496-15-1 | Indoline

Packsize	Purity	Availability	Price	Discounted Price
5g	97%	in stock	$6.00	$4.00
10g	97%	in stock	$7.00	$5.00
25g	97%	in stock	$9.00	$6.00
100g	97%	in stock	$15.00	$11.00
500g	97%	in stock	$72.00	$51.00

Description

• Catalog Number: AI51093
• Chemical Name: Indoline
• CAS Number: 496-15-1
• Molecular Formula: C8H9N
• Molecular Weight: 119.1638
• MDL Number: MFCD00005705
• SMILES: C1CNC2=CC=CC=C21

Computed Properties

• Complexity: 101
• Covalently-Bonded Unit Count: 1
• Heavy Atom Count: 9
• Hydrogen Bond Acceptor Count: 1
• Hydrogen Bond Donor Count: 1
• XLogP3: 1.9

Literature

• Metal-free catalyzed oxidative trimerization of indoles by using TEMPO in air: a biomimetic approach to 2-(1H-indol-3-yl)-2,3'-biindolin-3-ones.

  Organic & biomolecular chemistry 20121128

• Ultrafast dynamics of the indoline dye D149 on electrodeposited ZnO and sintered ZrO2 and TiO2 thin films.

  Physical chemistry chemical physics : PCCP 20121128

• Ordered networks of ZnO-nanowire hierarchical urchin-like structures for improved dye-sensitized solar cells.

  Physical chemistry chemical physics : PCCP 20121005

• Methyl (3S,3'R)-1-methyl-2,2''-dioxo-1',2',3',5',6',7',8',8a'-octa-hydro-dispiro-[indoline-3,2'-indolizine-3',3''-indoline]-1'-carboxyl-ate.

  Acta crystallographica. Section E, Structure reports online 20121001

• Methyl (3R*,3'S*)-1',1''-dimethyl-2,2''-dioxodispiro-[indoline-3,2'-pyrrolidine-3',3''-indoline]-4'-carboxyl-ate.

  Acta crystallographica. Section E, Structure reports online 20121001

• 5-Chloro-N-{4-oxo-2-[4-(trifluoro-meth-yl)phen-yl]-1,3-thia-zolidin-3-yl}-3-phenyl-1H-indole-2-carboxamide.

  Acta crystallographica. Section E, Structure reports online 20121001

• Stereoselective synthesis of 2,3-disubstituted indoline diastereoisomers by chemoenzymatic processes.

  The Journal of organic chemistry 20120921

• Spiro-fused pyrrolidine, piperidine, and oxindole scaffolds from lactams.

  Organic letters 20120921

• Structure and catalytic mechanism of a cyclic dipeptide prenyltransferase with broad substrate promiscuity.

  Journal of molecular biology 20120907

• Discovery of a potent, orally bioavailable and highly selective human neuronal nitric oxide synthase (nNOS) inhibitor, N-(1-(piperidin-4-yl)indolin-5-yl)thiophene-2-carboximidamide as a pre-clinical development candidate for the treatment of migraine.

  European journal of medicinal chemistry 20120901

• (3'R)-3'-Benzyl-2',3'-dihydro-1H-spiro-[indole-3,1'-naphtho-[2,3-c]pyrrole]-2,4',9'-trione.

  Acta crystallographica. Section E, Structure reports online 20120901

• Stable sensitization of ZnO by improved anchoring of indoline dyes.

  Chemphyschem : a European journal of chemical physics and physical chemistry 20120827

• Nucleophilic addition of Grignard reagents to 3-acylindoles: stereoselective synthesis of highly substituted indoline scaffolds.

  Organic letters 20120803

• (1S,3R)-3-Isobutyl-2,3-dihydro-spiro[benzo[f]isoindole-1,3'-indoline]-2',4,9-trione methanol monosolvate.

  Acta crystallographica. Section E, Structure reports online 20120801

• Ultrasound-promoted one-pot, three-component synthesis of spiro[indoline-3,1'-pyrazolo[1,2-b]phthalazine] derivatives.

  Molecules (Basel, Switzerland) 20120723

• Approach to the synthesis of indoline derivatives from diaryliodonium salts.

  The Journal of organic chemistry 20120706

• Enantioselective copper-catalyzed construction of aryl pyrroloindolines via an arylation-cyclization cascade.

  Journal of the American Chemical Society 20120704

• 1'-Butyl-2-methyl-1',2,2',3,4,9-hexa-hydro-spiro-[benzo[f]isoindole-1,3'-indole]-2',4,9-trione.

  Acta crystallographica. Section E, Structure reports online 20120701

• Constructing organic D-A-π-A-featured sensitizers with a quinoxaline unit for high-efficiency solar cells: the effect of an auxiliary acceptor on the absorption and the energy level alignment.

  Chemistry (Weinheim an der Bergstrasse, Germany) 20120625

• Regioselective synthesis of pyrimido[1,2-a][1,3,5]triazin-6-ones via reaction of 1-(6-oxo-1,6-dihydropyrimidin-2-yl)guanidines with triethylorthoacetate: observation of an unexpected rearrangement.

  Organic & biomolecular chemistry 20120621

• Synthesis of indolines, indoles, and benzopyrrolizidinones from simple aryl azides.

  Organic letters 20120615

• Improved protocol for indoline synthesis via palladium-catalyzed intramolecular C(sp2)-H amination.

  Organic letters 20120615

• Design and synthesis of new biprivileged molecular scaffolds: indolo-fused benzodiazepinyl/quinoxalinyl benzimidazoles.

  Chemistry, an Asian journal 20120601

• 1,1''-Bis(prop-2-en-1-yl)-1,1'',2,2''-tetra-hydro-dispiro-[indole-3,7'-[6,9]diaza-tricyclo-[7.3.0.0(2,6)]dodecane-8',3''-indole]-2,2''-dione.

  Acta crystallographica. Section E, Structure reports online 20120601

• 5,5''-Dibromo-1,1''-bis-(prop-2-en-1-yl)-1,1'',2,2''-tetra-hydro-dispiro-[indole-3,7'-[6,9]diaza-tricyclo-[7.3.0.0(2,6)]dodecane-8',3''-indole]-2,2''-dione.

  Acta crystallographica. Section E, Structure reports online 20120601

• 1,1'-Dibenzyl-5,5''-dichloro-1,1'',2,2''-tetra-hydro-dispiro-[indole-3,7'-[6,9]diaza-tricyclo-[7.3.0.0(2,6)]dodecane-8',3''-indole]-2,2''-dione.

  Acta crystallographica. Section E, Structure reports online 20120601

• Photoswitchable nanoparticles for triggered tissue penetration and drug delivery.

  Journal of the American Chemical Society 20120530

• Photovoltaic characteristics and dye regeneration kinetics in D149-sensitized ZnO with varied dye loading and film thickness.

  Physical chemistry chemical physics : PCCP 20120528

• What is the 'best' atomic charge model to describe through-space charge-transfer excitations?

  Physical chemistry chemical physics : PCCP 20120428

• Efficient construction of fused indolines with a 2-quaternary center via an intramolecular Heck reaction with a low catalyst loading.

  Organic letters 20120420

• Catalytic enantioselective alkene aminohalogenation/cyclization involving atom transfer.

  Angewandte Chemie (International ed. in English) 20120416

• Arynes and cyclohexyne in natural product synthesis.

