-
Human sex hormone-binding globulin binding affinities of 125 structurally diverse chemicals and comparison with their binding to androgen receptor, estrogen receptor, and α-fetoprotein.
Toxicological sciences : an official journal of the Society of Toxicology 20150201
-
Synthesis of end-functionalized polyacetylenes that contain polar groups by employing well-defined palladium catalysts.
Chemistry (Weinheim an der Bergstrasse, Germany) 20121029
-
Ormeloxifene inhibits osteoclast differentiation in parallel to downregulating RANKL-induced ROS generation and suppressing the activation of ERK and JNK in murine RAW264.7 cells.
Journal of molecular endocrinology 20120601
-
Pharmacokinetic evaluation of toremifene and its clinical implications for the treatment of osteoporosis.
Expert opinion on drug metabolism & toxicology 20120401
-
Evaluation of the OECD (Q)SAR Application Toolbox for the profiling of estrogen receptor binding affinities.
SAR and QSAR in environmental research 20120101
-
Development, characterization, and in vitro evaluation of tamoxifen microemulsions.
Journal of drug delivery 20120101
-
Lipophilic Pt(II) complexes with selective efficacy against cisplatin-resistant testicular cancer cells.
Journal of inorganic biochemistry 20111201
-
Breast cancer medications and vision: effects of treatments for early-stage disease.
Current eye research 20111001
-
Synthesis and characterization of triphenylethylene derivatives with aggregation-induced emission characteristics.
Journal of fluorescence 20110901
-
Piezofluorochromic and aggregation-induced-emission compounds containing triphenylethylene and tetraphenylethylene moieties.
Chemistry, an Asian journal 20110606
-
An integrated bioinformatics approach identifies elevated cyclin E2 expression and E2F activity as distinct features of tamoxifen resistant breast tumors.
PloS one 20110101
-
Sensitization of glioma cells to tamoxifen-induced apoptosis by Pl3-kinase inhibitor through the GSK-3β/β-catenin signaling pathway.
PloS one 20110101
-
Ficus platyphylla promotes fertility in female Rattus norvegicus Wistar strain: a preliminary study.
Reproductive biology and endocrinology : RB&E 20110101
-
Tamoxifen and raloxifene modulate gap junction coupling during early phases of retinoic acid-dependent neuronal differentiation of NTera2/D1 cells.
Cell biology and toxicology 20101201
-
Anti-breast cancer potential of SS1020, a novel antiestrogen lacking estrogenic and genotoxic actions.
International journal of cancer 20101001
-
Estrogen antagonist and development of macular hole.
Korean journal of ophthalmology : KJO 20101001
-
Structure-function relationships of estrogenic triphenylethylenes related to endoxifen and 4-hydroxytamoxifen.
Journal of medicinal chemistry 20100422
-
Selective estrogen receptor modulator (SERM) for the treatment of osteoporosis in postmenopausal women: focus on lasofoxifene.
Clinical interventions in aging 20100101
-
Granulosa cell tumor of the ovary and antecedent of adjuvant tamoxifen use for breast cancer.
World journal of surgical oncology 20100101
-
Female sex hormones mediate the allergic lung reaction by regulating the release of inflammatory mediators and the expression of lung E-selectin in rats.
Respiratory research 20100101
-
Ultrastructural effects of tamoxifen on uterus in rats.
The Tokai journal of experimental and clinical medicine 20090920
-
Lasofoxifene: Evidence of its therapeutic value in osteoporosis.
Core evidence 20090101
-
Bazedoxifene for the prevention of postmenopausal osteoporosis.
Therapeutics and clinical risk management 20081201
-
Selective estrogen receptor modulators: an update on recent clinical findings.
Obstetrical & gynecological survey 20080301
-
Nanoparticles loaded with ferrocenyl tamoxifen derivatives for breast cancer treatment.
International journal of pharmaceutics 20080122
-
Optimizing high-performance liquid chromatography method with fluorescence detection for quantification of tamoxifen and two metabolites in human plasma: application to a clinical study.
Journal of pharmaceutical and biomedical analysis 20080122
-
A mass spectrometric approach for the study of the metabolism of clomiphene, tamoxifen and toremifene by liquid chromatography time-of-flight spectroscopy.
European journal of mass spectrometry (Chichester, England) 20080101
-
By looking back we can see the way forward: enhancing the gains achieved with antihormone therapy.
Breast cancer research : BCR 20080101
-
Tamoxifen accelerates proteasomal degradation of O6-methylguanine DNA methyltransferase in human cancer cells.
International journal of cancer 20071115
-
Practical synthesis of unsymmetrical tetraarylethylenes and their application for the preparation of [triphenylethylene-spacer-triphenylethylene] triads.
The Journal of organic chemistry 20071012
-
Synthesis of 1,1,2-triphenylethylenes and their antiproliferative effect on human cancer cell lines.
Anti-cancer drugs 20071001
-
Tamoxifen stimulates calcium entry into human platelets.
Journal of cardiovascular pharmacology 20071001
-
The differential effects of bisphosphonates, SERMS (selective estrogen receptor modulators), and parathyroid hormone on bone remodeling in osteoporosis.
Clinical interventions in aging 20070301
-
Medicinal chemistry and emerging strategies applied to the development of selective estrogen receptor modulators (SERMs).
Current medicinal chemistry 20070101
-
Estrogenic or antiestrogenic therapies for multiple myeloma?
Molecular cancer 20070101
-
Decursin and decursinol angelate inhibit estrogen-stimulated and estrogen-independent growth and survival of breast cancer cells.
