-
3-Benzyl-5-methyl-1,2-benzoxazole 2-oxide.
Acta crystallographica. Section E, Structure reports online 20121001
-
3-Chloro-methyl-6,7-dimethyl-1,2-benz-oxazole.
Acta crystallographica. Section E, Structure reports online 20121001
-
Catalytic asymmetric hydrogenation of 3-substituted benzisoxazoles.
Molecules (Basel, Switzerland) 20120606
-
Benzisoxazole analogs as glycogen synthase activators, a patent evaluation (WO2011057956).
Expert opinion on therapeutic patents 20120601
-
Critical appraisal of lurasidone in the management of schizophrenia.
Neuropsychiatric disease and treatment 20120101
-
The role of paliperidone extended release for the treatment of bipolar disorder.
Neuropsychiatric disease and treatment 20120101
-
Genetic polymorphisms in CYP2E1: association with schizophrenia susceptibility and risperidone response in the Chinese Han population.
PloS one 20120101
-
Zonisamide: its pharmacology, efficacy and safety in clinical trials.
Acta neurologica Scandinavica. Supplementum 20120101
-
A divergent and selective synthesis of isomeric benzoxazoles from a single N-Cl imine.
Organic letters 20111202
-
Paliperidone: 3-{2-[4-(6-fluoro-1,2-benzoxazol-3-yl)piperidin-1-yl]eth-yl}-9-hy-droxy-2-methyl-1,6,7,8,9,9a-hexa-hydro-pyrido[1,2-a]pyrimidin-4-one.
Acta crystallographica. Section E, Structure reports online 20111101
-
3-[Chloro-(phen-yl)meth-yl]-6-methyl-1,2-benzoxazole.
Acta crystallographica. Section E, Structure reports online 20111101
-
Design, synthesis and SAR of indazole and benzoisoxazole containing 4-azetidinyl-1-aryl-cyclohexanes as CCR2 antagonists.
Bioorganic & medicinal chemistry letters 20111015
-
Biological evaluation of novel benzisoxazole derivatives as PPARδ agonists.
Bioorganic & medicinal chemistry 20110515
-
Optimization and in vitro toxicity evaluation of G4 PAMAM dendrimer-risperidone complexes.
European journal of medicinal chemistry 20110301
-
3-{[6-(4-Chloro-phen-yl)imidazo[2,1-b][1,3,4]thia-diazol-2-yl]meth-yl}-1,2-benzoxazole.
Acta crystallographica. Section E, Structure reports online 20110301
-
Elucidation of a novel bioactivation pathway of a 3,4-unsubstituted isoxazole in human liver microsomes: formation of a glutathione adduct of a cyanoacrolein derivative after isoxazole ring opening.
Drug metabolism and disposition: the biological fate of chemicals 20110201
-
Synthesis of elastin based peptides conjugated to benzisoxazole as a new class of potent antimicrobials--A novel approach to enhance biocompatibility.
European journal of medicinal chemistry 20110201
-
Synthesis of a novel human PPARδ selective agonist and its stimulatory effect on oligodendrocyte differentiation.
Bioorganic & medicinal chemistry letters 20110101
-
Paliperidone extended-release: does it have a place in antipsychotic therapy?
Drug design, development and therapy 20110101
-
3-{[5-(4-Bromo-phen-yl)imidazo[2,1-b][1,3,4]thia-diazol-2-yl]meth-yl}-1,2-benzoxazole.
Acta crystallographica. Section E, Structure reports online 20110101
-
Paliperidone ER in the Treatment of Borderline Personality Disorder: A Pilot Study of Efficacy and Tolerability.
Depression research and treatment 20110101
-
Clinical utility of the risperidone formulations in the management of schizophrenia.
Neuropsychiatric disease and treatment 20110101
-
Benzoxazinones as Human Peroxisome Proliferator Activated Receptor Gamma (PPARγ) Agonists: A Docking Study Using Glide.
Indian journal of pharmaceutical sciences 20110101
-
The effect of risperidone on D-amino acid oxidase activity as a hypothesis for a novel mechanism of action in the treatment of schizophrenia.
Journal of psychopharmacology (Oxford, England) 20100701
-
Intramolecular Fe(II)-catalyzed N-O or N-N bond formation from aryl azides.
Organic letters 20100618
-
An efficient entry to 1,2-benzisoxazoles via 1,3-dipolar cycloaddition of in situ generated nitrile oxides and benzyne.
Organic & biomolecular chemistry 20100607
-
Iloperidone for the treatment of schizophrenia.
