-
Increased GFR and renal excretory function by activation of TRPV1 in the isolated perfused kidney.
Pharmacological research 20080301
-
Lafutidine facilitates calcitonin gene-related peptide (CGRP) nerve-mediated vasodilation via vanilloid-1 receptors in rat mesenteric resistance arteries.
Journal of pharmacological sciences 20080301
-
ThermoTRP channels in nociceptors: taking a lead from capsaicin receptor TRPV1.
Current neuropharmacology 20080301
-
Herbal compounds and toxins modulating TRP channels.
Current neuropharmacology 20080301
-
The role of TRPV1 receptors in the antinociceptive effect of anandamide at spinal level.
Pain 20080201
-
Effect of capsaicin on plasma and tissue levels of insulin-like growth factor-I in spontaneously hypertensive rats.
Growth hormone & IGF research : official journal of the Growth Hormone Research Society and the International IGF Research Society 20080201
-
Transient receptor potential vanilloid type 1 channels act as mechanoreceptors and cause substance P release and sensory activation in rat kidneys.
American journal of physiology. Renal physiology 20080201
-
The vanilloid receptor TRPV1 is activated and sensitized by local anesthetics in rodent sensory neurons.
The Journal of clinical investigation 20080201
-
Partial restoration of mutant enzyme homeostasis in three distinct lysosomal storage disease cell lines by altering calcium homeostasis.
PLoS biology 20080201
-
Involvement of serotonin receptors 5-HT1 and 5-HT2 in 12(S)-HPETE-induced scratching in mice.
European journal of pharmacology 20080128
-
Transient receptor potential vanilloid 1 (TRPV1) channels in cultured rat Sertoli cells regulate an acid sensing chloride channel.
Biochemical pharmacology 20080115
-
Stereospecific high-affinity TRPV1 antagonists: chiral N-(2-benzyl-3-pivaloyloxypropyl) 2-[4-(methylsulfonylamino)phenyl]propionamide analogues.
Journal of medicinal chemistry 20080110
-
Inhibition of cancer cell invasion by cannabinoids via increased expression of tissue inhibitor of matrix metalloproteinases-1.
Journal of the National Cancer Institute 20080102
-
Discovery of a potent and long-acting bronchorelaxing capsazepinoid, RESPIR 4-95.
Pulmonary pharmacology & therapeutics 20080101
-
Control of excitatory synaptic transmission by capsaicin is unaltered in TRPV1 vanilloid receptor knockout mice.
Neurochemistry international 20080101
-
Ethanol causes neurogenic vasodilation by TRPV1 activation and CGRP release in the trigeminovascular system of the guinea pig.
Cephalalgia : an international journal of headache 20080101
-
TRPV1 receptor signaling mediates afferent nerve sensitization during colitis-induced motility disorders in rats.
American journal of physiology. Gastrointestinal and liver physiology 20080101
-
Perineural resiniferatoxin selectively inhibits inflammatory hyperalgesia.
Molecular pain 20080101
-
Molecular and cellular limits to somatosensory specificity.
Molecular pain 20080101
-
PPARgamma and Apoptosis in Cancer.
PPAR research 20080101
-
Histamine-induced itch and its relationship with pain.
Molecular pain 20080101
-
Direct activation of transient receptor potential vanilloid 1(TRPV1) by diacylglycerol (DAG).
Molecular pain 20080101
-
Differential stimulatory effects of cannabinoids on VIP release and NO synthase activity in synaptosomal fractions from rat ileum.
Neuropeptides 20080101
-
Human keratinocytes are vanilloid resistant.
PloS one 20080101
-
Mechanisms involved in an increment of multimodal excitability of medullary and upper cervical dorsal horn neurons following cutaneous capsaicin treatment.
Molecular pain 20080101
-
TRPM8 mechanism of cold allodynia after chronic nerve injury.
The Journal of neuroscience : the official journal of the Society for Neuroscience 20071212
-
Transient receptor potential vanilloid 1 activation induces inflammatory cytokine release in corneal epithelium through MAPK signaling.
Journal of cellular physiology 20071201
-
Anandamide improves the impaired nitric oxide-mediated neurogenic relaxation of the corpus cavernosum in diabetic rats: involvement of cannabinoid CB1 and vanilloid VR1 receptors.
BJU international 20071201
-
Neuroprotective effects of glyceryl nonivamide against microglia-like cells and 6-hydroxydopamine-induced neurotoxicity in SH-SY5Y human dopaminergic neuroblastoma cells.
The Journal of pharmacology and experimental therapeutics 20071201
-
Voltage is a partial activator of rat thermosensitive TRP channels.
The Journal of physiology 20071201
-
Delta9-tetrahydrocannabinol (THC) and AM 404 protect against cerebral ischaemia in gerbils through a mechanism involving cannabinoid and opioid receptors.
British journal of pharmacology 20071201
-
Increased depressor response to N-arachidonoyl-dopamine during high salt intake: role of the TRPV1 receptor.
Journal of hypertension 20071201
-
Cannabinoids in health and disease.
Dialogues in clinical neuroscience 20071201
-
Involvement of peripheral TRPV1 in TMJ hyperalgesia induced by ethanol withdrawal.
Life sciences 20071130
-
Characterization of the vasorelaxant mechanisms of the endocannabinoid anandamide in rat aorta.
British journal of pharmacology 20071101
-
Involvement of a capsaicin-sensitive TRPV1-independent mechanism in lipopolysaccharide-induced fever in chickens.
Comparative biochemistry and physiology. Part A, Molecular & integrative physiology 20071101
-
Delta 9-tetrahydrocannabinol inhibits electrically-evoked CGRP release and capsaicin-sensitive sensory neurogenic vasodilatation in the rat mesenteric arterial bed.
British journal of pharmacology 20071101
-
Anti-dyskinetic effects of cannabinoids in a rat model of Parkinson's disease: role of CB(1) and TRPV1 receptors.
Experimental neurology 20071101
-
Transient receptor potential vanilloid-1 mediates heat-shock-induced matrix metalloproteinase-1 expression in human epidermal keratinocytes.
The Journal of investigative dermatology 20071001
-
Capsaicin-induced avoidance behavior in the terrestrial Gastropoda Megalobulimus abbreviatus: evidence for TRPV-1 signaling and opioid modulation in response to chemical noxious stimuli.
Comparative biochemistry and physiology. Part A, Molecular & integrative physiology 20071001
-
Fatty acyl amides of endogenous tetrahydroisoquinolines are active at the recombinant human TRPV1 receptor.
Bioorganic & medicinal chemistry 20070915
-
Acid-induced modulation of airway basal tone and contractility: role of acid-sensing ion channels (ASICs) and TRPV1 receptor.
Life sciences 20070908
-
12-Lipoxygenase-derived eicosanoids protect against myocardial ischemia/reperfusion injury via activation of neuronal TRPV1.
FASEB journal : official publication of the Federation of American Societies for Experimental Biology 20070901
-
Surfactant-induced TRPV1 activity--a novel mechanism for eye irritation?
Toxicological sciences : an official journal of the Society of Toxicology 20070901
-
TRPV1 gene knockout impairs preconditioning protection against myocardial injury in isolated perfused hearts in mice.
American journal of physiology. Heart and circulatory physiology 20070901
-
Bladder afferent sensitivity in wild-type and TRPV1 knockout mice.
The Journal of physiology 20070901
-
Eugenol inhibits K+ currents in trigeminal ganglion neurons.
Journal of dental research 20070901
-
Hydroxy-alpha-sanshool activates TRPV1 and TRPA1 in sensory neurons.
The European journal of neuroscience 20070901
-
A pharmacological study of slowly adapting mechanoreceptors responsive to cold thermal stimulation.
Neuroscience 20070824
-
4-Hydroxynonenal, an endogenous aldehyde, causes pain and neurogenic inflammation through activation of the irritant receptor TRPA1.
Proceedings of the National Academy of Sciences of the United States of America 20070814
-
Role of capsaicin-sensitive sensory nerves in protease-activated receptor-2-mediated contraction of rat urinary bladder.
European journal of pharmacology 20070813
-
Expression of transient receptor potential vanilloid 1 (TRPV1) in synovial fibroblasts from patients with osteoarthritis and rheumatoid arthritis.
Biochemical and biophysical research communications 20070810
-
Capsaicin-induced apoptosis of glioma cells is mediated by TRPV1 vanilloid receptor and requires p38 MAPK activation.
Journal of neurochemistry 20070801
-
Activation of recombinant human TRPV1 receptors expressed in SH-SY5Y human neuroblastoma cells increases [Ca(2+)](i), initiates neurotransmitter release and promotes delayed cell death.
Journal of neurochemistry 20070801
-
Bradykinin-induced nuclear factor of activated T-cells-dependent transcription in rat dorsal root ganglion neurons.
Molecular pharmacology 20070801
-
Atrial natriuretic peptide reduces ischemia/reperfusion-induced spinal cord injury in rats by enhancing sensory neuron activation.
The Journal of pharmacology and experimental therapeutics 20070801
-
Effects of anandamide and noxious heat on intracellular calcium concentration in nociceptive drg neurons of rats.
Journal of neurophysiology 20070801
-
A potential role for the vanilloid receptor TRPV1 in the therapeutic effect of curcumin in dinitrobenzene sulphonic acid-induced colitis in mice.
Neurogastroenterology and motility : the official journal of the European Gastrointestinal Motility Society 20070801
-
Cannabidiol reduced the striatal atrophy caused 3-nitropropionic acid in vivo by mechanisms independent of the activation of cannabinoid, vanilloid TRPV1 and adenosine A2A receptors.
The European journal of neuroscience 20070801
-
A novel function of capsaicin-sensitive TRPV1 channels: involvement in cell migration.
Cell calcium 20070701
-
The synthetic cannabinoids attenuate allodynia and hyperalgesia in a rat model of trigeminal neuropathic pain.
Neuropharmacology 20070701
-
Involvement of the endocannabinoid system in retinal damage after high intraocular pressure-induced ischemia in rats.
Investigative ophthalmology & visual science 20070701
-
Preserving cardiac output with beta-adrenergic receptor blockade and inhibiting the Bezold-Jarisch reflex during resuscitation from hemorrhage.
The Journal of trauma 20070701
-
The anandamide transport inhibitor AM404 reduces ethanol self-administration.
The European journal of neuroscience 20070701
-
AM404 decreases Fos-immunoreactivity in the spinal cord in a model of inflammatory pain.
Brain research 20070604
-
Transient receptor potential vanilloid 1 antagonist, capsazepine, improves survival in a rat hemorrhagic shock model.
Annals of surgery 20070601
-
The potential of transient receptor potential vanilloid type 1 channel modulators for the treatment of pain.
