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Identification of N-(4-((1R,3S,5S)-3-Amino-5-methylcyclohexyl)pyridin-3-yl)-6-(2,6-difluorophenyl)-5-fluoropicolinamide (PIM447), a Potent and Selective Proviral Insertion Site of Moloney Murine Leukemia (PIM) 1, 2, and 3 Kinase Inhibitor in Clinical Trials for Hematological Malignancies.
Journal of medicinal chemistry 20151112
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Anion complexation and transport by isophthalamide and dipicolinamide derivatives: DNA plasmid transformation in E. coli.
Journal of the American Chemical Society 20120822
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Palladium-catalyzed alkenylation and alkynylation of ortho-C(sp2)-H bonds of benzylamine picolinamides.
Organic letters 20120615
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Improved protocol for indoline synthesis via palladium-catalyzed intramolecular C(sp2)-H amination.
Organic letters 20120615
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Integrin α PAT-2/CDC-42 signaling is required for muscle-mediated clearance of apoptotic cells in Caenorhabditis elegans.
PLoS genetics 20120501
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Relaxation of the rigid backbone of an oligoamide-foldamer-based α-helix mimetic: identification of potent Bcl-xL inhibitors.
Organic & biomolecular chemistry 20120421
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Structural polymorphism of human telomere G-quadruplex induced by a pyridyl carboxamide molecule.
Bioorganic & medicinal chemistry letters 20120415
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Evaluation of WO2012003387, Gilead's ASK1 inhibitors.
Expert opinion on therapeutic patents 20120401
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N-(3-Bromo-2-methyl-phen-yl)-2-oxo-1,2-di-hydro-pyridine-3-carboxamide.
Acta crystallographica. Section E, Structure reports online 20120401
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Metal ion-assisted transformations of 2-pyridinealdoxime and hexafluorophosphate.
Dalton transactions (Cambridge, England : 2003) 20120314
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Highly efficient syntheses of azetidines, pyrrolidines, and indolines via palladium catalyzed intramolecular amination of C(sp3)-H and C(sp2)-H bonds at γ and δ positions.
Journal of the American Chemical Society 20120111
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Heterocycle synthesis via direct C-H/N-H coupling.
Journal of the American Chemical Society 20120111
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New potent 5-HT(2A) receptor ligands containing an N'-cyanopicolinamidine nucleus: Synthesis and in vitro pharmacological evaluation.
European journal of medicinal chemistry 20120101
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Cobalt(II), nickel(II) and copper(II) complexes of a hexadentate pyridine amide ligand. Effect of donor atom (ether vs. thioether) on coordination geometry, spin-state of cobalt and M(III)-M(II) redox potential.
Dalton transactions (Cambridge, England : 2003) 20111028
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Antinociceptive and anti-inflammatory activities of nicotinamide and its isomers in different experimental models.
Pharmacology, biochemistry, and behavior 20111001
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4,4'-Bipyridine-3-(thio-phen-3-yl)acrylic acid (1/2).
Acta crystallographica. Section E, Structure reports online 20111001
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Palladium-catalyzed alkylation of ortho-C(sp2)-H bonds of benzylamide substrates with alkyl halides.
Organic letters 20110916
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Adamantyl ethanone pyridyl derivatives: potent and selective inhibitors of human 11β-hydroxysteroid dehydrogenase type 1.
ChemMedChem 20110905
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Bis(μ(2)-pyridine-2-carboxamide oximato)bis-[(pyridine-2-carboxamide oxime)zinc] dinitrate.
Acta crystallographica. Section E, Structure reports online 20110901
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Progress in structure based drug design for G protein-coupled receptors.
Journal of medicinal chemistry 20110714
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Lanthanide directed self-assembly formations of Tb(III) and Eu(III) luminescent complexes from tryptophan based pyridyl amide ligands.
Chemical communications (Cambridge, England) 20110707
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Photoinduced intramolecular tryptophan oxidation and excited-state behavior of [Re(L-AA)(CO)3(α-diimine)](+) (L = pyridine or imidazole, AA = tryptophan, tyrosine, phenylalanine).
Inorganic chemistry 20110704
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Synthesis and cytotoxic evaluation of novel N-methyl-4-phenoxypicolinamide derivatives.
Molecules (Basel, Switzerland) 20110620
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TTF salts of optically pure cobalt pyridine amidates; detection of soluble assemblies with stoichiometry corresponding to the solid state.