  Angewandte Chemie (International ed. in English) 20120416

• Total synthesis of (-)-herbindoles A, B, and C via transition-metal-catalyzed intramolecular [2 + 2 + 2] cyclization between ynamide and diynes.

  Organic letters 20120406

• Characterization of 1-(2-[18F] fluoro-3-pyridyl)-4-(2-isopropyl-1-oxo- isoindoline-5-yl)-5-methyl-1H-1,2,3-triazole, a PET ligand for imaging the metabotropic glutamate receptor type 1 in rat and monkey brains.

  Journal of neurochemistry 20120401

• Organic photosensitizers with a heteroleptic dual donor for dye-sensitized solar cells.

  Journal of nanoscience and nanotechnology 20120401

• Construction of polycyclic spiro-indolines via an intramolecular oxidative coupling/cyclization cascade reaction process.

  Organic letters 20120316

• Design of NIR-absorbing simple asymmetric squaraine dyes carrying indoline moieties for use in dye-sensitized solar cells with Pt-free electrodes.

  Organic letters 20120302

• High-performance plastic dye-sensitized solar cells based on low-cost commercial P25 TiO2 and organic dye.

  ACS applied materials & interfaces 20120301

• Rapid access to polycyclic indolines related to the stephacidin alkaloids using a radical cascade.

  Chemical communications (Cambridge, England) 20120214

• Tandem Rh(III)-catalyzed oxidative acylation of secondary benzamides with aldehydes and intramolecular cyclization: the direct synthesis of 3-hydroxyisoindolin-1-ones.

  Organic letters 20120203

• Highly efficient syntheses of azetidines, pyrrolidines, and indolines via palladium catalyzed intramolecular amination of C(sp3)-H and C(sp2)-H bonds at γ and δ positions.

  Journal of the American Chemical Society 20120111

• Asymmetric synthesis of trans-2,3-disubstituted indoline derivatives.

  The Journal of organic chemistry 20120106

• Preparing photochromic nanofibers and animal cells using a photochromic compound of 1',3',3'-trimethyl-6-nitrospiro (2H-1-benzopyran-2,2'-indoline).

  Colloids and surfaces. B, Biointerfaces 20120101

• Three-component reaction discovery enabled by mass spectrometry of self-assembled monolayers.

  Nature chemistry 20120101

• 3'-[Hy-droxy(4-oxo-4H-chromen-3-yl)meth-yl]-2-oxospiro-[indoline-3,2'-pyrrolidine]-3'-carbonitrile.

  Acta crystallographica. Section E, Structure reports online 20120101

• 6-Chloro-1-methyl-indoline-2,3-dione.

  Acta crystallographica. Section E, Structure reports online 20120101

• 4-Chloro-1-methyl-indoline-2,3-dione.

  Acta crystallographica. Section E, Structure reports online 20120101

• Spiroindolines identify the vesicular acetylcholine transporter as a novel target for insecticide action.

  PloS one 20120101

• Chiral aminophosphines as catalysts for enantioselective double-Michael indoline syntheses.

  Molecules (Basel, Switzerland) 20120101

• Density functional theory (DFT) study of triphenylamine-based dyes for their use as sensitizers in molecular photovoltaics.

  International journal of molecular sciences 20120101

• Enantioselective total syntheses of communesins A and B.

  Angewandte Chemie (International ed. in English) 20111209

• A novel metal-free panchromatic TiO2 sensitizer based on a phenylenevinylene-conjugated unit and an indoline derivative for highly efficient dye-sensitized solar cells.

  Chemical communications (Cambridge, England) 20111207

• 1-Benzyl-6-chloro-indoline-2,3-dione.

  Acta crystallographica. Section E, Structure reports online 20111201

• Ultrafast photoinduced relaxation dynamics of the indoline dye D149 in organic solvents.

  Physical chemistry chemical physics : PCCP 20111121

• Solvent-free, microwave-assisted N-arylation of indolines by using low palladium catalyst loadings.

  ChemSusChem 20111118

• Enantioselective synthesis of 2-methyl indolines by palladium catalysed asymmetric C(sp3)-H activation/cyclisation.

  Chemical communications (Cambridge, England) 20111107

• An unexpected C-C cleavage reaction: new and mild access to o-OH and o-NH-Tos benzoic acids or benzoamides.

  Molecular diversity 20111101

• Development of solid, dosage forms of medicinal drugs from indoline group alkaloids.

  Georgian medical news 20111101

• (E)-3-(1-Phenyl-ethyl-idene)indolin-2-one.

  Acta crystallographica. Section E, Structure reports online 20111101

• 2-(3-Cyano-4-{7-[1-(2-hy-droxy-eth-yl)-3,3-dimethyl-indolin-2-yl-idene]hepta-1,3,5-trien-yl}-5,5-dimethyl-2,5-dihydro-furan-2-yl-idene)malononitrile.

  Acta crystallographica. Section E, Structure reports online 20111101

• 3'-(4-Chloro-benzo-yl)-4'-(4-chloro-phen-yl)-1'-methyl-spiro-[indoline-3,2'-pyrrolidin]-2-one.

  Acta crystallographica. Section E, Structure reports online 20111101

• Biocatalysed halogenation of nucleobase analogues.

  Biotechnology letters 20111001

• Isocyanide insertion and cyclization reactions to form indolines using pincer-type complexes of scandium.

  Dalton transactions (Cambridge, England : 2003) 20110921

• QM and QM/MD simulations of the Vinca alkaloids docked to tubulin.

  Journal of molecular graphics & modelling 20110901

• Cyclization vs. cyclization/dimerization in o-amidostilbene radical cation cascade reactions: the amide question.

  Molecules (Basel, Switzerland) 20110825

• Samarium diiodide induced cyclizations of γ-, δ- and ε-indolyl ketones: reductive coupling, intermolecular trapping, and subsequent transformations of indolines.

  Chemistry (Weinheim an der Bergstrasse, Germany) 20110822

• Flustramine inspired synthesis and biological evaluation of pyrroloindoline triazole amides as novel inhibitors of bacterial biofilms.

  Organic & biomolecular chemistry 20110807

• 3-(Diphenyl-methyl-idene)indolin-2-one.

  Acta crystallographica. Section E, Structure reports online 20110801

• Synthesis of 3-(aminomethylene)-2-oxoindolines by palladium-catalyzed annulation of 3-chloro-2-iodo-N-arylacrylamides with amides or amines.

  Chemical communications (Cambridge, England) 20110728

• Straightforward four-component access to spiroindolines.

  Chemical communications (Cambridge, England) 20110728

• Stereoselective synthesis of tetracyclic indolines via gold-catalyzed cascade cyclization reactions.

  Chemical communications (Cambridge, England) 20110721

• Divergent synthesis of unsymmetrical annulated biheterocyclic compound libraries: benzimidazole linked indolo-benzodiazepines/quinoxaline.

  ACS combinatorial science 20110711

• CH activation and CH2 double activation of indolines by radical translocation: understanding the chemistry of the indolinyl radical.

  Organic & biomolecular chemistry 20110707

• 3-(Hetero)aryl-4-indolylamino-α-tetralones by diastereoselective internal redox cyclization: an 'azaenamine' conjugate addition.

  The Journal of organic chemistry 20110701

• 5-Fluoro-1-(4-meth-oxy-benz-yl)indoline-2,3-dione.