Journal of medicinal chemistry 20070531
-
Novel agonistic action of mustard oil on recombinant and endogenous porcine transient receptor potential V1 (pTRPV1) channels.
Biochemical pharmacology 20070515
-
Mouse colon sensory neurons detect extracellular acidosis via TRPV1.
American journal of physiology. Cell physiology 20070501
-
Endocannabinoid regulates blood pressure via activation of the transient receptor potential vanilloid type 1 in Wistar rats fed a high-salt diet.
The Journal of pharmacology and experimental therapeutics 20070501
-
Antinociceptive pharmacology of N-(4-chlorobenzyl)-N'-(4-hydroxy-3-iodo-5-methoxybenzyl) thiourea, a high-affinity competitive antagonist of the transient receptor potential vanilloid 1 receptor.
The Journal of pharmacology and experimental therapeutics 20070501
-
Cannabinoid and vanilloid effects of R(+)-methanandamide in the hemisected meningeal preparation.
Cephalalgia : an international journal of headache 20070501
-
Activation of TRPA1 channel facilitates excitatory synaptic transmission in substantia gelatinosa neurons of the adult rat spinal cord.
The Journal of neuroscience : the official journal of the Society for Neuroscience 20070418
-
Capsicum ethanol extracts and capsaicin enhance interleukin-2 and interferon-gamma production in cultured murine Peyer's patch cells ex vivo.
Life sciences 20070403
-
Capsaicin induces the production of IL-6 in human upper respiratory epithelial cells.
Life sciences 20070403
-
Involvement of endothelial cell-derived CGRP in heat stress-induced protection of endothelial function.
Vascular pharmacology 20070401
-
The endogenous cannabinoid anandamide produces delta-9-tetrahydrocannabinol-like discriminative and neurochemical effects that are enhanced by inhibition of fatty acid amide hydrolase but not by inhibition of anandamide transport.
The Journal of pharmacology and experimental therapeutics 20070401
-
Heat sensitization in skin and muscle nociceptors expressing distinct combinations of TRPV1 and TRPV2 protein.
Journal of neurophysiology 20070401
-
Capsaicin-induced mucus secretion in rat airways assessed in vivo and non-invasively by magnetic resonance imaging.
British journal of pharmacology 20070401
-
The preventive effect of Daikenchuto on postoperative adhesion-induced intestinal obstruction in rats.
Inflammopharmacology 20070401
-
Pharmacological characterization of receptor types mediating the dilator action of anandamide on blood vessels of the rat knee joint.
Life sciences 20070327
-
Vanilloid receptor agonists and antagonists are mitochondrial inhibitors: how vanilloids cause non-vanilloid receptor mediated cell death.
Biochemical and biophysical research communications 20070302
-
Analgesic actions of N-arachidonoyl-serotonin, a fatty acid amide hydrolase inhibitor with antagonistic activity at vanilloid TRPV1 receptors.
British journal of pharmacology 20070301
-
Pharmacological characterisation of capsaicin-induced relaxations in human and porcine isolated arteries.
Naunyn-Schmiedeberg's archives of pharmacology 20070301
-
TRPV1 mediates histamine-induced itching via the activation of phospholipase A2 and 12-lipoxygenase.
The Journal of neuroscience : the official journal of the Society for Neuroscience 20070227
-
The non-psychoactive cannabis constituent cannabidiol is an orally effective therapeutic agent in rat chronic inflammatory and neuropathic pain.
European journal of pharmacology 20070205
-
Inhibition of neutrophil activation by lafutidine, an H2-receptor antagonist, through enhancement of sensory neuron activation contributes to the reduction of stress-induced gastric mucosal injury in rats.
Digestive diseases and sciences 20070201
-
Vanilloid (subtype 1) receptor-modulatory drugs inhibit [3H]batrachotoxinin-A 20-alpha-benzoate binding to Na+ channels.
Basic & clinical pharmacology & toxicology 20070201
-
TRPV1 is a novel target for omega-3 polyunsaturated fatty acids.
The Journal of physiology 20070115
-
Effects of capsazepine on human small airway responsiveness unravel a novel class of bronchorelaxants.
Pulmonary pharmacology & therapeutics 20070101
-
Cannabinoid (CB1) receptor activation inhibits trigeminovascular neurons.
The Journal of pharmacology and experimental therapeutics 20070101
-
Halogenation of 4-hydroxy-3-methoxybenzyl thiourea TRPV1 agonists showed enhanced antagonism to capsaicin.
Bioorganic & medicinal chemistry letters 20070101
-
Danaparoid sodium reduces ischemia/reperfusion-induced liver injury in rats by attenuating inflammatory responses.
Thrombosis and haemostasis 20070101
-
Animal models of cough: literature review and presentation of a novel cigarette smoke-enhanced cough model in the guinea-pig.
Pulmonary pharmacology & therapeutics 20070101
-
TRPV1 is involved in stretch-evoked contractile changes in the rat autonomous bladder model: a study with piperine, a new TRPV1 agonist.
Neurourology and urodynamics 20070101
-
Transient receptor potential ion channels control thermoregulatory behaviour in reptiles.
PloS one 20070101
-
Anti-calmodulins and tricyclic adjuvants in pain therapy block the TRPV1 channel.
PloS one 20070101
-
TRPV1-mediated diuresis and natriuresis induced by hypertonic saline perfusion of the renal pelvis.
American journal of nephrology 20070101
-
Novel technique for estimating cerebrovascular permeability demonstrates capsazepine protection following ischemia-reperfusion.
Microcirculation (New York, N.Y. : 1994) 20070101
-
Roles of TRPV1 and neuropeptidergic receptors in dorsal root reflex-mediated neurogenic inflammation induced by intradermal injection of capsaicin.
Molecular pain 20070101
-
Species-specific pharmacology of Trichloro(sulfanyl)ethyl benzamides as transient receptor potential ankyrin 1 (TRPA1) antagonists.
Molecular pain 20070101
-
Inhibition of citric acid- and capsaicin-induced cough by novel TRPV-1 antagonist, V112220, in guinea-pig.
Cough (London, England) 20070101
-
Anandamide mediates hyperdynamic circulation in cirrhotic rats via CB(1) and VR(1) receptors.
British journal of pharmacology 20061201
-
Impaired vasodilation in response to perivascular nerve stimulation in mesenteric arteries of TRPV1-null mutant mice.
Journal of hypertension 20061201
-
Synergistic antinociceptive effects of anandamide, an endocannabinoid, and nonsteroidal anti-inflammatory drugs in peripheral tissue: a role for endogenous fatty-acid ethanolamides?
European journal of pharmacology 20061121
-
Role of substance P in hydrogen sulfide-induced pulmonary inflammation in mice.
American journal of physiology. Lung cellular and molecular physiology 20061101
-
TRPV1 receptors and nasal trigeminal chemesthesis.
Chemical senses 20061101
-
Capsaicin inhibits catecholamine secretion and synthesis by blocking Na+ and Ca2+ influx through a vanilloid receptor-independent pathway in bovine adrenal medullary cells.
Naunyn-Schmiedeberg's archives of pharmacology 20061101
-
Differential mechanisms mediating depressor and diuretic effects of anandamide.
Journal of hypertension 20061101
-
Hydrogen sulfide is a novel prosecretory neuromodulator in the Guinea-pig and human colon.
Gastroenterology 20061101
-
Characterization of the vasorelaxation to methanandamide in rat gastric arteries.
Canadian journal of physiology and pharmacology 20061101
-
Transient receptor potential vanilloid subtype 1 mediates microglial cell death in vivo and in vitro via Ca2+-mediated mitochondrial damage and cytochrome c release.
Journal of immunology (Baltimore, Md. : 1950) 20061001
-
Eugenol inhibits sodium currents in dental afferent neurons.
Journal of dental research 20061001
-
Thermal sensitivity of isolated vagal pulmonary sensory neurons: role of transient receptor potential vanilloid receptors.
American journal of physiology. Regulatory, integrative and comparative physiology 20060901
-
A role for vanilloid receptor 1 (TRPV1) and endocannabinnoid signalling in the regulation of spontaneous and L-DOPA induced locomotion in normal and reserpine-treated rats.
Neuropharmacology 20060901
-
Effect of anandamide on nonadrenergic noncholinergic-mediated relaxation of rat corpus cavernosum.
European journal of pharmacology 20060821
-
Effect of capsazepine on cytosolic Ca(2+) levels and proliferation of human prostate cancer cells.
Toxicology in vitro : an international journal published in association with BIBRA 20060801
-
Protease-activated receptor-2 activation exaggerates TRPV1-mediated cough in guinea pigs.
Journal of applied physiology (Bethesda, Md. : 1985) 20060801
-
Mediator mechanisms involved in TRPV1 and P2X receptor-mediated, ROS-evoked bradypneic reflex in anesthetized rats.
Journal of applied physiology (Bethesda, Md. : 1985) 20060801
-
Effect of intracochlear perfusion of vanilloids on cochlear neural activity in the guinea pig.
Hearing research 20060801
-
Characterization of acid signaling in rat vagal pulmonary sensory neurons.
American journal of physiology. Lung cellular and molecular physiology 20060701
-
Anandamide administration alone and after inhibition of fatty acid amide hydrolase (FAAH) increases dopamine levels in the nucleus accumbens shell in rats.
Journal of neurochemistry 20060701
-
Carbonic anhydrases and mucosal vanilloid receptors help mediate the hyperemic response to luminal CO2 in rat duodenum.
Gastroenterology 20060701
-
Expression and characteristics of vanilloid receptor 1 in the rabbit submandibular gland.
Biochemical and biophysical research communications 20060623
-
Modulation of neuropathic and inflammatory pain by the endocannabinoid transport inhibitor AM404 [N-(4-hydroxyphenyl)-eicosa-5,8,11,14-tetraenamide].
The Journal of pharmacology and experimental therapeutics 20060601
-
Ethanol dilates coronary arteries and increases coronary flow via transient receptor potential vanilloid 1 and calcitonin gene-related peptide.
Cardiovascular research 20060601
-
Antithrombin reduces endotoxin-induced hypotension by enhancing pulmonary sensory neuron activation in rats.
Thrombosis and haemostasis 20060601
-
Tactile allodynia initiated by local subcutaneous endothelin-1 is prolonged by activation of TRPV-1 receptors.
Experimental biology and medicine (Maywood, N.J.) 20060601
-
Gastro-protective action of lafutidine mediated by capsaicin-sensitive afferent neurons without interaction with TRPV1 and involvement of endogenous prostaglandins.
World journal of gastroenterology 20060521
-
Transient receptor potential vanilloid 1, calcitonin gene-related peptide, and substance P mediate nociception in acute pancreatitis.