Dalton transactions (Cambridge, England : 2003) 20110227
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Highly sensitive and selective turn-on fluorescent and chromogenic probe for Cu2+ and ClO- based on a N-picolinyl rhodamine B-hydrazide derivative.
Organic & biomolecular chemistry 20110121
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Sorafenib and its tosylate salt: a multikinase inhibitor for treating cancer.
Acta crystallographica. Section C, Crystal structure communications 20110101
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Heterologous expression, purification and characterization of nitrilase from Aspergillus niger K10.
BMC biotechnology 20110101
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SKLB610: a novel potential inhibitor of vascular endothelial growth factor receptor tyrosine kinases inhibits angiogenesis and tumor growth in vivo.
Cellular physiology and biochemistry : international journal of experimental cellular physiology, biochemistry, and pharmacology 20110101
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2D QSAR Studies of Several Potent Aminopyridine, Anilinopyrimidine and Pyridine Carboxamide-based JNK Inhibitors.
Indian journal of pharmaceutical sciences 20110101
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Synthesis, crystal structure, DNA-binding and cytotoxicity in vitro of novel cis-Pt(II) and trans-Pd(II) pyridine carboxamide complexes.
Bioorganic & medicinal chemistry letters 20101215
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Synthesis and SAR studies of 1,4-benzoxazine MenB inhibitors: novel antibacterial agents against Mycobacterium tuberculosis.
Bioorganic & medicinal chemistry letters 20101101
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Amide hydrogen bonding: control of the molecular and extended structures of two symmetrical pyridine-2-carboxamide derivatives.
Acta crystallographica. Section C, Crystal structure communications 20101101
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Unconventional hydrogen bonding and π-stacking in two substituted pyridine carboxamides.
Acta crystallographica. Section C, Crystal structure communications 20101001
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Intramolecular sigma-bond metathesis/protonolysis on zirconium(IV) and hafnium(IV) pyridylamido olefin polymerization catalyst precursors: exploring unexpected reactivity paths.
Inorganic chemistry 20100802
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Synthesis and evaluation of novel antifungal agents-quinoline and pyridine amide derivatives.
Bioorganic & medicinal chemistry letters 20100801
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Bis[N-(4-chloro-phen-yl)pyridine-3-carboxamide]-silver(I) nitrate.
Acta crystallographica. Section E, Structure reports online 20100801
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Kinetic and equilibrium studies of the removal of cadmium ions from acidic chloride solutions by hydrophobic pyridinecarboxamide extractants.
Journal of hazardous materials 20100715
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rac-N-[Hy-droxy(4-pyrid-yl)meth-yl]picolinamide: a hemiamidal.
Acta crystallographica. Section E, Structure reports online 20100701
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Hybridization of long pyridine-dicarboxamide oligomers into multi-turn double helices: slow strand association and dissociation, solvent dependence, and solid state structures.
Chemistry, an Asian journal 20100601
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2-Ferrocenyl-N-(6-methyl-2-pyrid-yl)benzamide.
Acta crystallographica. Section E, Structure reports online 20100401
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Bis{2-hydr-oxy-N-[2-(2-pyrid-yl)eth-yl]benzamide}copper(I) tetra-fluoridoborate.
Acta crystallographica. Section E, Structure reports online 20100201
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Role of heme oxygenase in inflammation, insulin-signalling, diabetes and obesity.
Mediators of inflammation 20100101
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Amide linkage isomerism as an activity switch for organometallic osmium and ruthenium anticancer complexes.
Journal of medicinal chemistry 20091210
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Interaction of nicotinamide and picolinamide with phosphatidylcholine and phosphatidylethanolamine membranes: a combined approach using dipole potential measurements and quantum chemical calculations.
Biochimica et biophysica acta 20091201
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2-Carbamylpyridinium tetra-chlorido-ferrate(III).
Acta crystallographica. Section E, Structure reports online 20091101
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Bis[μ-2-(aminosulfanyl)pyridine(1-)]bis-[(η-penta-methyl-cyclo-penta-dien-yl)iridium(III)] diiodide.
Acta crystallographica. Section E, Structure reports online 20091001
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New generation of metal string complexes: strengthening metal-metal interaction via naphthyridyl group modulated oligo-alpha-pyridylamido ligands.
Chemical communications (Cambridge, England) 20090807
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Cobalt complex as building blocks: synthesis, characterization, and catalytic applications of {Cd2+-Co3+-Cd2+} and {Hg2+-Co3+-Hg2+} heterobimetallic complexes.
Inorganic chemistry 20090615
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Investigation on the complex of diperoxovanadate with picolinamide.