  Acta crystallographica. Section E, Structure reports online 20110701

• Microwave-assisted solution-phase synthesis and DART-mass spectrometric monitoring of a combinatorial library of indolin-2,3-dione schiff bases with potential antimycobacterial activity.

  Molecules (Basel, Switzerland) 20110622

• Total synthesis of indoline alkaloids: A cyclopropanation strategy.

  Accounts of chemical research 20110621

• An efficient approach to fused indolines via a copper(I)-catalyzed reaction of sulfonyl azide with 2-ethynylaryl methylenecyclopropane.

  Organic letters 20110617

• Comparison of the SOD-like activity of hexacoordinate Mn(II), Fe(II) and Ni(II) complexes having isoindoline-based ligands.

  Journal of inorganic biochemistry 20110601

• Predicting binding to p-glycoprotein by flexible receptor docking.

  PLoS computational biology 20110601

• (S)-2-(1-Methyl-indolin-2-yl)-1,3-diphenyl-propan-2-ol.

  Acta crystallographica. Section E, Structure reports online 20110601

• Molecular engineering and theoretical investigation of organic sensitizers based on indoline dyes for quasi-solid state dye-sensitized solar cells.

  Physical chemistry chemical physics : PCCP 20110521

• Isolation and identification of five impurities of ALB 109564(a) drug substance.

  Journal of pharmaceutical and biomedical analysis 20110515

• Metal-ligand bifunctional activation and transfer of N-H bonds.

  Chemical communications (Cambridge, England) 20110507

• Palladium-catalyzed cascade reaction for the synthesis of substituted isoindolines.

  Angewandte Chemie (International ed. in English) 20110502

• 4-tert-Butyl-2-[2-(1,3,3-trimethyl-indolin-2-yl-idene)ethyl-idene]cyclo-hexa-none.

  Acta crystallographica. Section E, Structure reports online 20110501

• Soluble polymer supported divergent synthesis of tetracyclic benzene-fused pyrazino/diazepino indoles: an advanced synthetic approach to bioactive scaffolds.

  Organic & biomolecular chemistry 20110421

• Pd(II)-catalyzed intramolecular amidoarylation of alkenes with molecular oxygen as sole oxidant.

  Organic letters 20110415

• Potent inhibitors of hepatitis C core dimerization as new leads for anti-hepatitis C agents.

  Bioorganic & medicinal chemistry letters 20110415

• Dyeing behaviours of amino heterocyclic compounds as blue oxidative hair dye precursors applied to keratin fibres.

  International journal of cosmetic science 20110401

• tert-Butyl 3-benzyl-3-[(E)-2-benzyl-idene-3-oxocyclo-pent-yl]-2-oxoindoline-1-carboxyl-ate.

  Acta crystallographica. Section E, Structure reports online 20110401

• 2-{[(Biphenyl-2-yl)diazen-yl]methyl-idene}-1,3,3-trimethyl-indoline.

  Acta crystallographica. Section E, Structure reports online 20110401

• Thermodynamic analysis of strain in the five-membered oxygen and nitrogen heterocyclic compounds.

  The journal of physical chemistry. A 20110317

• Unexpected synthesis of indolo[1,2-c]quinazolines by a sequential Ugi 4CC-Staudinger-aza-Wittig-nucleophilic addition reaction.

  Organic & biomolecular chemistry 20110307

• Atomic force microscopy-based screening of drug-excipient miscibility and stability of solid dispersions.

  Pharmaceutical research 20110301

• Molybdenum-catalyzed asymmetric allylic alkylation of 3-alkyloxindoles: reaction development and applications.

  Chemistry (Weinheim an der Bergstrasse, Germany) 20110301

• Safety assessment of the pyridoindole derivative SMe1EC2: developmental neurotoxicity study in rats.

  Interdisciplinary toxicology 20110301

• Vinyl diazophosphonates as precursors to quaternary substituted indolines and cyclopentenes.

  Organic letters 20110218

• Redox isomerization via azomethine ylide intermediates: N-alkyl indoles from indolines and aldehydes.

  Organic letters 20110218

• Total synthesis of dictyodendrins A-E.

  Chemistry, an Asian journal 20110201

• 5-Chloro-1-(4-meth-oxy-benz-yl)indoline-2,3-dione.

  Acta crystallographica. Section E, Structure reports online 20110201

• 4-Bromo-3-hy-droxy-3-(4-hy-droxy-2-oxo-2H-chromen-3-yl)indolin-2-one.

  Acta crystallographica. Section E, Structure reports online 20110201

• X-ray and NMR crystallography in an enzyme active site: the indoline quinonoid intermediate in tryptophan synthase.

  Journal of the American Chemical Society 20110112

• ZnO-based dye solar cell with pure ionic-liquid electrolyte and organic sensitizer: the relevance of the dye–oxide interaction in an ionic-liquid medium.

  Physical chemistry chemical physics : PCCP 20110107

• Discovery of isoindoline and tetrahydroisoquinoline derivatives as potent, selective PPARδ agonists.

  Bioorganic & medicinal chemistry letters 20110101

• A novel series of potent and selective EP(4) receptor ligands: facile modulation of agonism and antagonism.

  Bioorganic & medicinal chemistry letters 20110101

• Zebrafish bioassay-guided natural product discovery: isolation of angiogenesis inhibitors from East African medicinal plants.

  PloS one 20110101

• Safety and efficacy of silodosin for the treatment of benign prostatic hyperplasia.

  Clinical interventions in aging 20110101

• Novel ionic liquid with both Lewis and Brønsted acid sites for Michael addition.

  International journal of molecular sciences 20110101

• Indoline-3-carboxylic acid derived organocatalysts for the anti-Mannich reaction.

  Chemistry (Weinheim an der Bergstrasse, Germany) 20101227

• Tandem nucleophilic addition-intramolecular aza-Michael reaction: facile synthesis of chiral fluorinated isoindolines.

  Organic letters 20101203

• Electron transfer properties of organic dye-sensitized solar cells based on indoline sensitizers with ZnO nanoparticles.

  Nanotechnology 20101203

• Tunable hydride transfer in the redox amination of indoline with aldehyde: an attractive intramolecular hydrogen-bond effect.

  Chemistry (Weinheim an der Bergstrasse, Germany) 20101203

• Colorectal cancer-specific cytochrome P450 2W1: intracellular localization, glycosylation, and catalytic activity.

  Molecular pharmacology 20101201

• Electrodeposited nanoporous versus nanoparticulate ZnO films of similar roughness for dye-sensitized solar cell applications.

  ACS applied materials & interfaces 20101201

• (Z)-3-Hydrazinyl-idene-1-phenyl-indolin-2-one.

  Acta crystallographica. Section E, Structure reports online 20101101

• Stereocontrolled creation of all-carbon quaternary stereocenters by organocatalytic conjugate addition of oxindoles to vinyl sulfone.

  Angewandte Chemie (International ed. in English) 20101011

• Hg(OTf)2-BINAPHANE-catalyzed enantioselective anilino sulfonamide allyl alcohol cyclization.

  Chemistry (Weinheim an der Bergstrasse, Germany) 20101004

• Novel indoline-1- or 3,4-dihydroquinoline-1(2H)-substituted carbothiohydrazides as TPO receptor agonists.

  Bioorganic & medicinal chemistry letters 20101001

• Synthesis, cytotoxicity and pro-apoptosis of novel benzoisoindolin hydrazones as anticancer agents.

