536-71-0 | 4,4'-(Triaz-1-ene-1,3-diyl)dibenzimidamide

Packsize	Purity	Availability	Price	Discounted Price
1g	99%	2 weeks	$26.00	$18.00
5g	99%	2 weeks	$39.00	$27.00
25g	99%	2 weeks	$98.00	$69.00
100g	99%	2 weeks	$345.00	$241.00

Description

• Catalog Number: AB52530
• Chemical Name: 4,4'-(Triaz-1-ene-1,3-diyl)dibenzimidamide
• CAS Number: 536-71-0
• Molecular Formula: C14H15N7
• Molecular Weight: 281.3158
• MDL Number: MFCD00866606
• SMILES: NC(=N)c1ccc(cc1)N/N=N/c1ccc(cc1)C(=N)N

Computed Properties

• Complexity: 390
• Covalently-Bonded Unit Count: 1
• Heavy Atom Count: 21
• Hydrogen Bond Acceptor Count: 5
• Hydrogen Bond Donor Count: 5
• Rotatable Bond Count: 5
• XLogP3: 1.9

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• Residual effect of antibabesial drugs on the live redwater blood vaccines.

  Annals of the New York Academy of Sciences 20021001

• Drug sensitivity of trypanosome populations from cattle in a peri-urban dairy production system in Uganda.

  Acta tropica 20021001

• Lipid-drug-conjugate (LDC) nanoparticles as novel carrier system for the hydrophilic antitrypanosomal drug diminazenediaceturate.

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  Expert opinion on emerging drugs 20020501

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  International journal of antimicrobial agents 20020301

• Inhibition of DNA replication by berenil in plasmids containing Poly(dA)poly(dT) sequences.

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• S-adenosylmethionine decarboxylase from Leishmania donovani. Molecular, genetic, and biochemical characterization of null mutants and overproducers.

  The Journal of biological chemistry 20020222

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  European biophysics journal : EBJ 20020201

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• Inhibition of DNA replication by berenil of bacterial plasmids containing poly(dA)-poly(dT) sequences. 2D gel analysis of replicative intermediates.

  Cellular and molecular biology (Noisy-le-Grand, France) 20020101

• Changes in properties of adenosine transporters in Trypanosoma evansi and modes of selection of resistance to the melaminophenyl arsenical drug, Mel Cy.

  Veterinary parasitology 20011213

• Enhancing effects of anti-CD40 treatment on the immune response of SCID-bovine mice to Trypanosoma congolense infection.

  Journal of leukocyte biology 20011201

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  African health sciences 20010801

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  Biochimica et biophysica acta 20010628

• A simple, high-resolution method for establishing DNA binding affinity and sequence selectivity.

  Journal of the American Chemical Society 20010627

• Standardised tests in mice and cattle for the detection of drug resistance in tsetse-transmitted trypanosomes of African domestic cattle.

  Veterinary parasitology 20010612

• Concentration-dependent inhibition of sheep erythrocyte ghost plasma membrane Ca2+-ATPase activity by Berenil.

  Journal of veterinary pharmacology and therapeutics 20010601

• DNA minor-groove recognition by small molecules.

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• The incidence of new and the prevalence and persistence of recurrent trypanosome infections in cattle in southwest Ethiopia exposed to a high challenge with drug-resistant parasites.

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• A comparative evaluation of parasitological tests and a PCR for Trypanosoma evansi diagnosis in experimentally infected water buffaloes.

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  International journal for parasitology 20010501

• Effect of clindamycin therapy on phagocytic and oxidative activity profiles of spleen mononuclear cells in Babesia rodhaini-infected mice.

  The Journal of veterinary medical science 20010501

• Validation of a polymerase chain reaction assay for monitoring the therapeutic efficacy of diminazene aceturate in trypanosome-infected sheep.

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  Molecular pharmacology 20010301

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  Parasitology international 20010301

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  Veterinary research communications 20010101

• In vitro effect of diamidines on intracellular polyamines of Acanthamoeba polyphaga.

  Drugs under experimental and clinical research 20010101

• Highly potent synthetic polyamides, bisdistamycins, and lexitropsins as inhibitors of human immunodeficiency virus type 1 integrase.

  Molecular pharmacology 19980801

• Linked lexitropsins and the in vitro inhibition of HIV-1 reverse transcriptase RNA-directed DNA polymerization: a novel induced-fit of 3,5 m-pyridyl bisdistamycin to enzyme-associated template-primer.

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  Annals of tropical medicine and parasitology 19961201

• New drug developments for opportunistic infections in immunosuppressed patients: Pneumocystis carinii.

  Journal of medicinal chemistry 19951124

• DNA-binding activity and biological effects of aromatic polyamidines.

  Biochemical pharmacology 19940211

• Efficacy of DL-alpha-difluoromethylornithine in a rat model of Pneumocystis carinii pneumonia.

  Antimicrobial agents and chemotherapy 19880801

• Cationic antitrypanosomal and other antimicrobial agents in the therapy of experimental Pneumocystis carinii pneumonia.

  Antimicrobial agents and chemotherapy 19880601

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