American journal of physiology. Gastrointestinal and liver physiology 20060501
-
Microsphere-based protease assays and screening application for lethal factor and factor Xa.
Cytometry. Part A : the journal of the International Society for Analytical Cytology 20060501
-
Caged vanilloid ligands for activation of TRPV1 receptors by 1- and 2-photon excitation.
Biochemistry 20060418
-
Pharmacological characterisation of the plant sesquiterpenes polygodial and drimanial as vanilloid receptor agonists.
Biochemical pharmacology 20060414
-
Cannabidiol reverses MK-801-induced disruption of prepulse inhibition in mice.
Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology 20060401
-
Cannabidiol-induced intracellular Ca2+ elevations in hippocampal cells.
Neuropharmacology 20060401
-
Inhibition of Ih reduces epileptiform activity in rodent hippocampal slices.
Synapse (New York, N.Y.) 20060401
-
Participation of the spinal TRPV1 receptors in formalin-evoked pain transduction: a study using a selective TRPV1 antagonist, iodo-resiniferatoxin.
The Journal of pharmacy and pharmacology 20060401
-
Role of TRPV1 and cannabinoid CB1 receptors in AM 404-evoked hypothermia in rats.
Pharmacology, biochemistry, and behavior 20060401
-
Endocannabinoids activate transient receptor potential vanilloid 1 receptors to reduce hyperdopaminergia-related hyperactivity: therapeutic implications.
Biological psychiatry 20060315
-
A novel mechanism contributing to development of Dahl salt-sensitive hypertension: role of the transient receptor potential vanilloid type 1.
Hypertension (Dallas, Tex. : 1979) 20060301
-
Vanilloid VR1 receptor is involved in rimonabant-induced neuroprotection.
British journal of pharmacology 20060301
-
Role of capsaicin-sensitive sensory nerves in mediation of the cardiovascular effects of the essential oil of croton zehntneri leaves in anaesthetized rats.
Clinical and experimental pharmacology & physiology 20060301
-
Role of cannabinoid receptors in Delta-9-tetrahydrocannabinol suppression of IL-12p40 in mouse bone marrow-derived dendritic cells infected with Legionella pneumophila.
European journal of pharmacology 20060217
-
Vanilloid type 1 receptor and the acid-sensing ion channel mediate acid phosphate activation of muscle afferent nerves in rats.
Journal of applied physiology (Bethesda, Md. : 1985) 20060201
-
Pain behaviors produced by capsaicin: influence of inflammatory mediators and nerve injury.
The journal of pain : official journal of the American Pain Society 20060201
-
Methanandamide hyperpolarizes gastric arteries by stimulation of TRPV1 receptors on perivascular CGRP containing nerves.
Journal of cardiovascular pharmacology 20060201
-
Identification and biological characterization of 6-aryl-7-isopropylquinazolinones as novel TRPV1 antagonists that are effective in models of chronic pain.
Journal of medicinal chemistry 20060126
-
Analgesic effects of capsazepine and resiniferatoxin on bone cancer pain in mice.
Neuroscience letters 20060123
-
Capsaicin-induced, capsazepine-insensitive relaxation of the guinea-pig ileum.
European journal of pharmacology 20060113
-
Mode of action of gingerols and shogaols on 5-HT3 receptors: binding studies, cation uptake by the receptor channel and contraction of isolated guinea-pig ileum.
European journal of pharmacology 20060113
-
Attenuation of acid induced oesophagitis in VR-1 deficient mice.
Gut 20060101
-
TRPV1 antagonists elevate cell surface populations of receptor protein and exacerbate TRPV1-mediated toxicities in human lung epithelial cells.
Toxicological sciences : an official journal of the Society of Toxicology 20060101
-
Activity and expression of the vanilloid receptor 1 (TRPV1) is altered by long-term diabetes in epineurial arterioles of the rat sciatic nerve.
Diabetes/metabolism research and reviews 20060101
-
Facilitation and inhibition by capsaicin of cholinergic neurotransmission in the guinea-pig small intestine.
Naunyn-Schmiedeberg's archives of pharmacology 20060101
-
Stimulation by bradykinin of HCO3- secretion in rat gastroduodenal mucosa.
Medical science monitor : international medical journal of experimental and clinical research 20060101
-
Induction of apoptosis in prostate tumor PC-3 cells and inhibition of xenograft prostate tumor growth by the vanilloid capsaicin.
Apoptosis : an international journal on programmed cell death 20060101
-
Effects of bee venom peptidergic components on rat pain-related behaviors and inflammation.
Neuroscience 20060101
-
Depression of presynaptic excitation by the activation of vanilloid receptor 1 in the rat spinal dorsal horn revealed by optical imaging.
Molecular pain 20060101
-
Effect of N-arachidonoyl-(2-methyl-4-hydroxyphenyl) amine (VDM11), an anandamide transporter inhibitor, on capsaicin-induced cough in mice.
Cough (London, England) 20060101
-
Capsaicin-resistant arterial baroreceptors.
Journal of negative results in biomedicine 20060101
-
Spinal afferent neurons projecting to the rat lung and pleura express acid sensitive channels.
Respiratory research 20060101
-
The mu opioid agonist morphine modulates potentiation of capsaicin-evoked TRPV1 responses through a cyclic AMP-dependent protein kinase A pathway.
Molecular pain 20060101
-
TRPV1 antagonists attenuate antigen-provoked cough in ovalbumin sensitized guinea pigs.
Cough (London, England) 20060101
-
A nonpungent component of steamed ginger--[10]-shogaol--increases adrenaline secretion via the activation of TRPV1.
Nutritional neuroscience 20060101
-
Recent advances in basic neurosciences and brain disease: from synapses to behavior.
Molecular pain 20060101
-
Molecular cloning, functional characterization of the porcine transient receptor potential V1 (pTRPV1) and pharmacological comparison with endogenous pTRPV1.
Biochemical pharmacology 20051219
-
Capsaicin evokes hypothermia independent of cannabinoid CB1 and CB2 receptors.
Brain research 20051214
-
TRPV1 gene knockout impairs postischemic recovery in isolated perfused heart in mice.
Circulation 20051206
-
Synergistic interactions between airway afferent nerve subtypes regulating the cough reflex in guinea-pigs.
The Journal of physiology 20051201
-
The endocannabinoid arachidonyl ethanolamide (anandamide) increases pulmonary arterial pressure via cyclooxygenase-2 products in isolated rabbit lungs.
American journal of physiology. Heart and circulatory physiology 20051201
-
Inhibition of fatty-acid amide hydrolase enhances cannabinoid stress-induced analgesia: sites of action in the dorsolateral periaqueductal gray and rostral ventromedial medulla.
Neuropharmacology 20051201
-
Proton activation does not alter antagonist interaction with the capsaicin-binding pocket of TRPV1.
Molecular pharmacology 20051201
-
The odontoblast as a sensory receptor cell? The expression of TRPV1 (VR-1) channels.
Archives of histology and cytology 20051201
-
TRPV1 desensitisation and endogenous vanilloid involvement in the enhanced analgesia induced by capsaicin in inflamed tissues.
Brain research bulletin 20051130
-
The mechanosensitivity of mouse colon afferent fibers and their sensitization by inflammatory mediators require transient receptor potential vanilloid 1 and acid-sensing ion channel 3.
The Journal of neuroscience : the official journal of the Society for Neuroscience 20051123
-
Anandamide suppression of Na+ currents in rat dorsal root ganglion neurons.
Brain research 20051116
-
Decreased endocannabinoid levels in the brain and beneficial effects of agents activating cannabinoid and/or vanilloid receptors in a rat model of multiple sclerosis.
Neurobiology of disease 20051101
-
Anandamide elicits an acute release of nitric oxide through endothelial TRPV1 receptor activation in the rat arterial mesenteric bed.
The Journal of physiology 20051015
-
Mechanisms underlying capsaicin-stimulated secretion in the stomach: comparison with mucosal acidification.
The Journal of pharmacology and experimental therapeutics 20051001
-
Icilin activates the delta-subunit of the human epithelial Na+ channel.
Molecular pharmacology 20051001
-
TRPV1 activation results in disruption of the blood-brain barrier in the rat.
British journal of pharmacology 20051001
-
Diuresis and natriuresis caused by activation of VR1-positive sensory nerves in renal pelvis of rats.
Hypertension (Dallas, Tex. : 1979) 20051001
-
Inhibitors of fatty acid amide hydrolase reduce carrageenan-induced hind paw inflammation in pentobarbital-treated mice: comparison with indomethacin and possible involvement of cannabinoid receptors.
British journal of pharmacology 20051001
-
Characterization of the endocannabinoid system in boar spermatozoa and implications for sperm capacitation and acrosome reaction.
Journal of cell science 20051001
-
VR1-mediated depressor effects during high-salt intake: role of anandamide.
Hypertension (Dallas, Tex. : 1979) 20051001
-
Cooling-induced contraction of the rat gastric fundus: mediation via transient receptor potential (TRP) cation channel TRPM8 receptor and Rho-kinase activation.
Clinical and experimental pharmacology & physiology 20051001
-
Camphor activates and strongly desensitizes the transient receptor potential vanilloid subtype 1 channel in a vanilloid-independent mechanism.
The Journal of neuroscience : the official journal of the Society for Neuroscience 20050928
-
Analysis of structure-activity relationships for the 'B-region' of N-(4-t-butylbenzyl)-N'-[4-(methylsulfonylamino)benzyl]-thiourea analogues as TRPV1 antagonists.
Bioorganic & medicinal chemistry letters 20050915
-
Analysis of structure-activity relationships for the 'A-region' of N-(4-t-butylbenzyl)-N'-[4-(methylsulfonylamino)benzyl]thiourea analogues as TRPV1 antagonists.
Bioorganic & medicinal chemistry letters 20050915
-
Activation of transient receptor potential vanilloid 1 (TRPV1) by resiniferatoxin.
The Journal of physiology 20050915
-
Effects of the novel TRPV1 receptor antagonist SB366791 in vitro and in vivo in the rat.
Neuroscience letters 20050909
-
Capsaicin regulates voltage-dependent sodium channels by altering lipid bilayer elasticity.
Molecular pharmacology 20050901
-
Type II vanilloid receptor signaling system: one of the possible mechanisms for the rise in asthma cases.
Frontiers in bioscience : a journal and virtual library 20050901
-
Characteristics of propofol-evoked vascular pain in anaesthetized rats.
British journal of anaesthesia 20050901
-
Vascular effects of anandamide and N-acylvanillylamines in the human forearm and skin microcirculation.