  Chemical & pharmaceutical bulletin 20101001

• Side reactions of nitroxide-mediated polymerization: N-O versus O-C cleavage of alkoxyamines.

  The journal of physical chemistry. A 20100930

• A comparative study of the binding of QSY 21 and Rhodamine 6G fluorescence probes to DNA: structure and dynamics.

  Physical chemistry chemical physics : PCCP 20100907

• Therapeutic Potential of Plants as Anti-microbials for Drug Discovery.

  Evidence-based complementary and alternative medicine : eCAM 20100901

• (Z)-1-Acetyl-3-[2-oxo-1-phenyl-2-(3-pyrid-yl)ethyl-idene]indolin-2-one.

  Acta crystallographica. Section E, Structure reports online 20100901

• 1'-Acetyl-3-phenyl-6-oxa-4-thia-2-aza-spiro-[bicyclo-[3.2.0]hept-2-ene-7,3'-indolin]-2'-one.

  Acta crystallographica. Section E, Structure reports online 20100901

• Total synthesis of dictyodendrin A and B.

  Angewandte Chemie (International ed. in English) 20100809

• Structure-activity relationship of indoline-2-carboxylic acid N-(substituted)phenylamide derivatives.

  Bioorganic & medicinal chemistry letters 20100801

• (Z)-2-(2-Isopropyl-5-methyl-phen-oxy)-N'-(2-oxoindolin-3-yl-idene)acetohydrazide.

  Acta crystallographica. Section E, Structure reports online 20100701

• 2'-Eth-oxy-1,3,3-trimethyl-spiro-[indoline-2,3'-3H-naphtho-[2,1-b][1,4]oxazine].

  Acta crystallographica. Section E, Structure reports online 20100701

• Cyclopropylazetoindolines as precursors to C(3)-quaternary-substituted indolines.

  Journal of the American Chemical Society 20100623

• Optically induced linking of protein and nanoparticles to gold surfaces.

  Bioconjugate chemistry 20100616

• The discovery and SAR of indoline-3-carboxamides--a new series of 5-HT6 antagonists.

  Bioorganic & medicinal chemistry letters 20100615

• Pd(II)-catalyzed o-C-H acetoxylation of phenylalanine and ephedrine derivatives with MeCOOO(t)Bu/Ac2O.

  Organic letters 20100604

• Spiro-[1,3-dioxolane-2,3'-indolin]-2'-one.

  Acta crystallographica. Section E, Structure reports online 20100601

• Total synthesis of kapakahine E and F.

  Organic letters 20100507

• Design, synthesis, and preliminary biological evaluation of pyrrolo[3,4-c]quinolin-1-one and oxoisoindoline derivatives as aggrecanase inhibitors.

  ChemMedChem 20100503

• One-pot synthesis of substituted isoindolin-1-ones via lithiation and substitution of N'-benzyl-N,N-dimethylureas.

  Chemical communications (Cambridge, England) 20100428

• Gold(I)-catalyzed tandem cyclization approach to tetracyclic indolines.

  Organic letters 20100402

• Methyl 2-acetamido-2-(1-acetyl-3-hydr-oxy-2-oxoindolin-3-yl)propanoate.

  Acta crystallographica. Section E, Structure reports online 20100401

• 1-(Indolin-1-yl)-1-phenyl-3-propan-2-olamines as potent and selective norepinephrine reuptake inhibitors.

  Journal of medicinal chemistry 20100311

• Diphosphine-catalyzed mixed double-Michael reaction: a unified synthesis of indolines, dihydropyrrolopyridines, benzimidazolines, tetrahydroquinolines, tetrahydroisoquinolines, dihydrobenzo-1,4-oxazines, and dihydrobenzo-3,1-oxazines.

  Organic letters 20100305

• Carboxymethylated cyclodextrins and their complexes with Pr(III) and Yb(III) as water-soluble chiral NMR solvating agents for cationic compounds.

  Chirality 20100301

• Regioselective synthesis of heterocycles containing nitrogen neighboring an aromatic ring by reductive ring expansion using diisobutylaluminum hydride and studies on the reaction mechanism.

  The Journal of organic chemistry 20100205

• Chemistry and biological applications of photo-labile organic molecules.

  Chemical Society reviews 20100201

• 3-(Phenyl-imino)indolin-2-one.

  Acta crystallographica. Section E, Structure reports online 20100201

• Aggregation of organic dyes on TiO2 in dye-sensitized solar cells models: an ab initio investigation.

  ACS nano 20100126

• Rhodium-catalyzed [3 + 2] annulation of indoles.

  Journal of the American Chemical Society 20100120

• One-pot, pseudo four-component synthesis of a spiro[diindeno[1,2-b:2',1'-e]pyridine-11,3'-indoline]-trione library.

  Journal of combinatorial chemistry 20100101

• Design and synthesis of orally-active and selective azaindane 5HT2c agonist for the treatment of obesity.

  Bioorganic & medicinal chemistry letters 20100101

• Novel Organotin(IV)-Schiff Base Complexes: Synthesis, Characterization, Antimicrobial Activity, and DNA Interaction Studies.

  Bioinorganic chemistry and applications 20100101

• A TD-DFT investigation of ground and excited state properties in indoline dyes used for dye-sensitized solar cells.

  Physical chemistry chemical physics : PCCP 20091221

• Tryptophan synthase: structure and function of the monovalent cation site.

  Biochemistry 20091124

• Water-soluble calix[4]resorcinarenes as chiral NMR solvating agents for bicyclic aromatic compounds.

  Chirality 20091101

• Nitro-chloromethylbenzindolines: hypoxia-activated prodrugs of potent adenine N3 DNA minor groove alkylators.

  Molecular cancer therapeutics 20091001

• Novel reactivity of dibenzothiophene monooxygenase from Bacillus subtilis WU-S2B.

  Bioscience, biotechnology, and biochemistry 20090901

• Synthesis, ex vivo and in vitro hydrolysis study of an indoline derivative designed as an anti-inflammatory with reduced gastric ulceration properties.

  Molecules (Basel, Switzerland) 20090826

• Intramolecular Ir(I)-catalyzed benzylic C-H bond amination of ortho-substituted aryl azides.

  Organic letters 20090820

• Tricyclic indole and dihydroindole derivatives as new inhibitors of soluble guanylate cyclase.

  Bioorganic & medicinal chemistry letters 20090815

• Novel indoline-based acyl-CoA: cholesterol acyltransferase inhibitor: Effects of introducing a methanesulfonamide group on physicochemical properties and biological activities.

  Bioorganic & medicinal chemistry 20090815

• Pd(II)-catalyzed amination of C-H bonds using single-electron or two-electron oxidants.

  Journal of the American Chemical Society 20090812

• An interrupted Fischer indolization approach toward fused indoline-containing natural products.

  Organic letters 20090806

• Design and synthesis of indole, 2,3-dihydro-indole, and 3,4-dihydro-2H-quinoline-1-carbothioic acid amide derivatives as novel HCV inhibitors.

  Bioorganic & medicinal chemistry letters 20090801

• Novel orally active NPY Y5 receptor antagonists: Synthesis and structure-activity relationship of spiroindoline class compounds.

  Bioorganic & medicinal chemistry 20090715

• Asymmetric synthesis of indolines through intramolecular shifting of aromatic sulfinyl groups. Role of the pi,pi-stacking interactions in these unusual S(N)Ar processes.