Breast cancer research : BCR 20070101
-
Prediction of estrogen receptor agonists and characterization of associated molecular descriptors by statistical learning methods.
Journal of molecular graphics & modelling 20061101
-
Modulation of estrogen receptor transactivation and estrogen-induced gene expression by ormeloxifene-a triphenylethylene derivative.
Steroids 20061101
-
Fragmentation of 2,2,2-triphenylethoxychlorocarbene: evidence for ultrafast fragmentation-rearrangement in excited diazirines.
Organic letters 20061012
-
Functional inhibition of intestinal and uterine muscles by non-permeant triphenylethylene derivatives.
European journal of pharmacology 20060217
-
Identification of covalent attachment site of antiestrogenic estradiol 11 beta-derivatives on human estrogen receptor alpha ligand-binding domain.
The Journal of steroid biochemistry and molecular biology 20060201
-
[Interactions between radiation and hormonal therapy in breast cancer: simultaneous or sequential treatment].
Orvosi hetilap 20060122
-
Additive growth inhibitory effects of ibandronate and antiestrogens in estrogen receptor-positive breast cancer cell lines.
Breast cancer research : BCR 20060101
-
Effects of tamoxifen on vaginal blood flow and epithelial morphology in the rat.
BMC women's health 20060101
-
Dielectric and shear mechanical alpha and beta relaxations in seven glass-forming liquids.
The Journal of chemical physics 20051215
-
Investigation of radical cation in electrophilic fluorination by ESI-MS.
Organic letters 20050901
-
Synthesis, structure-activity relationships and antagonistic effects in human MCF-7 breast cancer cells of flexible estrogen receptor modulators.
Medicinal chemistry (Shariqah (United Arab Emirates)) 20050701
-
Endometrial K-ras mutations in postmenopausal breast cancer patients treated with adjuvant tamoxifen or toremifene.
Cancer chemotherapy and pharmacology 20050401
-
K-ras mutation in the endometrium of tamoxifen-treated breast cancer patients, with a comparison of tamoxifen and toremifene.
British journal of cancer 20050328
-
Recycling nanoparticles stabilized in water-in-CO2 microemulsions for catalytic hydrogenations.
Langmuir : the ACS journal of surfaces and colloids 20050301
-
Endocrinology and hormone therapy in breast cancer: selective oestrogen receptor modulators and downregulators for breast cancer - have they lost their way?
Breast cancer research : BCR 20050101
-
Selective estrogen receptor modulators inhibit growth and progression of premalignant lesions in a mouse model of ductal carcinoma in situ.
Breast cancer research : BCR 20050101
-
Advances in estrogen receptor biology: prospects for improvements in targeted breast cancer therapy.
Breast cancer research : BCR 20040101
-
Study of 202 natural, synthetic, and environmental chemicals for binding to the androgen receptor.
Chemical research in toxicology 20031001
-
The effect of estradiol in the striatum is blocked by ICI 182,780 but not tamoxifen: pharmacological and behavioral evidence.
Neuroendocrinology 20030401
-
Effects of tamoxifen on ischemia-induced angiogenesis in the mouse lung.
Angiogenesis 20030101
-
Triphenylethylene antiestrogen-induced acute relaxation of mouse duodenal muscle. Possible involvement of Ca2+ channels.
European journal of pharmacology 20020612
-
Tamoxifen and toremifene impair retrieval, but not acquisition, of spatial information processing in mice.
Pharmacology, biochemistry, and behavior 20020501
-
Some coumarins and triphenylethene derivatives as inhibitors of human testes microsomal 17beta-hydroxysteroid dehydrogenase (17beta-HSD type 3): further studies with tamoxifen on the rat testes microsomal enzyme.
Journal of enzyme inhibition and medicinal chemistry 20020401
-
[Selective estrogen receptor modulators (SERMs) in the practice].
Magyar onkologia 20020101
-
The preparation of phenyl-stilbene derivatives using the safety catch linker.
Methods in molecular biology (Clifton, N.J.) 20020101
-
Endocrine manipulation in advanced breast cancer: recent advances with SERM therapies.
Clinical cancer research : an official journal of the American Association for Cancer Research 20011201
-
Future use of selective estrogen receptor modulators and aromatase inhibitors.
Clinical cancer research : an official journal of the American Association for Cancer Research 20011201
-
Okadaic acid-sensitive activation of Maxi Cl(-) channels by triphenylethylene antioestrogens in C1300 mouse neuroblastoma cells.
The Journal of physiology 20011001
-
Molecular classification of estrogens.
Cancer research 20010915
-
Differential SERM activation of the estrogen receptors (ERalpha and ERbeta) at AP-1 sites.
Chemistry & biology 20010501
-
Flexible estrogen receptor modulators: design, synthesis, and antagonistic effects in human MCF-7 breast cancer cells.
Journal of medicinal chemistry 20010329
-
[Synthesis of triphenylethylene with aliphatic cyclic moiety and its antagonism on estrogen receptor].
Yao xue xue bao = Acta pharmaceutica Sinica 20010301
-
Update on endocrine aspects of breast cancer: report from the 23rd San Antonio Breast Cancer Symposium, San Antonio, Texas, USA, 6-9 December 2000.
Breast cancer research : BCR 20010101
-
Selective estrogen receptor modulation: the search for an ideal hormonal therapy for breast cancer.
Cancer investigation 20010101
-
Cone voltage and collision cell collision-induced dissociation study of triphenylethylenes of pharmaceutical interest.
Rapid communications in mass spectrometry : RCM 20010101
-
Estrogen receptor binding affinity and uterotrophic activity of triphenylhaloethylenes.
Journal of steroid biochemistry 19880601
