52-52-8 | Cycloleucine

Packsize	Purity	Availability	Price	Discounted Price
1g	98%	in stock	$13.00	$9.00
5g	98%	in stock	$20.00	$14.00
10g	98%	in stock	$28.00	$19.00
25g	98%	in stock	$60.00	$42.00
100g	98%	in stock	$239.00	$167.00

Description

• Catalog Number: AB45808
• Chemical Name: Cycloleucine
• CAS Number: 52-52-8
• Molecular Formula: C6H11NO2
• Molecular Weight: 129.157
• MDL Number: MFCD00001381
• SMILES: OC(=O)C1(N)CCCC1
• NSC Number: 1026

Computed Properties

• Complexity: 127
• Covalently-Bonded Unit Count: 1
• Heavy Atom Count: 9
• Hydrogen Bond Acceptor Count: 3
• Hydrogen Bond Donor Count: 2
• Rotatable Bond Count: 1
• XLogP3: -2.6

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• Activation of metabotropic glutamate receptors induces gamma frequency oscillations in the rat dentate gyrus in vivo.

  Neuropharmacology 20010301

• Task-dependent role for dorsal striatum metabotropic glutamate receptors in memory.

  Learning & memory (Cold Spring Harbor, N.Y.) 20010301

• Upregulation of preprodynorphin and preproenkephalin mRNA expression by selective activation of group I metabotropic glutamate receptors in characterized primary cultures of rat striatal neurons.

  Brain research. Molecular brain research 20010131

• Regional distribution and pharmacological characteristics of [3H]N-acetyl-aspartyl-glutamate (NAAG) binding sites in rat brain.

  Neurochemistry international 20010101

• Slow dorsal-ventral rhythm generator in the lamprey spinal cord.

  Journal of neurophysiology 20010101

• cAMP-dependent presynaptic regulation of spontaneous glycinergic IPSCs in mechanically dissociated rat spinal cord neurons.

  Journal of neurophysiology 20010101

• Sustained L-type calcium currents in dissociated deep dorsal horn neurons of the rat: characteristics and modulation.

  Neuroscience 20010101

• Traumatic injury of cultured astrocytes alters inositol (1,4,5)-trisphosphate-mediated signaling.

  Glia 20010101

• Metabotropic glutamate receptors modify ionotropic glutamate responses in neocortical pyramidal cells and interneurons.

  Experimental brain research 20010101

• Developmental changes in the modulation of cyclic amp accumulation by activation of metabotropic glutamate receptors.

  Polish journal of pharmacology 20010101

• Locomotor activity and accumbens Fos expression driven by ventral hippocampal stimulation require D1 and D2 receptors.

  Neuroscience 19990101

• Behavioral activity of 1S,3R-ACPD, an agonist of metabotropic glutamate receptors.

  Polish journal of pharmacology 19970801

• Pharmacological characterization of 1-aminoindan-1,5-dicarboxylic acid, a potent mGluR1 antagonist.

  The Journal of pharmacology and experimental therapeutics 19970501

• Anti-Candida activity of cispentacin: the active transport by amino acid permeases and possible mechanisms of action.

  Biochemical and biophysical research communications 19930215

• Effects of D-cycloserine and cycloleucine, ligands for the NMDA-associated strychnine-insensitive glycine site, on brain-stimulation reward and spontaneous locomotion.

  Pharmacology, biochemistry, and behavior 19900801