  Journal of the American Chemical Society 20090708

• In vitro metabolism of the novel, highly selective oral angiogenesis inhibitor motesanib diphosphate in preclinical species and in humans.

  Drug metabolism and disposition: the biological fate of chemicals 20090701

• Thiourea-catalyzed highly enantio- and diastereoselective additions of oxindoles to nitroolefins: application to the formal synthesis of (+)-physostigmine.

  Journal of the American Chemical Society 20090701

• 5-Bromo-1-methyl-indolin-2-one.

  Acta crystallographica. Section E, Structure reports online 20090701

• 4'-(4-Methoxy-phen-yl)-1,1',1''-trimethyl-dispiro-[indoline-3,2'-pyrrolidine-3',3''-pyrrolidine]-2,2'',5''-trione.

  Acta crystallographica. Section E, Structure reports online 20090701

• 2-(4-{3-[1-(3-Bromo-prop-yl)-3,3-dimethyl-2,3-dihydro-1H-indol-2-yl-idene]prop-1-en-yl}-3-cyano-5,5-dimethyl-2,5-dihydro-furan-2-yl-idene)malononitrile.

  Acta crystallographica. Section E, Structure reports online 20090601

• Stereospecific synthesis of aszonalenins by using two recombinant prenyltransferases.

  Organic & biomolecular chemistry 20090521

• Palladium-catalyzed highly diastereoselective oxidative cascade cyclization reactions.

  Organic letters 20090507

• Differentiating solvation mechanisms at polar solid/liquid interfaces.

  Journal of the American Chemical Society 20090506

• Alkyne-linked 2,2-disubstituted-indolin-3-one oligomers as extended beta-strand mimetics.

  Journal of the American Chemical Society 20090408

• Identification of novel and orally active spiroindoline NPY Y5 receptor antagonists.

  Bioorganic & medicinal chemistry letters 20090315

• Discovery of indoline-based, natural-product-like compounds as probes of focal adhesion kinase signaling pathways.

  Journal of combinatorial chemistry 20090309

• Dehydrogenation of the indoline-containing drug 4-chloro-N-(2-methyl-1-indolinyl)-3-sulfamoylbenzamide (indapamide) by CYP3A4: correlation with in silico predictions.

  Drug metabolism and disposition: the biological fate of chemicals 20090301

• 1-(2,6-Dichloro-phen-yl)indolin-2-one.

  Acta crystallographica. Section E, Structure reports online 20090301

• Palladium-catalyzed annulation of haloanilines and halobenzamides using norbornadiene as an acetylene synthon: a route to functionalized indolines, isoquinolinones, and indoles.

  The Journal of organic chemistry 20090220

• Asymmetric C2-C3 cyclopentannulation of the indole ring.

  Journal of the American Chemical Society 20090218

• 2-[(2,3-dihydro-1H-indol-1-yl)methyl]melatonin analogues: a novel class of MT2-selective melatonin receptor antagonists.

  Journal of medicinal chemistry 20090212

• Glycogen synthase kinase-3 inhibition by 3-anilino-4-phenylmaleimides: insights from 3D-QSAR and docking.

  Journal of computer-aided molecular design 20090201

• (Z)-3-[(E)-3-Phenyl-allyl-idene]indolin-2-one.

  Acta crystallographica. Section E, Structure reports online 20090201

• Acetylaszonalenin biosynthesis in Neosartorya fischeri. Identification of the biosynthetic gene cluster by genomic mining and functional proof of the genes by biochemical investigation.

  The Journal of biological chemistry 20090102

• Synthesis of 2-substituted indoles and indolines via Suzuki-Miyaura coupling/5-endo-trig cyclization strategies.

  The Journal of organic chemistry 20090102

• General approach to the total synthesis of 9-methoxy-substituted indole alkaloids: synthesis of mitragynine, as well as 9-methoxygeissoschizol and 9-methoxy-N(b)-methylgeissoschizol.

  The Journal of organic chemistry 20090102

• Structure-based CoMFA and CoMSIA study of indolinone inhibitors of PDK1.

  Journal of computer-aided molecular design 20090101

• Asymmetric radical and anionic cyclizations of axially chiral carbamates.

  Organic letters 20090101

• Highly efficient and regioselective platinum(II)-catalyzed tandem synthesis of multiply substituted indolines and tetrahydroquinolines.

  Angewandte Chemie (International ed. in English) 20090101

• A study of 3-substituted benzylidene-1,3-dihydro-indoline derivatives as antimicrobial and antiviral agents.

  Zeitschrift fur Naturforschung. C, Journal of biosciences 20090101

• Palladium-catalyzed amidation of unactivated C(sp(3))-H bonds: from anilines to indolines.

  Angewandte Chemie (International ed. in English) 20090101

• Catalytic enantioselective stereoablative alkylation of 3-halooxindoles: facile access to oxindoles with C3 all-carbon quaternary stereocenters.

  Angewandte Chemie (International ed. in English) 20090101

• Catalytic asymmetric 6pi electrocyclization: enantioselective synthesis of functionalized indolines.

  Angewandte Chemie (International ed. in English) 20090101

• Production of H2 from combined endothermic and exothermic hydrogen carriers.

  Journal of the American Chemical Society 20081217

• A high efficiency indoline-sensitized solar cell based on a nanocrystalline TiO(2) surface doped with copper.

  Nanotechnology 20081203

• Experimental and computational study on the molecular energetics of indoline and indole.

  The journal of physical chemistry. A 20081127

• In silico optimization of merocyanine-spiropyran compounds as second-order nonlinear optical molecular switches.

  Physical chemistry chemical physics : PCCP 20081107

• High-conversion-efficiency organic dye-sensitized solar cells with a novel indoline dye.

  Chemical communications (Cambridge, England) 20081107

• Building skeletally diverse architectures on the Indoline Scaffold: the discovery of a chemical probe of focal adhesion kinase signaling networks.

  Bioorganic & medicinal chemistry 20081101

• Ethyl 4'-ethenyl-2'-oxo-4-phenyl-2-(3,4,5-trimethoxy-phen-yl)spiro-[pyrrolidine-3,3'-indoline]-5-carboxyl-ate monohydrate.

  Acta crystallographica. Section E, Structure reports online 20081101

• 1-(3-Chloro-benz-yl)-5-iodo-indoline-2,3-dione.

  Acta crystallographica. Section E, Structure reports online 20081101

• Conversion efficiency versus sensitizer for electrospun TiO(2) nanorod electrodes in dye-sensitized solar cells.

  Nanotechnology 20081022

• Structure and orientation of puroindolines into wheat galactolipid monolayers.

  Langmuir : the ACS journal of surfaces and colloids 20081007

• Titanocene(III)-catalyzed formation of indolines and azaindolines.

  Organic letters 20081002

• Synthesis and biological evaluation of (-)- and (+)-debromoflustramine B and its analogues as selective butyrylcholinesterase inhibitors.

  Journal of medicinal chemistry 20080911

• Synthesis and evaluation of indolinyl- and indolylphenylacetylenes as PET imaging agents for beta-amyloid plaques.

  Bioorganic & medicinal chemistry letters 20080901

• Novel synthesis of cinnolines and 1-aminoindolines via Cu-catalyzed intramolecular N-arylation of hydrazines and hydrazones prepared from 3-haloaryl-3-hydroxy-2-diazopropanoates.