British journal of pharmacology 20050901
-
Heat and mechanical hyperalgesia in mice model of cancer pain.
Pain 20050901
-
Multiple types of sensory neurons respond to irritating volatile organic compounds (VOCs): calcium fluorimetry of trigeminal ganglion neurons.
Pain 20050901
-
Mechanisms involved in the nociception produced by peripheral protein kinase c activation in mice.
Pain 20050901
-
Eugenol inhibits calcium currents in dental afferent neurons.
Journal of dental research 20050901
-
Conservation of functional and pharmacological properties in the distantly related temperature sensors TRVP1 and TRPM8.
Molecular pharmacology 20050801
-
Hydrogen sulfide causes vanilloid receptor 1-mediated neurogenic inflammation in the airways.
British journal of pharmacology 20050801
-
Capsazepine, a vanilloid receptor antagonist, inhibits allergen-induced tracheal contraction.
European journal of pharmacology 20050725
-
The taming of capsaicin. Reversal of the vanilloid activity of N-acylvanillamines by aromatic iodination.
Journal of medicinal chemistry 20050714
-
Vanilloid receptor expressed in the sarcoplasmic reticulum of rat skeletal muscle.
Biochemical and biophysical research communications 20050708
-
Pharmacological characterization of the TRPV1 receptor antagonist JYL1421 (SC0030) in vitro and in vivo in the rat.
European journal of pharmacology 20050704
-
A-425619 [1-isoquinolin-5-yl-3-(4-trifluoromethyl-benzyl)-urea], a novel and selective transient receptor potential type V1 receptor antagonist, blocks channel activation by vanilloids, heat, and acid.
The Journal of pharmacology and experimental therapeutics 20050701
-
Characterization of rat transient receptor potential vanilloid 1 receptors lacking the N-glycosylation site N604.
Neuroreport 20050621
-
Sensory transduction of pulmonary reactive oxygen species by capsaicin-sensitive vagal lung afferent fibres in rats.
The Journal of physiology 20050601
-
The effects of Delta9-tetrahydrocannabinol in rat mesenteric vasculature, and its interactions with the endocannabinoid anandamide.
British journal of pharmacology 20050601
-
Peripheral, but not central effects of cannabidiol derivatives: mediation by CB(1) and unidentified receptors.
Neuropharmacology 20050601
-
Evidence that (-)-7-hydroxy-4'-dimethylheptyl-cannabidiol activates a non-CB(1), non-CB(2), non-TRPV1 target in the mouse vas deferens.
Neuropharmacology 20050601
-
Expression of the transient receptor potential vanilloid 1 (TRPV1) in LNCaP and PC-3 prostate cancer cells and in human prostate tissue.
European journal of pharmacology 20050516
-
Hyperthermia increases sensitivity of pulmonary C-fibre afferents in rats.
The Journal of physiology 20050515
-
2-aminoethoxydiphenyl borate stimulates pulmonary C neurons via the activation of TRPV channels.
American journal of physiology. Lung cellular and molecular physiology 20050501
-
Characterization and comparison of recombinant human and rat TRPV1 receptors: effects of exo- and endocannabinoids.
British journal of anaesthesia 20050501
-
Cannabidiol prevents cerebral infarction via a serotonergic 5-hydroxytryptamine1A receptor-dependent mechanism.
Stroke 20050501
-
The protective effects of rutaecarpine on gastric mucosa injury in rats.
Planta medica 20050501
-
Cloning and functional characterization of dog transient receptor potential vanilloid receptor-1 (TRPV1).
European journal of pharmacology 20050418
-
Oleoylethanolamide excites vagal sensory neurones, induces visceral pain and reduces short-term food intake in mice via capsaicin receptor TRPV1.
The Journal of physiology 20050415
-
Differential responses of bladder lumbosacral and thoracolumbar dorsal root ganglion neurons to purinergic agonists, protons, and capsaicin.
The Journal of neuroscience : the official journal of the Society for Neuroscience 20050413
-
Protective effects of Delta(9)-tetrahydrocannabinol against N-methyl-d-aspartate-induced AF5 cell death.
Brain research. Molecular brain research 20050404
-
AMG 9810 [(E)-3-(4-t-butylphenyl)-N-(2,3-dihydrobenzo[b][1,4] dioxin-6-yl)acrylamide], a novel vanilloid receptor 1 (TRPV1) antagonist with antihyperalgesic properties.
The Journal of pharmacology and experimental therapeutics 20050401
-
TRPV1b, a functional human vanilloid receptor splice variant.
Molecular pharmacology 20050401
-
Transient receptor potential vanilloid (TRPV-1) promotes neurogenic inflammation in the pancreas via activation of the neurokinin-1 receptor (NK-1R).
Pancreas 20050401
-
Role of sensory neuron in reduction of endotoxin-induced hypotension in rats.
Critical care medicine 20050401
-
Identification and biological evaluation of 4-(3-trifluoromethylpyridin-2-yl)piperazine-1-carboxylic acid (5-trifluoromethylpyridin-2-yl)amide, a high affinity TRPV1 (VR1) vanilloid receptor antagonist.
Journal of medicinal chemistry 20050324
-
Acid-sensing properties in rat gastric sensory neurons from normal and ulcerated stomach.
The Journal of neuroscience : the official journal of the Society for Neuroscience 20050309
-
Capsazepine, a vanilloid antagonist, abolishes tonic responses induced by 20-HETE on guinea pig airway smooth muscle.
American journal of physiology. Lung cellular and molecular physiology 20050301
-
Capsaicin exhibits neuroprotective effects in a model of transient global cerebral ischemia in Mongolian gerbils.
British journal of pharmacology 20050301
-
Effects of piperine, the pungent component of black pepper, at the human vanilloid receptor (TRPV1).
British journal of pharmacology 20050301
-
CB(1) cannabinoid receptor stimulation modulates transient receptor potential vanilloid receptor 1 activities in calcium influx and substance P Release in cultured rat dorsal root ganglion cells.
Journal of pharmacological sciences 20050301
-
Pharmacological investigation of hydrogen sulfide (H2S) contractile activity in rat detrusor muscle.
European journal of pharmacology 20050221
-
Involvement of CGRP in the inhibitory effect of rutaecarpine on vasoconstriction induced by anaphylaxis in guinea pig.
Regulatory peptides 20050215
-
A biochemical and pharmacological examination of Rhamphiophis oxyrhynchus (Rufous beaked snake) venom.
Toxicon : official journal of the International Society on Toxinology 20050201
-
Vagal selective effects of ruthenium red on the jejunal afferent fibre response to ischaemia in the rat.
Neurogastroenterology and motility : the official journal of the European Gastrointestinal Motility Society 20050201
-
Involvement of peroxynitrite in capsaicin-induced apoptosis of C6 glioma cells.
Neuroscience research 20050201
-
AM404, an inhibitor of anandamide reuptake decreases Fos-immunoreactivity in the spinal cord of neuropathic rats after non-noxious stimulation.
European journal of pharmacology 20050131
-
Evaluation of the anti-emetic potential of anti-migraine drugs to prevent resiniferatoxin-induced emesis in Suncus murinus (house musk shrew).
European journal of pharmacology 20050131
-
Transient receptor potential vanilloid subtype 1 mediates cell death of mesencephalic dopaminergic neurons in vivo and in vitro.
The Journal of neuroscience : the official journal of the Society for Neuroscience 20050119
-
Discovery of potent, orally available vanilloid receptor-1 antagonists. Structure-activity relationship of N-aryl cinnamides.
Journal of medicinal chemistry 20050113
-
Early painful diabetic neuropathy is associated with differential changes in the expression and function of vanilloid receptor 1.
The Journal of biological chemistry 20050107
-
Role of capsaicin-sensitive primary afferent inputs from the masseter muscle in the C1 spinal neurons responding to tooth-pulp stimulation in rats.
Experimental brain research 20050101
-
Contribution of capsaicin-sensitive sensory neurons to antithrombin-induced reduction of ischemia/reperfusion-induced liver injury in rats.
Thrombosis and haemostasis 20050101
-
Lafutidine-induced increase in intracellular ca(2+) concentrations in PC12 and endothelial cells.
Journal of pharmacological sciences 20050101
-
A phospholipase C-dependent intracellular Ca2+ release pathway mediates the capsaicin-induced apoptosis in HepG2 human hepatoma cells.
Archives of pharmacal research 20050101
-
How cold is it? TRPM8 and TRPA1 in the molecular logic of cold sensation.
Molecular pain 20050101
-
Multiple-signaling pathways are involved in the inhibitory effects of galangin on urinary bladder contractility.
Neurourology and urodynamics 20050101
-
Calcium-dependent and independent mechanisms of capsaicin receptor (TRPV1)-mediated cytokine production and cell death in human bronchial epithelial cells.
Journal of biochemical and molecular toxicology 20050101
-
Inflammatory mediators convert anandamide into a potent activator of the vanilloid type 1 transient receptor potential receptor in nociceptive primary sensory neurons.
Neuroscience 20050101
-
Contrasting phenotypes of putative proprioceptive and nociceptive trigeminal neurons innervating jaw muscle in rat.
Molecular pain 20050101
-
Anandamide-evoked activation of vanilloid receptor 1 contributes to the development of bladder hyperreflexia and nociceptive transmission to spinal dorsal horn neurons in cystitis.
The Journal of neuroscience : the official journal of the Society for Neuroscience 20041215
-
Human brain endothelium: coexpression and function of vanilloid and endocannabinoid receptors.
Brain research. Molecular brain research 20041206
-
Expression of vanilloid VR1 receptor in PC12 cells.
Neurochemistry international 20041201
-
Distinct thymocyte subsets express the vanilloid receptor VR1 that mediates capsaicin-induced apoptotic cell death.
Cell death and differentiation 20041201
-
Lipopolysaccharide fever is initiated via a capsaicin-sensitive mechanism independent of the subtype-1 vanilloid receptor.
British journal of pharmacology 20041201
-
Current perspectives on the therapeutic utility of VR1 antagonists.
Current medicinal chemistry 20041201
-
Vanilloid receptor 1 antagonists attenuate disease severity in dextran sulphate sodium-induced colitis in mice.
Neurogastroenterology and motility : the official journal of the European Gastrointestinal Motility Society 20041201
-
Protective effects of evodiamine on myocardial ischemia-reperfusion injury in rats.
Planta medica 20041201
-
Combined determination with functional and morphological studies of origin of nerve fibers expressing transient receptor potential vanilloid 1 in the myenteric plexus of the rat jejunum.
Autonomic neuroscience : basic & clinical 20041130
-
Evidence that TRPM8 is an androgen-dependent Ca2+ channel required for the survival of prostate cancer cells.