Spectrochimica acta. Part A, Molecular and biomolecular spectroscopy 20090601
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Hydrogen-bonded structures of the isomeric 2-, 3- and 4-carbamoylpyridinium hydrogen chloranilates.
Acta crystallographica. Section C, Crystal structure communications 20090601
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Discovery of novel 3,6-disubstituted 2-pyridinecarboxamide derivatives as GK activators.
Bioorganic & medicinal chemistry letters 20090515
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Utility of MetaSite in improving metabolic stability of the neutral indomethacin amide derivative and selective cyclooxygenase-2 inhibitor 2-(1-(4-chlorobenzoyl)-5-methoxy-2-methyl-1H-indol-3-yl)-N-phenethyl-acetamide.
Drug metabolism and disposition: the biological fate of chemicals 20090501
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IRAK-4 inhibitors for inflammation.
Current topics in medicinal chemistry 20090501
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The discovery of biaryl carboxamides as novel small molecule agonists of the motilin receptor.
Bioorganic & medicinal chemistry letters 20081215
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Dimer formation in nicotinamide and picolinamide in the gas and condensed phases probed by infrared spectroscopy.
Physical chemistry chemical physics : PCCP 20081214
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Synthesis, characterization and antibacterial activity of cobalt(III) complexes with pyridine-amide ligands.
European journal of medicinal chemistry 20081001
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A photolabile ligand for light-activated release of caged copper.
Journal of the American Chemical Society 20080917
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Diaqua-{2,6-bis-[N-(2-pyridinylmeth-yl)-carbamo-yl]-phenolato-κO,O}zinc(II).
Acta crystallographica. Section E, Structure reports online 20080701
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[Synthesis and DNA-binding properties of three compounds containing pyridinecarboxamide].
Guang pu xue yu guang pu fen xi = Guang pu 20080601
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[N,N'-(1,2-Diphenyl-ethane-1,2-di-yl)bis-(pyridine-2-carboxamidato)]nickel(II) diethyl ether hemisolvate.
Acta crystallographica. Section E, Structure reports online 20080301
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cis-Bis(azido-κN)bis-(pyridine-2-carbox-amide-κN,O)nickel(II).
Acta crystallographica. Section E, Structure reports online 20080201
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Bis[N-(8-quinol-yl)pyridine-2-carbox-amidato-κN,N',N'']manganese(III) perchlorate monohydrate.
Acta crystallographica. Section E, Structure reports online 20080201
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Molecular structure, vibrational spectra, quantum chemical calculations and photochemistry of picolinamide and isonicotinamide isolated in cryogenic inert matrixes and in the neat low-temperature solid phases.
The journal of physical chemistry. A 20080110
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14N NQR study of nicotinamide and related compounds.
Magnetic resonance in chemistry : MRC 20080101
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Matrix-assisted laser desorption/ionization signal enhancement of peptides by picolinamidination of amino groups.
Rapid communications in mass spectrometry : RCM 20080101
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Characterisation of the substrate specificity of the nitrile hydrolyzing system of the acidotolerant black yeast Exophiala oligosperma R1.
Studies in mycology 20080101
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Flonicamid, a novel insecticide with a rapid inhibitory effect on aphid feeding.
Pest management science 20071001
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Cofactor-specific modulation of 11beta-hydroxysteroid dehydrogenase 1 inhibitor potency.
Biochimica et biophysica acta 20070901
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Solution equilibria of copper(II) complexation with N,N'-(2,2'-azanediylbis(ethane-2,1-diyl))dipicolinamide: a bio-distribution and dermal absorption study.
Journal of inorganic biochemistry 20070801
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Mechanism of activation of a hafnium pyridyl-amide olefin polymerization catalyst: ligand modification by monomer.
Journal of the American Chemical Society 20070627
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Development of a disposable mercury ion-selective optode based on trityl-picolinamide as ionophore.
Analytica chimica acta 20070522
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Structural variation in copper(I) complexes with pyridylmethylamide ligands: structural analysis with a new four-coordinate geometry index, tau4.
Dalton transactions (Cambridge, England : 2003) 20070307
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[Poly(ADP-ribosa)polymerase--the relationships with life span and carcinogenesis].
Advances in gerontology = Uspekhi gerontologii 20070101
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Effects of hydrogen bonding on the ring stretching modes of pyridine.
The journal of physical chemistry. A 20061221
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Copper(I) coordination chemistry of (pyridylmethyl)amide ligands.
