170851-70-4 | 2-Methylalanyl-L-histidyl-3-(2-naphthalenyl)-D-alanyl-D-phenylalanyl-L-lysinamide

Packsize	Purity	Availability	Price	Discounted Price
5mg	98%	in stock	$106.00	$75.00
25mg	98%	in stock	$291.00	$204.00
50mg	98%	in stock	$520.00	$364.00
100mg	98%	in stock	$936.00	$655.00

Description

• Catalog Number: AE98751
• Chemical Name: 2-Methylalanyl-L-histidyl-3-(2-naphthalenyl)-D-alanyl-D-phenylalanyl-L-lysinamide
• CAS Number: 170851-70-4
• Molecular Formula: C38H49N9O5
• Molecular Weight: 711.8529600000002
• MDL Number: MFCD02179658
• SMILES: NCCCC[C@@H](C(=O)N)NC(=O)[C@@H](Cc1ccccc1)NC(=O)[C@@H](Cc1ccc2c(c1)cccc2)NC(=O)[C@H](Cc1cnc[nH]1)NC(=O)C(N)(C)C

Computed Properties

• Complexity: 1200
• Covalently-Bonded Unit Count: 1
• Defined Atom Stereocenter Count: 4
• Heavy Atom Count: 52
• Hydrogen Bond Acceptor Count: 8
• Hydrogen Bond Donor Count: 8
• Rotatable Bond Count: 19
• XLogP3: 1.8

Literature

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  Nihon rinsho. Japanese journal of clinical medicine 20040901

• Growth hormone (GH) hypersecretion and GH receptor resistance in streptozotocin diabetic mice in response to a GH secretagogue.

  Experimental diabesity research 20030101

• The influence of conformational restriction in the C-terminus of growth hormone secretagogues on their potency.

  European journal of medicinal chemistry 20020601

• The growth hormone secretagogue ipamorelin counteracts glucocorticoid-induced decrease in bone formation of adult rats.

  Growth hormone & IGF research : official journal of the Growth Hormone Research Society and the International IGF Research Society 20011001

• Highly potent growth hormone secretagogues: hybrids of NN703 and ipamorelin.

  Bioorganic & medicinal chemistry letters 20010723

• Structural similarity of ghrelin derivatives to peptidyl growth hormone secretagogues.

  Biochemical and biophysical research communications 20010615