Cancer research 20041115
-
Vanilloid receptor TRPV1, sensory C-fibers, and vascular autoregulation: a novel mechanism involved in myogenic constriction.
Circulation research 20041112
-
Cloning and pharmacological characterization of mouse TRPV1.
Neuroscience letters 20041103
-
Muscle pressor reflex: potential role of vanilloid type 1 receptor and acid-sensing ion channel.
Journal of applied physiology (Bethesda, Md. : 1985) 20041101
-
Jejunal afferent nerve sensitivity in wild-type and TRPV1 knockout mice.
The Journal of physiology 20041101
-
Perivascular nerves induce cardiorespiratory reflexes in response to algogens in anaesthetised rats.
Neuroscience research 20041101
-
Inhibition of the vanilloid receptor subtype-1 attenuates TNBS-colitis.
Journal of gastrointestinal surgery : official journal of the Society for Surgery of the Alimentary Tract 20041101
-
Capsazepine is a novel activator of the delta subunit of the human epithelial Na+ channel.
The Journal of biological chemistry 20041022
-
Capsazepine elevates intracellular Ca2+ in human osteosarcoma cells, questioning its selectivity as a vanilloid receptor antagonist.
Life sciences 20041008
-
Characterization of the human HCN1 channel and its inhibition by capsazepine.
British journal of pharmacology 20041001
-
Ischemic preconditioning of remote organs attenuates gastric ischemia-reperfusion injury through involvement of prostaglandins and sensory nerves.
European journal of pharmacology 20040919
-
Stimulation of calcitonin gene-related peptide synthesis and release: mechanisms for a novel antihypertensive drug, rutaecarpine.
Journal of hypertension 20040901
-
Vanilloid TRPV1 receptor mediates the antihyperalgesic effect of the nonpsychoactive cannabinoid, cannabidiol, in a rat model of acute inflammation.
British journal of pharmacology 20040901
-
Antitussive activity of iodo-resiniferatoxin in guinea pigs.
Thorax 20040901
-
Nociceptin inhibits vanilloid TRPV-1-mediated neurosensitization induced by fenoterol in human isolated bronchi.
Naunyn-Schmiedeberg's archives of pharmacology 20040901
-
AM404 enhances the spontaneous release of L-glutamate in a manner sensitive to capsazepine in adult rat substantia gelatinosa neurones.
Brain research 20040827
-
Evodiamine functions as an agonist for the vanilloid receptor TRPV1.
Organic & biomolecular chemistry 20040821
-
Regulation of calcitonin gene-related peptide release from rat trigeminal nucleus caudalis slices in vitro.
Neuroscience letters 20040819
-
Transient receptor potential vanilloid subfamily 1 expressed in pancreatic islet beta cells modulates insulin secretion in rats.
Biochemical and biophysical research communications 20040813
-
Anandamide transport inhibitor AM404 and structurally related compounds inhibit synaptic transmission between rat hippocampal neurons in culture independent of cannabinoid CB1 receptors.
European journal of pharmacology 20040802
-
Functional TRPV4 channels are expressed in human airway smooth muscle cells.
American journal of physiology. Lung cellular and molecular physiology 20040801
-
Vanilloid receptors mediate adrenergic nerve- and CGRP-containing nerve-dependent vasodilation induced by nicotine in rat mesenteric resistance arteries.
British journal of pharmacology 20040801
-
Inhibition by anandamide and synthetic cannabimimetics of the release of [3H]D-aspartate and [3H]GABA from synaptosomes isolated from the rat hippocampus.
Neurochemical research 20040801
-
Anandamide acts as a vasodilator of dural blood vessels in vivo by activating TRPV1 receptors.
British journal of pharmacology 20040801
-
The cannabinomimetic arachidonyl-2-chloroethylamide (ACEA) acts on capsaicin-sensitive TRPV1 receptors but not cannabinoid receptors in rat joints.
British journal of pharmacology 20040801
-
[Functional analysis of acid sensing ion channels].
Nihon shinkei seishin yakurigaku zasshi = Japanese journal of psychopharmacology 20040801
-
Discovery of small molecule antagonists of TRPV1.
Bioorganic & medicinal chemistry letters 20040716
-
TRPV channels and modulation by hepatocyte growth factor/scatter factor in human hepatoblastoma (HepG2) cells.
Cell calcium 20040701
-
The mammalian amiloride-insensitive non-specific salt taste receptor is a vanilloid receptor-1 variant.
The Journal of physiology 20040701
-
TRPV1 and CB(1) receptor-mediated effects of the endovanilloid/endocannabinoid N-arachidonoyl-dopamine on primary afferent fibre and spinal cord neuronal responses in the rat.
The European journal of neuroscience 20040701
-
Inhibitory effect of the antidepressant St. John's wort (hypericum perforatum) on rat bladder contractility in vitro.
Urology 20040701
-
N-isoquinolin-5-yl-N'-aralkyl-urea and -amide antagonists of human vanilloid receptor 1.
Bioorganic & medicinal chemistry letters 20040621
-
Sex-linked differences in the vasorelaxant effects of anandamide in vascular mesenteric beds: role of oestrogens.
European journal of pharmacology 20040616
-
Ethanol causes inflammation in the airways by a neurogenic and TRPV1-dependent mechanism.
The Journal of pharmacology and experimental therapeutics 20040601
-
Effects of TRPV1 receptor antagonists on stimulated iCGRP release from isolated skin of rats and TRPV1 mutant mice.
Pain 20040601
-
Presynaptic cannabinoid CB(1) receptors are involved in the inhibition of the neurogenic vasopressor response during septic shock in pithed rats.
British journal of pharmacology 20040601
-
Vanilloid receptor TRPV1 antagonists as the next generation of painkillers. Are we putting the cart before the horse?
Journal of medicinal chemistry 20040520
-
Purinergic and vanilloid receptor activation releases glutamate from separate cranial afferent terminals in nucleus tractus solitarius.
The Journal of neuroscience : the official journal of the Society for Neuroscience 20040519
-
The analgesic effect induced by capsaicin is enhanced in inflammatory states.
Life sciences 20040514
-
Involvement of vanilloid-like receptors in the effects of anandamide on motor behavior and nigrostriatal dopaminergic activity: in vivo and in vitro evidence.
Brain research 20040508
-
Molecular determinants of vanilloid sensitivity in TRPV1.
The Journal of biological chemistry 20040507
-
Histamine-induced Ca(2+) influx via the PLA(2)/lipoxygenase/TRPV1 pathway in rat sensory neurons.
Neuroscience letters 20040506
-
Activation of capsaicin-sensitive sensory neurons by carvedilol, a nonselective beta-blocker, in spontaneous hypertensive rats.
The Journal of pharmacology and experimental therapeutics 20040501
-
Activation of protein kinase C reverses capsaicin-induced calcium-dependent desensitization of TRPV1 ion channels.
Cell calcium 20040501
-
Cannabinoid receptor-independent actions of the aminoalkylindole WIN 55,212-2 on trigeminal sensory neurons.
British journal of pharmacology 20040501
-
Identification of species-specific determinants of the action of the antagonist capsazepine and the agonist PPAHV on TRPV1.
The Journal of biological chemistry 20040423
-
Inhibitory effect of ginger (Zingiber officinale) on rat ileal motility in vitro.
Life sciences 20040423
-
N-4-methansulfonamidobenzyl-N'-2-substituted-4-tert-butyl-benzyl thioureas as potent vanilloid receptor antagonistic ligands.
Bioorganic & medicinal chemistry letters 20040405
-
Chain-branched 1,3-dibenzylthioureas as vanilloid receptor 1 antagonists.
Bioorganic & medicinal chemistry letters 20040405
-
Modulation of trigeminal sensory neuron activity by the dual cannabinoid-vanilloid agonists anandamide, N-arachidonoyl-dopamine and arachidonyl-2-chloroethylamide.
British journal of pharmacology 20040401
-
Multiple actions of anandamide on neonatal rat cultured sensory neurones.
British journal of pharmacology 20040401
-
Protective role of vanilloid receptor type 1 in HCl-induced gastric mucosal lesions in rats.
Scandinavian journal of gastroenterology 20040401
-
Characterization of capsaicin-induced, capsazepine-insensitive relaxation of ileal smooth muscle of rats.
European journal of pharmacology 20040308
-
Antitumor effects of cannabidiol, a nonpsychoactive cannabinoid, on human glioma cell lines.
The Journal of pharmacology and experimental therapeutics 20040301
-
TRPV1 receptors mediate particulate matter-induced apoptosis.
American journal of physiology. Lung cellular and molecular physiology 20040301
-
Effects of the vanilloid agonist olvanil and antagonist capsazepine on rat behaviors.
Progress in neuro-psychopharmacology & biological psychiatry 20040301
-
Characterisation of the vasorelaxant properties of the novel endocannabinoid N-arachidonoyl-dopamine (NADA).
British journal of pharmacology 20040301
-
Contribution of vanilloid receptors to the overt nociception induced by B2 kinin receptor activation in mice.
British journal of pharmacology 20040301
-
Background potassium channel block and TRPV1 activation contribute to proton depolarization of sensory neurons from humans with neuropathic pain.
The European journal of neuroscience 20040301
-
An efficient parallel synthesis of capsazepine and capsazepine analogs.
Combinatorial chemistry & high throughput screening 20040301
-
An assessment of vascular pain using the flexor reflex in anesthetized rats.
Methods and findings in experimental and clinical pharmacology 20040301
-
N-4-Substituted-benzyl-N'-tert-butylbenzyl thioureas as vanilloid receptor ligands: investigation on the role of methanesulfonamido group in antagonistic activity.
Bioorganic & medicinal chemistry letters 20040209
-
Design of a high-affinity competitive antagonist of the vanilloid receptor selective for the calcium entry-linked receptor population.
Molecular pharmacology 20040201
-
Characterization of the mouse cold-menthol receptor TRPM8 and vanilloid receptor type-1 VR1 using a fluorometric imaging plate reader (FLIPR) assay.
British journal of pharmacology 20040201
-
7-Hydroxynaphthalen-1-yl-urea and -amide antagonists of human vanilloid receptor 1.
Bioorganic & medicinal chemistry letters 20040119
-
N-[4-(methylsulfonylamino)benzyl]thiourea analogues as vanilloid receptor antagonists: analysis of structure-activity relationships for the 'C-Region'.
Bioorganic & medicinal chemistry 20040115
-
Cannabinoids modulate neuronal firing in the rat basolateral amygdala: evidence for CB1- and non-CB1-mediated actions.
Neuropharmacology 20040101
-
Identification and characterisation of SB-366791, a potent and selective vanilloid receptor (VR1/TRPV1) antagonist.