The Annals of pharmacotherapy 20100501
-
Zonisamide: a new drug for Parkinson's disease.
Drugs of today (Barcelona, Spain : 1998) 20100401
-
An improved synthesis of 1,2-benzisoxazoles: TBAF mediated 1,3-dipolar cycloaddition of nitrile oxides and benzyne.
Chemical communications (Cambridge, England) 20100227
-
Microwave-promoted synthesis of 3-amino-substituted 1,2-benzisoxazoles.
Future medicinal chemistry 20100201
-
New atypical antipsychotics for schizophrenia: iloperidone.
Drug design, development and therapy 20100101
-
Emerging treatments in the management of bipolar disorder - focus on risperidone long acting injection.
Neuropsychiatric disease and treatment 20100101
-
Once-monthly paliperidone injection for the treatment of schizophrenia.
Neuropsychiatric disease and treatment 20100101
-
Acute administration of clozapine and risperidone altered dopamine metabolism more in rat caudate than in nucleus accumbens: a dose-response relationship.
Scientia pharmaceutica 20100101
-
[The review of acute risperidone poisoning].
Przeglad lekarski 20100101
-
An Open-label Trial of Risperidone and Fluoxetine in Children with Autistic Disorder.
Indian journal of psychological medicine 20100101
-
4-[(E)-(2,4-Difluoro-phen-yl)(hydroxy-imino)meth-yl]piperidinium picrate.
Acta crystallographica. Section E, Structure reports online 20091001
-
Theoretical investigations of the photochemical isomerizations of indoxazene and isoxazole.
The Journal of organic chemistry 20090821
-
Ethyl 6-(6-meth-oxy-2-naphth-yl)-2-oxo-4-(2-thien-yl)cyclo-hex-3-ene-1-carboxyl-ate.
Acta crystallographica. Section E, Structure reports online 20090701
-
4-(6-Fluoro-1,2-benzisoxazol-3-yl)-1-[2-(2-methyl-4-oxo-6,7,8,9-tetra-hydro-4H-pyrido[1,2-a]pyrimidin-3-yl)eth-yl]piperidinium nitrate.
Acta crystallographica. Section E, Structure reports online 20090701
-
In thrombin stimulated human platelets Citalopram, Promethazine, Risperidone, and Ziprasidone, but not Diazepam, may exert their pharmacological effects also through intercalation in membrane phospholipids in a receptor-independent manner.
Journal of chemical biology 20090601
-
Synthesis of alkenyldiarylmethanes (ADAMs) containing benzo[d]isoxazole and oxazolidin-2-one rings, a new series of potent non-nucleoside HIV-1 reverse transcriptase inhibitors.
European journal of medicinal chemistry 20090301
-
A systematic review of quality of life and weight gain-related issues in patients treated for severe and persistent mental disorders: focus on aripiprazole.
Neuropsychiatric disease and treatment 20090101
-
Long-term safety and effectiveness of zonisamide in the treatment of epilepsy: a review of the literature.
Neuropsychiatric disease and treatment 20090101
-
HPLC method for simultaneous determination of impurities and degradation products in zonisamide.
Indian journal of pharmaceutical sciences 20090101
-
3-(4-Chloro-phen-yl)-2,1-benzisoxazole-5-carbonyl chloride.
Acta crystallographica. Section E, Structure reports online 20081201
-
[Novel access to indazoles based on palladium-catalyzed amination chemistry].
Yakugaku zasshi : Journal of the Pharmaceutical Society of Japan 20080701
-
Kemp elimination: a probe reaction to study ionic liquids properties.
The Journal of organic chemistry 20080502
-
Absorption, metabolism, and excretion of paliperidone, a new monoaminergic antagonist, in humans.
Drug metabolism and disposition: the biological fate of chemicals 20080401
-
Paliperidone for schizophrenia.
American journal of health-system pharmacy : AJHP : official journal of the American Society of Health-System Pharmacists 20080301
-
Reductive isoxazole ring opening of the anticoagulant razaxaban is the major metabolic clearance pathway in rats and dogs.
Drug metabolism and disposition: the biological fate of chemicals 20080201
-
Review of risperidone for the treatment of pediatric and adolescent bipolar disorder and schizophrenia.
Neuropsychiatric disease and treatment 20080201
-
Iloperidone: a new benzisoxazole atypical antipsychotic drug. Is it novel enough to impact the crowded atypical antipsychotic market?
Expert opinion on investigational drugs 20080101
-
RP-HPLC Estimation of Risperidone in Tablet Dosage Forms.