  The Journal of organic chemistry 20080815

• Novel indoline-based acyl-CoA:cholesterol acyltransferase inhibitor with antiperoxidative activity: improvement of physicochemical properties and biological activities by introduction of carboxylic acid.

  Journal of medicinal chemistry 20080814

• 5',6-Dichloro-1',3',3'-trimethyl-spiro-[2H-1-benzopyran-2,2'-indoline].

  Acta crystallographica. Section E, Structure reports online 20080801

• Improved protocol for asymmetric, intramolecular heteroatom Michael addition using organocatalysis: enantioselective syntheses of homoproline, pelletierine, and homopipecolic acid.

  The Journal of organic chemistry 20080704

• Synthesis of indolines via a domino Cu-catalyzed amidation/cyclization reaction.

  Organic letters 20080703

• Facile and general synthesis of quaternary 3-aminooxindoles.

  Organic letters 20080703

• Electronic tera-order stabilization of photoinduced metastable species: structure of the photochromic product of spiropyran determined with in situ single crystal X-ray photodiffraction.

  The journal of physical chemistry. A 20080703

• 1-Acetyl-5,6-dimethoxy-indoline at 123 K.

  Acta crystallographica. Section E, Structure reports online 20080701

• Interplay of hydrogenation and dehydrogenation in isoindoline and indoline isomers: a density functional theory study.

  The journal of physical chemistry. A 20080612

• A highly sensitive and selective chemosensor for cyanide.

  Talanta 20080515

• Palladium-catalyzed intramolecular C-arylation of benzylic carbon: synthesis of 3-benzoxazolylisoindolinones by a sequence of Ugi-4CR/postfunctionalization.

  The Journal of organic chemistry 20080502

• Palladium-catalyzed sp(3) CH activation of simple alkyl groups: direct preparation of indoline derivatives from N-alkyl-2-bromoanilines.

  Organic letters 20080501

• 1-Allyl-3,3-di-p-tolyl-indolin-2-one.

  Acta crystallographica. Section E, Structure reports online 20080501

• Free radical-mediated aryl amination: convergent two- and three-component couplings to chiral 2,3-disubstituted indolines.

  The Journal of organic chemistry 20080418

• Preparation of the isomeric azaindoline family by intramolecular carbolithiation.

  Organic letters 20080320

• A new route to indolines by the Cu-catalyzed cyclization reaction of 2-ethynylanilines with sulfonyl azides.

  Organic letters 20080320

• CYP2D6-Mediated metabolism of a novel acyl coenzyme A:cholesterol acyltransferase inhibitor, pactimibe, and its unique plasma metabolite, R-125528.

  Drug metabolism and disposition: the biological fate of chemicals 20080301

• Studies on the SAR and pharmacophore of milnacipran derivatives as monoamine transporter inhibitors.

  Bioorganic & medicinal chemistry letters 20080215

• Orthogonal synthesis of indolines and isoquinolines via aryne annulation.

  Journal of the American Chemical Society 20080206

• Organic dye-sensitized ionic liquid based solar cells: remarkable enhancement in performance through molecular design of indoline sensitizers.

  Angewandte Chemie (International ed. in English) 20080101

• Reagent-based, modular, tandem Michael approach for obtaining different indoline alkaloid-inspired polycyclic architectures.

  Journal of combinatorial chemistry 20080101

• Gold-catalyzed synthesis of chroman, dihydrobenzofuran, dihydroindole, and tetrahydroquinoline derivatives.

  Chemistry (Weinheim an der Bergstrasse, Germany) 20080101

• Synthesis of indolines and tetrahydroisoquinolines from arylethylamines by Pd(II)-catalyzed C-H activation reactions.

  Angewandte Chemie (International ed. in English) 20080101

• Anionic-anionic asymmetric tandem reactions: one-pot synthesis of optically pure fluorinated indolines from 2-p-tolylsulfinyl alkylbenzenes.

  Angewandte Chemie (International ed. in English) 20080101

• Efficient singlet-state deactivation of cyano-substituted indolines in protic solvents via CN--HO hydrogen bonds.

  Chemphyschem : a European journal of chemical physics and physical chemistry 20071221

• Design, structure-activity relationship, and pharmacokinetic profile of pyrazole-based indoline factor Xa inhibitors.

  Bioorganic & medicinal chemistry letters 20071201

• Potent achiral agonists of the ghrelin (growth hormone secretagogue) receptor. Part I: Lead identification.

  Bioorganic & medicinal chemistry letters 20071201

• One-pot cyclization of 2-aminophenethyl alcohols: a novel and direct approach to the synthesis of N-acyl indolines.

  The Journal of organic chemistry 20071123

• 5'-Phenyl-3'H-spiro[indoline-3,2'-[1,3,4]thiadiazol]-2-one inhibitors of ADAMTS-5 (aggrecanase-2).

  Bioorganic & medicinal chemistry letters 20071015

• Catalytic activation of the leaving group in the S(N)2 reaction.

  Organic letters 20070927

• 1'-Methylcyclooctane-1-spiro-3'-pyrrolidine-2'-spiro-3''-indoline-2,2''-dione and 1,1'-dimethylpiperidine-3-spiro-3'-pyrrolidine-2'-spiro-3''-indoline-2'',4-dione.

  Acta crystallographica. Section C, Crystal structure communications 20070901

• Acido-triggered nonlinear optical switches: benzazolo-oxazolidines.

  The journal of physical chemistry. B 20070823

• Strategies for the synthesis of 2-substituted indoles and indolines starting from acyclic alpha-phosphoryloxy enecarbamates.

  Organic letters 20070816

• Dehydrogenation of indoline by cytochrome P450 enzymes: a novel 'aromatase' process.

  The Journal of pharmacology and experimental therapeutics 20070801

• Practical synthesis of 7-prenylindole.

  The Journal of organic chemistry 20070720

• Synthesis of substituted 1,2-dihydroquinolines and quinolines from aromatic amines and alkynes by gold(I)-catalyzed tandem hydroamination-hydroarylation under microwave-assisted conditions.

  Organic letters 20070705

• Synthesis and properties of novel porphyrin spin probes containing isoindoline nitroxides.

  Free radical biology & medicine 20070701

• Selective inhibition of carboxylesterases by isatins, indole-2,3-diones.

  Journal of medicinal chemistry 20070419

• Polyhydroxylated indolines and oxindoles from C-glycosides via sequential Henry reaction, Michael addition, and reductive amination/amidation.

  The Journal of organic chemistry 20070330

• Indoline derivatives II: synthesis and factor Xa (FXa) inhibitory activities.

  Chemical & pharmaceutical bulletin 20070301

• Lead optimization of [(S)-gamma-(arylamino)prolyl]thiazolidine focused on gamma-substituent: Indoline compounds as potent DPP-IV inhibitors.

  Bioorganic & medicinal chemistry 20070115

• Non-metathesis reactions of ruthenium carbene catalysts and their application to the synthesis of nitrogen-containing heterocycles.

  Chemical record (New York, N.Y.) 20070101

• New procedure to mask the 2,3-pi bond of the indole nucleus and its application to the preparation of potent opioid receptor agonists with a Corynanthe skeleton.

  Organic letters 20061207

• Exploration of the diketoacid integrase inhibitor chemotype leading to the discovery of the anilide-ketoacids chemotype.

  Bioorganic & medicinal chemistry letters 20061115

• Kinetic resolutions of indolines by a nonenzymatic acylation catalyst.