Neuropharmacology 20040101
-
An investigation of the effects of ruthenium red, nitric oxide and endothelin-1 on infrared receptor activity in a crotaline snake.
Neuroscience 20040101
-
Proton conductance of human transient receptor potential-vanilloid type-1 expressed in oocytes of Xenopus laevis and in Chinese hamster ovary cells.
Neuroscience 20040101
-
Differential pH and capsaicin responses of Griffonia simplicifolia IB4 (IB4)-positive and IB4-negative small sensory neurons.
Neuroscience 20040101
-
Capsaicin, a spicy component of hot pepper, induces apoptosis by activation of the peroxisome proliferator-activated receptor gamma in HT-29 human colon cancer cells.
Journal of medicinal food 20040101
-
Novel non-vanilloid VR1 antagonist of high analgesic effects and its structural requirement for VR1 antagonistic effects.
Bioorganic & medicinal chemistry letters 20031215
-
Contribution of capsaicin-sensitive sensory neurons to stress-induced increases in gastric tissue levels of prostaglandins in rats.
American journal of physiology. Gastrointestinal and liver physiology 20031201
-
A novel neuroimmune mechanism in cannabinoid-mediated attenuation of nerve growth factor-induced hyperalgesia.
Anesthesiology 20031201
-
The endogenous cannabinoid, anandamide, activates the hypothalamo-pituitary-adrenal axis in CB1 cannabinoid receptor knockout mice.
Neuroendocrinology 20031201
-
Capsazepine protects against neuronal injury caused by oxygen glucose deprivation by inhibiting I(h).
The Journal of neuroscience : the official journal of the Society for Neuroscience 20031105
-
Capsaicin-sensitive neurogenic sensory vasodilatation in the dura mater of the rat.
The Journal of physiology 20031101
-
Signal transduction for inhibition of inducible nitric oxide synthase and cyclooxygenase-2 induction by capsaicin and related analogs in macrophages.
British journal of pharmacology 20031101
-
Insulin induces cobalt uptake in a subpopulation of rat cultured primary sensory neurons.
The European journal of neuroscience 20031101
-
Thermal properties of acid-induced depolarization in cultured rat small primary afferent neurons.
Neuroscience letters 20031023
-
4-(2-pyridyl)piperazine-1-carboxamides: potent vanilloid receptor 1 antagonists.
Bioorganic & medicinal chemistry letters 20031020
-
Capsaicin infused into the PAG affects rat tail flick responses to noxious heat and alters neuronal firing in the RVM.
Journal of neurophysiology 20031001
-
Hypotensive effect of anandamide through the activation of CB1 and VR1 spinal receptors in urethane-anesthetized rats.
Naunyn-Schmiedeberg's archives of pharmacology 20031001
-
A novel capsaicin derivative VOA induced relaxation in rat mesenteric and aortic arteries: involvement of CGRP, NO, cGMP, and endothelium-dependent activities.
Journal of cardiovascular pharmacology 20031001
-
Activation of vanilloid receptor 1 (VR1) by eugenol.
Journal of dental research 20031001
-
Vanilloid type 1 receptors (VR1) on trigeminal sensory nerve fibres play a minor role in neurogenic dural vasodilatation, and are involved in capsaicin-induced dural dilation.
British journal of pharmacology 20031001
-
Vanilloid receptor activation by 2- and 10-microm particles induces responses leading to apoptosis in human airway epithelial cells.
Toxicology and applied pharmacology 20031001
-
Cannabinoids inhibit the release of [3H]glutamate from rodent hippocampal synaptosomes via a novel CB1 receptor-independent action.
The European journal of neuroscience 20031001
-
Expression of vanilloid receptors in rat gastric epithelial cells: role in cellular protection.
Biochemical pharmacology 20030915
-
Inhibition of C6 glioma cell proliferation by anandamide, 1-arachidonoylglycerol, and by a water soluble phosphate ester of anandamide: variability in response and involvement of arachidonic acid.
Biochemical pharmacology 20030901
-
An endogenous cannabinoid tone attenuates cholera toxin-induced fluid accumulation in mice.
Gastroenterology 20030901
-
Stimulation by capsaicin of duodenal HCO3(-) secretion via afferent neurons and vanilloid receptors in rats: comparison with acid-induced HCO3(-) response.
Digestive diseases and sciences 20030901
-
Capsaicin-like effects of N-arachidonoyl-dopamine in the isolated guinea pig bronchi and urinary bladder.
European journal of pharmacology 20030815
-
Halogenation of a capsaicin analogue leads to novel vanilloid TRPV1 receptor antagonists.
British journal of pharmacology 20030802
-
Increased expression of vanilloid receptor 1 on myelinated primary afferent neurons contributes to the antihyperalgesic effect of capsaicin cream in diabetic neuropathic pain in mice.
The Journal of pharmacology and experimental therapeutics 20030801
-
Function and regulation of the vanilloid receptor in rats fed a high salt diet.
Journal of hypertension 20030801
-
Involvement of vanilloid receptors in heat stress-induced delayed protection against myocardial ischemia-reperfusion injury.
Neuropeptides 20030801
-
Mechanisms of sensitization of the response of single dorsal root ganglion cells from adult rat to noxious heat.
The European journal of neuroscience 20030801
-
Proton-induced calcitonin gene-related peptide release from rat sciatic nerve axons, in vitro, involving TRPV1.
The European journal of neuroscience 20030801
-
Modifications of capsaicin-sensitive neurons in isolated guinea pig ileum by [6]-gingerol and lafutidine.
Journal of pharmacological sciences 20030801
-
Albaconol from the mushroom Albatrellus confluens induces contraction and desensitization in guinea pig trachea.
Planta medica 20030801
-
N-(3-acyloxy-2-benzylpropyl)-N'-[4-(methylsulfonylamino)benzyl]thiourea analogues: novel potent and high affinity antagonists and partial antagonists of the vanilloid receptor.
Journal of medicinal chemistry 20030703
-
Vanilloid receptors in hearing: altered cochlear sensitivity by vanilloids and expression of TRPV1 in the organ of corti.
Journal of neurophysiology 20030701
-
N-(4-Tertiarybutylphenyl)-4-(3-cholorphyridin-2-yl)tetrahydropyrazine -1(2H)-carbox-amide (BCTC), a novel, orally effective vanilloid receptor 1 antagonist with analgesic properties: II. in vivo characterization in rat models of inflammatory and neuropathic pain.
The Journal of pharmacology and experimental therapeutics 20030701
-
N-(4-tertiarybutylphenyl)-4-(3-chloropyridin-2-yl)tetrahydropyrazine -1(2H)-carbox-amide (BCTC), a novel, orally effective vanilloid receptor 1 antagonist with analgesic properties: I. in vitro characterization and pharmacokinetic properties.
The Journal of pharmacology and experimental therapeutics 20030701
-
New evidence on the mechanisms underlying bradykinin-mediated contraction of the pig iris sphincter in vitro.
Peptides 20030701
-
Involvement of capsaicin-sensitive sensory nerves in cardioprotection of rutaecarpine in rats.
Regulatory peptides 20030615
-
Calcium signaling in single peripheral sensory nerve terminals.
The Journal of neuroscience : the official journal of the Society for Neuroscience 20030615
-
The effects of local and intravenous anesthetics on recombinant rat VR1 vanilloid receptors.
Anesthesia and analgesia 20030601
-
Electrostatic charge activates inflammatory vanilloid (VR1) receptors.
Neurotoxicology 20030601
-
Adrenergic regulation of capsaicin-sensitive neurons in dental pulp.
Journal of endodontics 20030601
-
Anandamide induces cell death independently of cannabinoid receptors or vanilloid receptor 1: possible involvement of lipid rafts.
Cellular and molecular life sciences : CMLS 20030601
-
Inhibitory effect of the plant flavonoid galangin on rat vas deferens in vitro.
Life sciences 20030516
-
Neuroprotection by the endogenous cannabinoid anandamide and arvanil against in vivo excitotoxicity in the rat: role of vanilloid receptors and lipoxygenases.
The Journal of neuroscience : the official journal of the Society for Neuroscience 20030515
-
Chain-branched acyclic phenethylthiocarbamates as vanilloid receptor antagonists.
Bioorganic & medicinal chemistry letters 20030505
-
Vanilloid receptor-1 containing primary sensory neurones mediate dextran sulphate sodium induced colitis in rats.
Gut 20030501
-
Capsaicin-induced reactivation of latent herpes simplex virus type 1 in sensory neurons in culture.
The Journal of general virology 20030501
-
State-dependent phosphorylation of epsilon-isozyme of protein kinase C in adult rat dorsal root ganglia after inflammation and nerve injury.
Journal of neurochemistry 20030501
-
Anandamide induces apoptosis in human endothelial cells: its regulation system and clinical implications.
Thrombosis and haemostasis 20030501
-
Capsaicinoids cause inflammation and epithelial cell death through activation of vanilloid receptors.
Toxicological sciences : an official journal of the Society of Toxicology 20030501
-
The nociceptive and anti-nociceptive effects of evodiamine from fruits of Evodia rutaecarpa in mice.
Planta medica 20030501
-
Peripheral tackykinin and excitatory amino acid receptors mediate hyperalgesia induced by Phoneutria nigriventer venom.
European journal of pharmacology 20030425
-
Impact on the bowel of amtolmetin guacyl, a new gastroprotective non-steroidal anti-inflammatory drug.
European journal of pharmacology 20030425
-
Presynaptic facilitation of glutamatergic synapses to dopaminergic neurons of the rat substantia nigra by endogenous stimulation of vanilloid receptors.
The Journal of neuroscience : the official journal of the Society for Neuroscience 20030415
-
The actions of anandamide on rat superficial medullary dorsal horn neurons in vitro.
The Journal of physiology 20030401
-
Differential effects of intraplantar capsazepine and ruthenium red on capsaicin-induced desensitization in mice.
Pharmacology, biochemistry, and behavior 20030401
-
Capsaicin exhibits anti-inflammatory property by inhibiting IkB-a degradation in LPS-stimulated peritoneal macrophages.
Cellular signalling 20030301
-
Compounds acting at the endocannabinoid and/or endovanilloid systems reduce hyperkinesia in a rat model of Huntington's disease.
Journal of neurochemistry 20030301
-
A role for TRPV1 in bradykinin-induced excitation of vagal airway afferent nerve terminals.
The Journal of pharmacology and experimental therapeutics 20030301
-
Selective ligands and cellular effectors of a G protein-coupled endothelial cannabinoid receptor.
Molecular pharmacology 20030301
-
Anandamide-induced depressor effect in spontaneously hypertensive rats: role of the vanilloid receptor.
