271-29-4 | 6-Azaindole

Packsize	Purity	Availability	Price	Discounted Price
1g	98%	in stock	$20.00	$14.00
5g	98%	in stock	$24.00	$17.00
10g	98%	in stock	$37.00	$26.00
25g	98%	in stock	$88.00	$62.00
100g	98%	in stock	$332.00	$233.00

Description

• Catalog Number: AB69687
• Chemical Name: 6-Azaindole
• CAS Number: 271-29-4
• Molecular Formula: C7H6N2
• Molecular Weight: 118.1359
• MDL Number: MFCD01686899
• SMILES: c1ncc2c(c1)cc[nH]2

Computed Properties

• Complexity: 103
• Covalently-Bonded Unit Count: 1
• Heavy Atom Count: 9
• Hydrogen Bond Acceptor Count: 1
• Hydrogen Bond Donor Count: 1
• XLogP3: 1

Literature

• Synthesis of 2,5-disubstituted 6-azaindoles from substituted aziridines via intramolecular cyclization.

  Organic letters 20120615

• Structure-based optimization of potent 4- and 6-azaindole-3-carboxamides as renin inhibitors.

  Bioorganic & medicinal chemistry letters 20110915

• Synthesis of azaheterocycles from aryl ketone O-acetyl oximes and internal alkynes by Cu-Rh bimetallic relay catalysts.

  The Journal of organic chemistry 20110805

• Access to pyrrolo-pyridines by gold-catalyzed hydroarylation of pyrroles tethered to terminal alkynes.

  Beilstein journal of organic chemistry 20110101

• Novel 1H-pyrrolo[2,3-c]pyridines as acid pump antagonists (APAs).

  Bioorganic & medicinal chemistry letters 20100901

• Evaluation of basic, heterocyclic ring systems as templates for use as potassium competitive acid blockers (pCABs).

  Bioorganic & medicinal chemistry letters 20091201

• Synthesis of 4- and 6-azaindoles via the Fischer reaction.

  Organic letters 20091119

• Discovery of 1-[4-(3-chlorophenylamino)-1-methyl-1H-pyrrolo[3,2-c]pyridin-7-yl]-1-morpholin-4-ylmethanone (GSK554418A), a brain penetrant 5-azaindole CB2 agonist for the treatment of chronic pain.

  Journal of medicinal chemistry 20091008

• Design, synthesis and dopamine D4 receptor binding activities of new N-heteroaromatic 5/6-ring Mannich bases.

  Bioorganic & medicinal chemistry 20090701

• Magnetic interactions in two heterobridged dinuclear copper(II) complexes: orbital complementarity or countercomplementarity?

  The journal of physical chemistry. A 20080911

• Solvent-dependent oxidations of 5- and 6-azaindoles to trioxopyrrolopyridines and functionalised azaindoles.

  Organic & biomolecular chemistry 20080421

• A novel one-step synthesis of 2-substituted 6-azaindoles from 3-amino-4-picoline and carboxylic esters.

  The Journal of organic chemistry 20050805

• Novel potent 5-HT(1F) receptor agonists: structure-activity studies of a series of substituted N-[3-(1-methyl-4-piperidinyl)-1H-pyrrolo[3,2-b]pyridin-5-yl]amides.

  Journal of medicinal chemistry 20030703