  Journal of the American Chemical Society 20061108

• Studies in sigmatropic rearrangements of N-prenylindole derivatives--a formal enantiomerically pure synthesis of tryprostatin B.

  Organic & biomolecular chemistry 20061107

• Biophysical characterization of an indolinone inhibitor in the ATP-binding site of DNA gyrase.

  Biochemical and biophysical research communications 20061103

• DNA interstrand crosslinking agents: synthesis, DNA interactions, and cytotoxicity of dimeric achiral seco-amino-CBI and conjugates of achiral seco-amino-CBI with pyrrolobenzodiazepine (PBD).

  Bioorganic & medicinal chemistry letters 20061101

• A metal-free approach to the synthesis of indoline derivatives by a phenyliodine(III) bis(trifluoroacetate)-mediated amidohydroxylation reaction.

  The Journal of organic chemistry 20061013

• [Asymmetric intramolecular conjugate addition of chiral enolates via non-equilibrium].

  Yakugaku zasshi : Journal of the Pharmaceutical Society of Japan 20060801

• [Recent advances in the study of pharmacological activities and solid-phase synthesis of indoles and their analogues].

  Yao xue xue bao = Acta pharmaceutica Sinica 20060801

• A phase I study with oral SU5416 in patients with advanced solid tumors: a drug inducing its clearance.

  Investigational new drugs 20060701

• 2-thioindoles as precursors to spiro-fused indolines: synthesis of (+/-)-dehaloperophoramidine.

  Angewandte Chemie (International ed. in English) 20060626

• Efficient synthesis of achiral seco-cyclopropylbenz[2,3-e]indoline analogues: [4-amino-2-(5,6,7-trimethoxyindole-2-carboxamido)naphthalen-1-yl]ethyl chloride and [4-hydroxy-2-(5,6,7-trimethoxyindole-2-carboxamido)naphthalen-1-yl]ethyl chloride.

  The Journal of organic chemistry 20060609

• Preparation of 7-Halo-indoles by Thallation of N-formylindoline and their attempted use for synthesis of the right-hand segment of chloropeptin.

  Chemical & pharmaceutical bulletin 20060601

• Synthesis of tricyclic pyrano[2,3-e]isoindolin-3-ones as the core structure of stachybotrin A, B, and C.

  Chemical communications (Cambridge, England) 20060514

• Design and synthesis of 8-octyl-benzolactam-V9, a selective activator for protein kinase C epsilon and eta.

  Journal of medicinal chemistry 20060504

• Pd(II)-catalyzed enantioselective oxidative tandem cyclization reactions. Synthesis of indolines through C-N and C-C bond formation.

  Journal of the American Chemical Society 20060315

• Indoline derivatives I: synthesis and factor Xa (FXa) inhibitory activities.

  Chemical & pharmaceutical bulletin 20060201

• Chromogenic oxazines for cyanide detection.

  The Journal of organic chemistry 20060120

• Synthesis and antiproliferative activities of diversely substituted glycosyl-isoindigo derivatives.

  European journal of medicinal chemistry 20060101

• Solution- and solid-phase, modular approaches for obtaining different natural product-like polycyclic architectures from an aminoindoline scaffold for combinatorial chemistry.

  Journal of combinatorial chemistry 20060101

• Synergistic effects on escape of a ligand from the closed tryptophan synthase bienzyme complex.

  Biochemistry 20051227

• Scope and mechanistic study of the ruthenium-catalyzed ortho-C-H bond activation and cyclization reactions of arylamines with terminal alkynes.

  Journal of the American Chemical Society 20051207

• Inhibitors of tripeptidyl peptidase II. 3. Derivation of butabindide by successive structure optimizations leading to a potential general approach to designing exopeptidase inhibitors.

  Journal of medicinal chemistry 20051117

• Synthesis, structure and DNA interaction of cobalt(III) bis-complexes of 1,3-bis(2-pyridylimino)isoindoline and 1,4,7-triazacyclononane.

  Journal of inorganic biochemistry 20051101

• A domino amidation route to indolines and indoles: rapid syntheses of anhydrolycorinone, hippadine, oxoassoanine, and pratosine.

  Organic letters 20051013

• Fast and stable photochromic oxazines.

  The Journal of organic chemistry 20050930

• Indole- and indoline-based kainate analogues with antagonist activity at ionotropic glutamate receptors.

  Bioorganic & medicinal chemistry letters 20050901

• Synthesis of 4-(1-oxo-isoindoline) and 4-(5,6-dimethoxy-1-oxo-isoindoline)-substituted phenoxypropanolamines and their beta1-, beta2-adrenergic receptor binding studies.

  Bioorganic chemistry 20050801

• Scavenging of reactive oxygen species by novel indolin-2-one and indoline-2-thione derivatives.

  Biopolymers 20050701

• Amino acid promoted CuI-catalyzed C-N bond formation between aryl halides and amines or N-containing heterocycles.

  The Journal of organic chemistry 20050624

• Prediction of genotoxicity of chemical compounds by statistical learning methods.

  Chemical research in toxicology 20050601

• Design and synthesis of subtype-selective cyclooxygenase (COX) inhibitors derived from thalidomide.

  Bioorganic & medicinal chemistry 20050502

• Molecular diversity via amino acid derived alpha-amino nitriles: synthesis of spirocyclic 2,6-dioxopiperazine derivatives.

  The Journal of organic chemistry 20050429

• A concise stereoselective route to the indoline spiroaminal framework of neoxaline and oxaline.

  Organic letters 20050303

• Solvent-dependent vibrational frequencies and reorganization energies of two merocyanine chromophores.

  The journal of physical chemistry. A 20050303

• Stereoselective synthesis of E-64 and related cysteine proteases inhibitors from 2,3-epoxyamides.

  Bioorganic & medicinal chemistry 20050301

• Stereocontrolled solid-phase synthesis of a 90-membered library of indoline-alkaloid-like polycycles from an enantioenriched aminoindoline scaffold.

  Angewandte Chemie (International ed. in English) 20050218

• Regio- and stereoselective synthesis of isoindolin-1-ones via electrophilic cyclization.

  The Journal of organic chemistry 20050218

• Novel isoindoline compounds for potent and selective inhibition of prolyl dipeptidase DPP8.

  Bioorganic & medicinal chemistry letters 20050201

• The diastereoselective synthesis of quaternary substituted thioindolines from sulfur ylide intermediates.

  The Journal of organic chemistry 20050121

• Asymmetric synthesis of a prostaglandin D2 receptor antagonist.

  The Journal of organic chemistry 20050107

• Regioselective glycosylation: synthesis of alpha-indoline nucleosides.

  Nucleosides, nucleotides & nucleic acids 20050101

• Design, synthesis and evaluation of bicyclic benzamides as novel 5-HT1F receptor agonists.

  Bioorganic & medicinal chemistry letters 20041220

• The design and enzyme-bound crystal structure of indoline based peptidomimetic inhibitors of hepatitis C virus NS3 protease.

  Journal of medicinal chemistry 20041216

• Asymmetric synthesis of pyrrolidinoindolines. Application for the practical total synthesis of (-)-phenserine.

  Journal of the American Chemical Society 20041103

• Conformational insights into furo- and thieno[2,3-b]indolines derived from coupling constants and molecular modeling.

  Magnetic resonance in chemistry : MRC 20041101

• High efficiency of dye-sensitized solar cells based on metal-free indoline dyes.