Hypertension (Dallas, Tex. : 1979) 20030301
-
Neurogenic responses mediated by vanilloid receptor-1 (TRPV1) are blocked by the high affinity antagonist, iodo-resiniferatoxin.
British journal of pharmacology 20030301
-
Synthesis of N,N',N'-trisubstituted thiourea derivatives and their antagonist effect on the vanilloid receptor.
Bioorganic & medicinal chemistry letters 20030224
-
Effect of arvanil (N-arachidonoyl-vanillyl-amine), a nonpungent anandamide-capsaicin hybrid, on ion currents in NG108-15 neuronal cells.
Biochemical pharmacology 20030215
-
Versatile regulation of cytosolic Ca2+ by vanilloid receptor I in rat dorsal root ganglion neurons.
The Journal of biological chemistry 20030214
-
Endocannabinoids induce ileitis in rats via the capsaicin receptor (VR1).
The Journal of pharmacology and experimental therapeutics 20030201
-
The depressor and vasodilator effects of rutaecarpine are mediated by calcitonin gene-related peptide.
Planta medica 20030201
-
Synthesis of 2-substituted-pyrrolidinethiourea derivatives and their antagonist effect on vanilloid receptor.
Bioorganic & medicinal chemistry letters 20030120
-
Concentration-dependent dual effect of anandamide on sensory neuropeptide release from isolated rat tracheae.
Neuroscience letters 20030116
-
Negatively charged 2- and 10-microm particles activate vanilloid receptors, increase cAMP, and induce cytokine release.
Toxicology and applied pharmacology 20030115
-
R+-methanandamide inhibits tracheal response to endogenously released acetylcholine via capsazepine-sensitive receptors.
European journal of pharmacology 20030110
-
The VR1 antagonist capsazepine reverses mechanical hyperalgesia in models of inflammatory and neuropathic pain.
The Journal of pharmacology and experimental therapeutics 20030101
-
Potentiation of anandamide effects in mesenteric beds isolated from endotoxemic rats.
The Journal of pharmacology and experimental therapeutics 20030101
-
Activation of epidermal vanilloid receptor-1 induces release of proinflammatory mediators in human keratinocytes.
The Journal of pharmacology and experimental therapeutics 20030101
-
Neurokinin release produced by capsaicin acting on the central terminals and axons of primary afferents: relationship with N-methyl-D-aspartate and GABA(B) receptors.
Neuroscience 20030101
-
Functional properties of the high-affinity TRPV1 (VR1) vanilloid receptor antagonist (4-hydroxy-5-iodo-3-methoxyphenylacetate ester) iodo-resiniferatoxin.
The Journal of pharmacology and experimental therapeutics 20021201
-
Comparison of effects of anandamide at recombinant and endogenous rat vanilloid receptors.
British journal of anaesthesia 20021201
-
Effect of olvanil (N-vanillyl-cis-9-octadecenoamide) on cytosolic Ca2+ increase in renal tubular cells.
Life sciences 20021115
-
Upregulation of proinflammatory cytokines and nerve growth factor by intraplantar injection of capsaicin in rats.
The Journal of physiology 20021115
-
Characterization of the vanilloid receptor 1 antagonist iodo-resiniferatoxin on the afferent and efferent function of vagal sensory C-fibers.
The Journal of pharmacology and experimental therapeutics 20021101
-
Gingerols: a novel class of vanilloid receptor (VR1) agonists.
British journal of pharmacology 20021101
-
Anandamide induces cough in conscious guinea-pigs through VR1 receptors.
British journal of pharmacology 20021101
-
Amiloride-blockable acid-sensing ion channels are leading acid sensors expressed in human nociceptors.
The Journal of clinical investigation 20021015
-
High affinity antagonists of the vanilloid receptor.
Molecular pharmacology 20021001
-
Anandamide is a partial agonist at native vanilloid receptors in acutely isolated mouse trigeminal sensory neurons.
British journal of pharmacology 20021001
-
Cellular mechanisms of nociception in the frog.
Journal of neurophysiology 20021001
-
The putative role of vanilloid receptor-like protein-1 in mediating high threshold noxious heat-sensitivity in rat cultured primary sensory neurons.
The European journal of neuroscience 20021001
-
Use of a fluorescent imaging plate reader--based calcium assay to assess pharmacological differences between the human and rat vanilloid receptor.
Journal of biomolecular screening 20021001
-
Effect of piperine, the active ingredient of black pepper, on intestinal secretion in mice.
Life sciences 20020927
-
Protein kinase C(alpha) is required for vanilloid receptor 1 activation. Evidence for multiple signaling pathways.
The Journal of biological chemistry 20020920
-
Vanilloid receptors presynaptically modulate cranial visceral afferent synaptic transmission in nucleus tractus solitarius.
The Journal of neuroscience : the official journal of the Society for Neuroscience 20020915
-
Mechanisms underlying tissue selectivity of anandamide and other vanilloid receptor agonists.
Molecular pharmacology 20020901
-
Characterization of the anandamide induced depolarization of guinea-pig isolated vagus nerve.
British journal of pharmacology 20020901
-
Prostaglandin and protein kinase A-dependent modulation of vanilloid receptor function by metabotropic glutamate receptor 5: potential mechanism for thermal hyperalgesia.
The Journal of neuroscience : the official journal of the Society for Neuroscience 20020901
-
Phosphorylation of extracellular signal-regulated kinase in primary afferent neurons by noxious stimuli and its involvement in peripheral sensitization.
The Journal of neuroscience : the official journal of the Society for Neuroscience 20020901
-
Capsaicin activation of glutamatergic synaptic transmission in the rat locus coeruleus in vitro.
The Journal of physiology 20020901
-
Mechanisms of acid-induced activation of airway afferent nerve fibres in guinea-pig.
The Journal of physiology 20020901
-
Cloning and functional characterization of the guinea pig vanilloid receptor 1.
Neuropharmacology 20020901
-
Pharmacological separation of cannabinoid sensitive receptors on hippocampal excitatory and inhibitory fibers.
Neuropharmacology 20020901
-
Binding, degradation and apoptotic activity of stearoylethanolamide in rat C6 glioma cells.
The Biochemical journal 20020815
-
The cardioprotection of rutaecarpine is mediated by endogenous calcitonin related-gene peptide through activation of vanilloid receptors in guinea-pig hearts.
Planta medica 20020801
-
Effects of peripheral nerve injury on functional spinal VR1 receptors.
Neuroreport 20020702
-
Activation of protein kinase C sensitizes human VR1 to capsaicin and to moderate decreases in pH at physiological temperatures in Xenopus oocytes.
Pain 20020701
-
A heat-sensitive TRP channel expressed in keratinocytes.
Science (New York, N.Y.) 20020614
-
Ethanol elicits and potentiates nociceptor responses via the vanilloid receptor-1.
Nature neuroscience 20020601
-
Anandamide-induced vasorelaxation in rabbit aortic rings has two components: G protein dependent and independent.
American journal of physiology. Heart and circulatory physiology 20020601
-
The arginine-rich hexapeptide R4W2 is a stereoselective antagonist at the vanilloid receptor 1: a Ca2+ imaging study in adult rat dorsal root ganglion neurons.
The Journal of pharmacology and experimental therapeutics 20020601
-
DRASIC contributes to pH-gated currents in large dorsal root ganglion sensory neurons by forming heteromultimeric channels.
Journal of neurophysiology 20020601
-
Capsazepine inhibits thermal hyperalgesia but not nociception triggered by protease-activated receptor-2 in rats.
Japanese journal of pharmacology 20020601
-
Contractile response to a cannabimimetic eicosanoid, 2-arachidonoylglycerol, of longitudinal smooth muscle from the guinea-pig distal colon in vitro.
European journal of pharmacology 20020531
-
Comparison of capsaicin-evoked calcium transients between rat nodose and jugular ganglion neurons.
Autonomic neuroscience : basic & clinical 20020531
-
Spinal administration of capsazepine inhibits noxious evoked responses of dorsal horn neurons in non-inflamed and carrageenan inflamed rats.
Brain research 20020510
-
3-D-QSAR analysis of N-(3-acyloxy-2-benzylpropyl)-N'-dihydroxytetrahydrobenzazepine and tetrahydroisoquinoline and N-(3-acyloxy-2-benzylpropyl)-N'-(4-hydroxy-3-methoxybenzyl) thioureas analogues as potent vanilloid receptor ligands.
Bioorganic & medicinal chemistry 20020501
-
Gastric hyperemic response induced by acid back-diffusion in rat stomachs following barrier disruption -- relation to vanilloid type-1 receptors.
Medical science monitor : international medical journal of experimental and clinical research 20020501
-
Sustained ER Ca2+ depletion suppresses protein synthesis and induces activation-enhanced cell death in mast cells.
The Journal of biological chemistry 20020419
-
Capsazepine partially inhibits neurally mediated gastric mucus secretion following activation of protease-activated receptor 2.
Clinical and experimental pharmacology & physiology 20020401
-
Ischemia/reperfusion-induced increase in the hepatic level of prostacyclin is mainly mediated by activation of capsaicin-sensitive sensory neurons in rats.
The Journal of laboratory and clinical medicine 20020401
-
Interaction between vanilloid and glutamate receptors in the central modulation of nociception.
European journal of pharmacology 20020329
-
Arvanil-induced inhibition of spasticity and persistent pain: evidence for therapeutic sites of action different from the vanilloid VR1 receptor and cannabinoid CB(1)/CB(2) receptors.
European journal of pharmacology 20020329
-
Stimulation of pulmonary vagal C-fibres by anandamide in anaesthetized rats: role of vanilloid type 1 receptors.
The Journal of physiology 20020315
-
Protease-activated receptor-2 activation causes EDHF-like coronary vasodilation: selective preservation in ischemia/reperfusion injury: involvement of lipoxygenase products, VR1 receptors, and C-fibers.
Circulation research 20020308
-
Evidence of a novel site mediating anandamide-induced negative inotropic and coronary vasodilatator responses in rat isolated hearts.
British journal of pharmacology 20020301
-
Relaxant effect of capsazepine in the isolated rat ileum.
Naunyn-Schmiedeberg's archives of pharmacology 20020301
-
Functional vanilloid receptors in cultured normal human epidermal keratinocytes.
Biochemical and biophysical research communications 20020215
-
Particulate matter inflammation and receptor sensitivity are target cell specific.
Inhalation toxicology 20020201
-
Pharmacological characterization of vanilloid receptor located in the brain.
Brain research. Molecular brain research 20020131
-
Simultaneous intracellular calcium and sodium flux imaging in human vanilloid receptor 1 (VR1)-transfected human embryonic kidney cells: a method to resolve ionic dependence of VR1-mediated cell death.