Inorganic chemistry 20061113
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Synthesis and biological evaluation of purine derivatives incorporating metal chelating ligands as HIV integrase inhibitors.
Bioorganic & medicinal chemistry 20060815
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Multinuclear copper complexes of pyridylmethylamide ligands.
Dalton transactions (Cambridge, England : 2003) 20060421
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Electrophilic activation of lactams with Tf2O and pyridine: expedient synthesis of (+/-)-tetraponerine T4.
Organic letters 20051124
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Novel metal-linked face-to-face porphyrazine dimer.
Inorganic chemistry 20051114
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Mechanistic explanation to the catalysis by pyrazinamide and ethambutol of reaction between rifampicin and isoniazid in anti-TB FDCs.
Journal of pharmaceutical and biomedical analysis 20051004
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Bivalent and trivalent iron complexes of acyclic hexadentate ligands providing pyridyl/pyrazine-amide-thioether coordination.
Inorganic chemistry 20050808
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In vitro alpha-glucosidase inhibitory effect of Zn(II) complex with 6-methyl-2-picolinmethylamide.
Chemical & pharmaceutical bulletin 20050401
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The amide rotational barrier in isonicotinamide: Dynamic NMR and ab initio studies.
The journal of physical chemistry. A 20050217
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Supramolecular copper hydroxide tennis balls: self-assembly, structures, and magnetic properties of octanuclear [Cu(8)L(8)(OH)(4)](4+) clusters (HL = N-(2-pyridylmethyl)acetamide).
Inorganic chemistry 20041101
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Correlation of mass spectrometry identified bacterial biomarkers from a fielded pyrolysis-gas chromatography-ion mobility spectrometry biodetector with the microbiological gram stain classification scheme.
Analytical chemistry 20041101
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Molecular, supramolecular and solution structures of peroxovanadium complexes with ON and O3N donor set ligands: two new types of cationic-anionic peroxovanadium(V) peroxovanadates(V).
Dalton transactions (Cambridge, England : 2003) 20041021
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Picolinamidium squarate and di-p-toluidinium squarate dihydrate.
Acta crystallographica. Section C, Crystal structure communications 20040801
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Diaquabis(pyridine-2-carboxamide-kappa2N1,O2)nickel(II) disaccharinate tetrahydrate.
Acta crystallographica. Section C, Crystal structure communications 20040701
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Tris[N-(4-fluorophenyl)pyridine-2-carboxamidato-kappa2N,N']cobalt(III) trihydrate: a novel meridional complex.
Acta crystallographica. Section C, Crystal structure communications 20040501
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New pyridine carboxamide ligands and their complexation to copper(II). X-Ray crystal structures of mono-, di, tri- and tetranuclear copper complexes.
Dalton transactions (Cambridge, England : 2003) 20040321
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Solid-state and solution properties of cationic lanthanide complexes of a new neutral heptadentate N4O3 tripodal ligand.
Inorganic chemistry 20031201
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The amide rotational barriers in picolinamide and nicotinamide: NMR and ab initio studies.
Journal of the American Chemical Society 20030820
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Synthesis and characterization of cobalt(III) complexes containing 2-pyridinecarboxamide ligands and their application in catalytic oxidation of ethylbenzene with dioxygen.
Chemical communications (Cambridge, England) 20030607
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ECNI GC-MS analysis of picolinic and quinolinic acids and their amides in human plasma, CSF, and brain tissue.
Advances in experimental medicine and biology 20030101
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Amination of pyridylketenes: experimental and computational studies of strong amide enol stabilization by the 2-pyridyl group.
Journal of the American Chemical Society 20021120
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Spontaneous reduction of a low-spin Fe(III) complex of a neutral pentadentate N(5) Schiff base ligand to the corresponding Fe(II) species in acetonitrile.
Inorganic chemistry 20021021
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Unusual reactivity of methylene group adjacent to pyridine-2-carboxamido moiety in iron(III) and cobalt(III) complexes.
Inorganic chemistry 20020520
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Potential insulinominetic agents of zinc(II) complexes with picolinamide derivatives: preparations of complexes, in vitro and in vivo studies.
Chemical & pharmaceutical bulletin 20020301
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Oxygen capture by lithiated organozinc reagents containing aromatic 2-pyridylamide ligands.
Chemistry (Weinheim an der Bergstrasse, Germany) 20010903
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Molecularly imprinted polymers from nicotinamide and its positional isomers.
Journal of molecular recognition : JMR 20010101
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Tumorigenic action of streptozotocin on the pancreas and kidney in male Wistar rats.
Cancer research 19780701