  Journal of the American Chemical Society 20041006

• A new indolinepeptide from Paecilomyces sp. J300.

  Archives of pharmacal research 20040601

• Synthesis of phakellistatin 13 and oxidation to phakellistatin 3 and isophakellistatin 3.

  Organic letters 20040527

• Indoline derivatives as 5-HT(2C) receptor agonists.

  Bioorganic & medicinal chemistry letters 20040503

• Synthesis and evaluation of some new spiro indoline-based heterocycles as potentially active antimicrobial agents.

  Bioorganic & medicinal chemistry 20040501

• Structure determination of tetrahydroquinazoline antifolates in complex with human and Pneumocystis carinii dihydrofolate reductase: correlations between enzyme selectivity and stereochemistry.

  Acta crystallographica. Section D, Biological crystallography 20040401

• Novel non-peptidic neuropeptide Y Y2 receptor antagonists.

  Bioorganic & medicinal chemistry letters 20040308

• Spirobipyridopyrans, spirobinaphthopyrans, indolinospiropyridopyrans, indolinospironaphthopyrans and indolinospironaphtho-1,4-oxazines: synthesis, study of X-ray crystal structure, antitumoral and antiviral evaluation.

  Bioorganic & medicinal chemistry 20040301

• Unexpected syntheses of seco-cyclopropyltetrahydroquinolines - from a radical 5-exo-trig cyclization reaction: analogs of CC-1065 and the duocarmycins.

  Molecules (Basel, Switzerland) 20040227

• Highly-efficient metal-free organic dyes for dye-sensitized solar cells.

  Chemical communications (Cambridge, England) 20031221

• Aptamers switch on fluorescence of triphenylmethane dyes.

  Journal of the American Chemical Society 20031203

• The effect of remote chirality on the antibacterial activity of indolinyl, tetrahydroquinolyl and dihydrobenzoxazinyl oxazolidinones.

  Bioorganic & medicinal chemistry letters 20031201

• A convergent synthetic approach to the nucleoside-type liposidomycin antibiotics.

  Organic letters 20031016

• Stereospecific construction of contiguous quaternary and tertiary stereocenters by rearrangement from indoline-2-methanol to 2,2,3-trisubstituted tetrahydroquinoline: application to an efficient total synthesis of natural virantmycin.

  Angewandte Chemie (International ed. in English) 20030606

• Total synthesis of the duocarmycins.

  Journal of the American Chemical Society 20030604

• Preparation and pharmacological profile of 7-(alpha-azolylbenzyl)-1H-indoles and indolines as new aromatase inhibitors.

  Bioorganic & medicinal chemistry letters 20030505

• Cardioselective anti-ischemic ATP-sensitive potassium channel (KATP) openers: benzopyranyl indoline and indole analogues.

  European journal of medicinal chemistry 20030501

• Synthesis of 6H-pyrrolo[3',4':2,3][1,4]diazepino[6,7,1-hi]indole-8,10(7H,9H)-diones using 3-bromo-4-(indol-1-yl)maleimide scaffold.

  Organic & biomolecular chemistry 20030307

• Sulfur ylide-initiated thio-claisen rearrangements. The synthesis of highly substituted indolines.

  The Journal of organic chemistry 20030207

• Novel strategies for the solid phase synthesis of substituted indolines and indoles.

  Bioorganic & medicinal chemistry 20030206

• The reaction of cyclic carbinol amides with triflic anhydride as a method to prepare alpha-trifluoromethyl-sulfonamido furans.

  Organic letters 20030123

• Free radical-mediated aryl amination and its use in a convergent [3 + 2] strategy for enantioselective indoline alpha-amino acid synthesis.

  Journal of the American Chemical Society 20030108

• Indoline and piperazine containing derivatives as a novel class of mixed D(2)/D(4) receptor antagonists. Part 1: identification and structure-activity relationships.

  Bioorganic & medicinal chemistry letters 20021104

• Indoline and piperazine containing derivatives as a novel class of mixed D(2)/D(4) receptor antagonists. Part 2: asymmetric synthesis and biological evaluation.

  Bioorganic & medicinal chemistry letters 20021104

• Novel furano analogues of duocarmycin C1 and C2: design, synthesis, and biological evaluation of seco-iso-cyclopropylfurano[2,3-e]indoline (seco-iso-CFI) and seco-cyclopropyltetrahydrofurano[2,3-f]quinoline (seco-CFQ) analogues.

  Bioorganic & medicinal chemistry 20020901

• A convergent approach to 3-substituted-5-methoxyindoles. Application to the synthesis of melatonin [correction].

  Chemical communications (Cambridge, England) 20020821

• Intermediate trapping via a conformational switch in the Na(+)-activated tryptophan synthase bienzyme complex.

  Biochemistry 20020806

• A new strychnobrasiline base of Strychnos mattogrossensis.

  Natural product letters 20020801

• Nature of non-radiative processes involved in the excited state of 9-cyanoanthracene in presence of 2-methylindole/2-methylindoline quenchers. A laser flash photolysis study to reveal the medium effects.

  Spectrochimica acta. Part A, Molecular and biomolecular spectroscopy 20020601

• Antimicrobial activities of a new schizozygane indoline alkaloid from Schizozygia coffaeoides and the revised structure of isoschizogaline.

  Journal of natural products 20020401

• Erythropoietin mimetics derived from solution phase combinatorial libraries.

  Journal of the American Chemical Society 20020130

• Theoretical elucidation on structure-antioxidant activity relationships for indolinonic hydroxylamines.

  Bioorganic & medicinal chemistry letters 20020121

• Design, synthesis, and biological activity of diiminoisoindolines as complement component 3a antagonists.

  Bioorganic & medicinal chemistry letters 20011105

• Multiple mutations at the active site of naphthalene dioxygenase affect regioselectivity and enantioselectivity.

  Journal of industrial microbiology & biotechnology 20010801

• The discovery of linezolid, the first oxazolidinone antibacterial agent.

  Current drug targets. Infectious disorders 20010801

• Asymmetric synthesis of novel isoindolines: azasaccharide mimics as potential enzyme inhibitors.

  The Journal of pharmacy and pharmacology 20010701

• Beta D305A mutant of tryptophan synthase shows strongly perturbed allosteric regulation and substrate specificity.

  Biochemistry 20010626

• A new and general synthetic pathway to strychnos indole alkaloids: total syntheses of (-)-dehydrotubifoline and (-)-tubifoline by palladium-catalyzed asymmetric allylic substitution.

  Organic letters 20010614

• A novel series of thromboxane A2 synthetase inhibitors with free radical scavenging and anti-peroxidative activities.

  Chemical & pharmaceutical bulletin 20010501

• N-Aminoindoline derivatives as inhibitors of 5-lipoxygenase.

  Bioorganic & medicinal chemistry letters 20010326

• 1-Nitroindoline.

  Acta crystallographica. Section C, Crystal structure communications 20010301

• Human beta3 adrenergic receptor agonists containing cyanoguanidine and nitroethylenediamine moieties.

  Bioorganic & medicinal chemistry letters 20010212

• Trapping of the putative cationic intermediate in the Morin rearrangement with carbon nucleophiles.

  The Journal of organic chemistry 20010209

• [[Intramolecular alkylation of aromatic compounds. 35. Di- and tetrahydropyridinemethylindolines as potential precursors of ergolines] ].

  Die Pharmazie 20010101