The Journal of pharmacology and experimental therapeutics 20020101
-
Activation of capsaicin receptors on the sciatic nerve induces FOS expression in the spinal dorsal horn of adult rats.
Neuro-Signals 20020101
-
Effects of ginsenosides on vanilloid receptor (VR1) channels expressed in Xenopus oocytes.
Molecules and cells 20011231
-
Acidic stimuli activates two distinct pathways in taste receptor cells from rat fungiform papillae.
Brain research 20011227
-
Inhibition of rat C6 glioma cell proliferation by endogenous and synthetic cannabinoids. Relative involvement of cannabinoid and vanilloid receptors.
The Journal of pharmacology and experimental therapeutics 20011201
-
The endogenous cannabinoid anandamide activates vanilloid receptors in the rat hippocampal slice.
Neuropharmacology 20011201
-
Anandamide and methanandamide induce both vanilloid VR1- and cannabinoid CB1 receptor-mediated changes in heart rate and blood pressure in anaesthetized rats.
Naunyn-Schmiedeberg's archives of pharmacology 20011201
-
Involvement of vanilloid receptor VR1 and prostanoids in the acid-induced writhing responses of mice.
Life sciences 20011102
-
Capsaicin vanilloid receptor-1 mediates substance P release in experimental pancreatitis.
American journal of physiology. Gastrointestinal and liver physiology 20011101
-
Anandamide-induced relaxation of sheep coronary arteries: the role of the vascular endothelium, arachidonic acid metabolites and potassium channels.
British journal of pharmacology 20011101
-
Capsaicin-, resiniferatoxin-, and olvanil-induced adrenaline secretions in rats via the vanilloid receptor.
Bioscience, biotechnology, and biochemistry 20011101
-
Propofol activates vanilloid receptor channels expressed in human embryonic kidney 293 cells.
Neuroscience letters 20011012
-
Stimulatory effect of centrally injected capsaicin, an agonist of vanilloid receptors, on gastric acid secretion in rats.
European journal of pharmacology 20011012
-
Capsaicin inhibits Jurkat T-cell activation by blocking calcium entry current I(CRAC).
The Journal of pharmacology and experimental therapeutics 20011001
-
Pharmacological modulation of monovalent cation currents through the epithelial Ca2+ channel ECaC1.
British journal of pharmacology 20011001
-
Anandamide induces cardiovascular and respiratory reflexes via vasosensory nerves in the anaesthetized rat.
British journal of pharmacology 20011001
-
Molecular targets for cannabidiol and its synthetic analogues: effect on vanilloid VR1 receptors and on the cellular uptake and enzymatic hydrolysis of anandamide.
British journal of pharmacology 20011001
-
Mechanisms of anandamide-induced vasorelaxation in rat isolated coronary arteries.
British journal of pharmacology 20011001
-
Capsaicin-evoked CGRP release from rat buccal mucosa: development of a model system for studying trigeminal mechanisms of neurogenic inflammation.
The European journal of neuroscience 20011001
-
Noxious heat-induced CGRP release from rat sciatic nerve axons in vitro.
The European journal of neuroscience 20011001
-
Long-term inhibition of nitric oxide synthase potentiates effects of anandamide in the rat mesenteric bed.
European journal of pharmacology 20010921
-
The capsaicin VR1 receptor mediates substance P release in toxin A-induced enteritis in rats.
Peptides 20010901
-
A possible role of lipoxygenase in the activation of vanilloid receptors by anandamide in the guinea-pig bronchus.
British journal of pharmacology 20010901
-
Differential effects of anandamide on acetylcholine release in the guinea-pig ileum mediated via vanilloid and non-CB1 cannabinoid receptors.
British journal of pharmacology 20010901
-
Anandamide activates vanilloid receptor 1 (VR1) at acidic pH in dorsal root ganglia neurons and cells ectopically expressing VR1.
The Journal of biological chemistry 20010817
-
Effects of capsaicin on Ca(2+) release from the intracellular Ca(2+) stores in the dorsal root ganglion cells of adult rats.
Biochemical and biophysical research communications 20010803
-
Protein kinase C activation potentiates gating of the vanilloid receptor VR1 by capsaicin, protons, heat and anandamide.
The Journal of physiology 20010801
-
CH-19 sweet, nonpungent cultivar of red pepper, increased body temperature in mice with vanilloid receptors stimulation by capsiate.
Journal of nutritional science and vitaminology 20010801
-
Analysis of the native quaternary structure of vanilloid receptor 1.
The Journal of biological chemistry 20010727
-
Cannabinoid activation of recombinant and endogenous vanilloid receptors.
European journal of pharmacology 20010727
-
Temperature-dependent activation of recombinant rat vanilloid VR1 receptors expressed in HEK293 cells by capsaicin and anandamide.
European journal of pharmacology 20010706
-
Effects of capsaicin on human intestinal cell line Caco-2.
Cytotechnology 20010701
-
Genital grooming and emesis induced by vanilloids in Suncus murinus, the house musk shrew.
European journal of pharmacology 20010622
-
Vanilloid receptor expression and capsaicin excitation of rat dental primary afferent neurons.
Journal of dental research 20010601
-
Hypolocomotor effects in rats of capsaicin and two long chain capsaicin homologues.
European journal of pharmacology 20010525
-
Capsaicin-induced relaxation in rabbit coronary artery.
The Journal of veterinary medical science 20010501
-
Mechanism of atropine-resistant contraction induced by Dai-kenchu-to in guinea pig ileum.
Japanese journal of pharmacology 20010501
-
The activity of anandamide at vanilloid VR1 receptors requires facilitated transport across the cell membrane and is limited by intracellular metabolism.
The Journal of biological chemistry 20010420
-
Low pH modulation of recombinant vanilloid receptors and perivascular capsaicin-sensitive sensory neurotransmission.
Autonomic neuroscience : basic & clinical 20010412
-
Characterisation using FLIPR of human vanilloid VR1 receptor pharmacology.
European journal of pharmacology 20010406
-
Effect of vanilloid drugs on gastrointestinal transit in mice.
British journal of pharmacology 20010401
-
Capsaicin-evoked release of immunoreactive calcitonin gene-related peptide from rat trigeminal ganglion: evidence for intraganglionic neurotransmission.
Pain 20010401
-
The positive inotropic and chronotropic effects of evodiamine and rutaecarpine, indoloquinazoline alkaloids isolated from the fruits of Evodia rutaecarpa, on the guinea-pig isolated right atria: possible involvement of vanilloid receptors.
Planta medica 20010401
-
Capsazepine, a vanilloid receptor antagonist, inhibits the expression of inducible nitric oxide synthase gene in lipopolysaccharide-stimulated RAW264.7 macrophages through the inactivation of nuclear transcription factor-kappa B.
International immunopharmacology 20010401
-
Sensory pathways and cyclooxygenase regulate mucus gel thickness in rat duodenum.
American journal of physiology. Gastrointestinal and liver physiology 20010301
-
Pharmacological differences between the human and rat vanilloid receptor 1 (VR1).
British journal of pharmacology 20010301
-
The endogenous cannabinoid agonist, anandamide stimulates sensory nerves in guinea-pig airways.
British journal of pharmacology 20010301
-
Anandamide excites central terminals of dorsal root ganglion neurons via vanilloid receptor-1 activation.
The Journal of neuroscience : the official journal of the Society for Neuroscience 20010215
-
Anandamide activates peripheral nociceptors in normal and arthritic rat knee joints.
British journal of pharmacology 20010201
-
Structure-activity relationship for the endogenous cannabinoid, anandamide, and certain of its analogues at vanilloid receptors in transfected cells and vas deferens.
British journal of pharmacology 20010201
-
Capsaicin inhibits activation of voltage-gated sodium currents in capsaicin-sensitive trigeminal ganglion neurons.
Journal of neurophysiology 20010201
-
Regional differences in anandamide- and methanandamide-induced membrane potential changes in rat mesenteric arteries.
The Journal of pharmacology and experimental therapeutics 20010201
-
ACTH inhibits the capsaicin-evoked release of CGRP from rat adrenal afferent nerves.
American journal of physiology. Regulatory, integrative and comparative physiology 20010101
-
Iodo-resiniferatoxin, a new potent vanilloid receptor antagonist.
Molecular pharmacology 20010101
-
Characterization of a novel mechanism accounting for the adverse cholinergic effects of the anticancer drug irinotecan.
British journal of pharmacology 20010101
-
Comparison of intracellular calcium signals evoked by heat and capsaicin in cultured rat dorsal root ganglion neurons and in a cell line expressing the rat vanilloid receptor, VR1.
Neuroscience 20010101
-
Changes in cytosolic calcium in response to noxious heat and their relationship to vanilloid receptors in rat dorsal root ganglion neurons.
Neuroscience 20010101
-
Pharmacology of airway afferent nerve activity.
Respiratory research 20010101
-
Induction of vanilloid receptor channel activity by protein kinase C.
Nature 20001201
-
Characterization using FLIPR of rat vanilloid receptor (rVR1) pharmacology.
British journal of pharmacology 20000601
-
Direct activation of capsaicin receptors by products of lipoxygenases: endogenous capsaicin-like substances.
Proceedings of the National Academy of Sciences of the United States of America 20000523
-
The anandamide transport inhibitor AM404 activates vanilloid receptors.
European journal of pharmacology 20000512
-
Involvement of vanilloid receptors and purinoceptors in the Phoneutria nigriventer spider venom-induced plasma extravasation in rat skin.
European journal of pharmacology 20000317
-
Vanilloid receptors on sensory nerves mediate the vasodilator action of anandamide.
Nature 19990729
-
Identification of the L-menthol binding site in guinea-pig lung membranes.
British journal of pharmacology 19980201
-
Mechanism of acid-induced mesenteric hyperemia in rats.
Life sciences 19980101
-
The selective capsaicin antagonist capsazepine abolishes the antinociceptive action of eugenol and guaiacol.
Journal of dental research 19970401
-
Substance P and capsaicin-induced mechanical hyperalgesia in the rat knee joint; the involvement of bradykinin B1 and B2 receptors.
British journal of pharmacology 19960801
-
Release of beta-endorphin immunoreactivity into ventriculo-cisternal perfusate by lumbar intrathecal capsaicin in the rat.
Brain research 19951201
-
Evidence that glutamate is released from capsaicin-sensitive primary afferent fibers in rats: study with on-line continuous monitoring of glutamate.
Neuroscience research 19940901
-
Regulation of neuropeptide release from pulmonary capsaicin-sensitive afferents in relation to bronchoconstriction.
Acta physiologica Scandinavica. Supplementum 19930101