Indian journal of pharmaceutical sciences 20080101
-
Isolation of liver aldehyde oxidase containing fractions from different animals and determination of kinetic parameters for benzaldehyde.
Indian journal of pharmaceutical sciences 20080101
-
Paliperidone ER: a review of the clinical trial data.
Neuropsychiatric disease and treatment 20071201
-
Benefit of liquid crystal moieties in the MIP technique.
Analytica chimica acta 20070515
-
Novel base catalysed rearrangement of sultone oximes to 1,2-benzisoxazole-3-methane sulfonate derivatives.
Beilstein journal of organic chemistry 20070101
-
Atypical antipsychotics to treat the neuropsychiatric symptoms of dementia.
Neuropsychiatric disease and treatment 20061201
-
Decomposition and isomerization of 1,2-benzisoxazole: single-pulse shock-tube experiments, quantum chemical and transition-state theory calculations.
The journal of physical chemistry. A 20061019
-
Zonisamide - a review of experience and use in partial seizures.
Neuropsychiatric disease and treatment 20060901
-
Risperidone in the treatment of bipolar mania.
Neuropsychiatric disease and treatment 20060601
-
Development of hypoxia selective cytotoxins for cancer treatment: an update.
Medicinal chemistry (Shariqah (United Arab Emirates)) 20060501
-
Synthesis and anti-HIV activity of new alkenyldiarylmethane (ADAM) non-nucleoside reverse transcriptase inhibitors (NNRTIs) incorporating benzoxazolone and benzisoxazole rings.
Bioorganic & medicinal chemistry 20060401
-
Is subnanomolar binding affinity required for the in vivo imaging of acetylcholinesterase? Studies on 18F-labeled G379.
Nuclear medicine and biology 20060101
-
Successful treatment of six patients with neuroleptic malignant syndrome associated with myoglobulinemic acute renal failure.
Renal failure 20060101
-
Novel indole-based peroxisome proliferator-activated receptor agonists: design, SAR, structural biology, and biological activities.
Journal of medicinal chemistry 20051229
-
Identification of the structural requirements of the receptor-binding affinity of diphenolic azoles to estrogen receptors alpha and beta by three-dimensional quantitative structure-activity relationship and structure-activity relationship analysis.
Journal of medicinal chemistry 20051201
-
An efficient synthesis of a dual PPAR alpha/gamma agonist and the formation of a sterically congested alpha-aryloxyisobutyric acid via a Bargellini reaction.
The Journal of organic chemistry 20051014
-
Carbonic anhydrase inhibitors. Zonisamide is an effective inhibitor of the cytosolic isozyme II and mitochondrial isozyme V: solution and X-ray crystallographic studies.
Bioorganic & medicinal chemistry letters 20050502
-
Mechanistic study of proton transfer and hysteresis in catalytic antibody 16E7 by site-directed mutagenesis and homology modeling.
Bioorganic & medicinal chemistry 20050215
-
Design, synthesis and evaluation of bicyclic benzamides as novel 5-HT1F receptor agonists.
Bioorganic & medicinal chemistry letters 20041220
-
Overview of Japanese experience-controlled and uncontrolled trials.
Seizure 20041201
-
A high-performance liquid chromatographic-atmospheric pressure chemical ionization-tandem mass spectrometric method for determination of risperidone and 9-hydroxyrisperidone in human plasma.
Journal of analytical toxicology 20040901
-
1,2-benzisoxazole phosphorodiamidates as novel anticancer prodrugs requiring bioreductive activation.
Journal of medicinal chemistry 20031204
-
2-(2,1-benzoxazol-3-yl)-3,5-dimethoxyphenol and 3-phenyl-2,1-benzoxazole.
Acta crystallographica. Section C, Crystal structure communications 20030901
-
Substituent effect on the reductive N-dearylation of 3-(indol-1-yl)-1,2-benzisoxazoles by rat liver microsomes.
Drug metabolism and disposition: the biological fate of chemicals 20030801
-
Isoxazole --> benzisoxazole rearrangement promoted cascade reactions affording stereodefined polycycles.
Organic letters 20030220
-
Stimulation by antipsychotic agents of mitogen-activated protein kinase (MAPK) coupled to cloned, human (h)serotonin (5-HT)(1A) receptors.
Psychopharmacology 20020701
-
Biocatalysis of isomerization of 1,2-benzisoxazole by bovine serum albumin in an organic solvent.
Biotechnology and bioengineering 20010920