63-45-6 | N-(5-aminopentan-2-yl)-6-methoxyquinolin-8-amine; bis(phosphoric acid)

Packsize	Purity	Availability	Price	Discounted Price
5g	97%	in stock	$25.00	$17.00
25g	97%	in stock	$73.00	$51.00
100g	97%	in stock	$201.00	$141.00

Description

• Catalog Number: AI54029
• Chemical Name: N-(5-aminopentan-2-yl)-6-methoxyquinolin-8-amine; bis(phosphoric acid)
• CAS Number: 63-45-6
• Molecular Formula: C15H27N3O9P2
• Molecular Weight: 455.33710199999996
• MDL Number: MFCD00013166
• SMILES: OP(=O)(O)O.OP(=O)(O)O.NCCCC(Nc1cc(OC)cc2c1nccc2)C

Computed Properties

• Complexity: 312
• Covalently-Bonded Unit Count: 3
• Heavy Atom Count: 29
• Hydrogen Bond Acceptor Count: 12
• Hydrogen Bond Donor Count: 8
• Rotatable Bond Count: 6
• Undefined Atom Stereocenter Count: 1

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• A case of symptomatic splenic infarction in vivax malaria.

  The Korean journal of parasitology 20070301

• Nature of the main contaminant in the drug primaquine diphosphate: SFC and SFC-MS methods of analysis.

  Journal of pharmaceutical and biomedical analysis 20070219

• When the book is wrong.

  Lancet (London, England) 20070203

• A rare glimpse at the efficacy of primaquine.

  The American journal of tropical medicine and hygiene 20070201

• Regional differences in the response of Plasmodium vivax malaria to primaquine as anti-relapse therapy.

  The American journal of tropical medicine and hygiene 20070201

• Primaquine for preventing relapses in people with Plasmodium vivax malaria.

  The Cochrane database of systematic reviews 20070124

• Self-gelling primaquine-gum arabic conjugate: an injectable controlled delivery system for primaquine.

  Biomacromolecules 20070101

• Operational feasibility of rapid diagnostic kits & blister packs use for malaria control in high transmission areas of Orissa & Chhattisgarh.

  The Indian journal of medical research 20070101

• Primaquine clears submicroscopic Plasmodium falciparum gametocytes that persist after treatment with sulphadoxine-pyrimethamine and artesunate.

  PloS one 20070101

• [Association of methemoglobinemia and glucose-6-phosphate dehydrogenase deficiency in malaria patients treated with primaquine].

  Revista da Sociedade Brasileira de Medicina Tropical 20070101

• Relapsing vivax malaria after 6 months of daily atovaquone/proguanil in Afghanistan: the case for expanded use of primaquine as a causal prophylactic.

  Journal of travel medicine 20070101

• Photophysical properties and photobiological behavior of amodiaquine, primaquine and chloroquine.

  Photochemistry and photobiology 20070101

• A randomized open-label trial of artesunate- sulfadoxine-pyrimethamine with or without primaquine for elimination of sub-microscopic P. falciparum parasitaemia and gametocyte carriage in eastern Sudan.

  PloS one 20070101

• Plasmodium vivax malaria relapses after primaquine prophylaxis.

  Emerging infectious diseases 20061101

• Glucose 6-phosphate dehydrogenase deficiency: from genotype to phenotype.

  Haematologica 20061001

• Efficacy of three chloroquine-primaquine regimens for treatment of Plasmodium vivax malaria in Colombia.

  The American journal of tropical medicine and hygiene 20061001

• Primaquine: report from CDC expert meeting on malaria chemoprophylaxis I.

  The American journal of tropical medicine and hygiene 20060901

• Cost considerations of malaria chemoprophylaxis including use of primaquine for primary or terminal chemoprophylaxis.

  The American journal of tropical medicine and hygiene 20060901

• Safety and tolerability of elubaquine (bulaquine, CDRI 80/53) for treatment of Plasmidium vivax malaria in Thailand.

  The Korean journal of parasitology 20060901

• Prevalence of glucose-6-phosphate dehydrogenase deficiency in U.S. Army personnel.

  Military medicine 20060901

• [Plasmodium vivax malaria: treatment of primary attacks with primaquine, in three different doses, and a fixed dose of chloroquine, Antioquia, Colombia, 2003-2004].

  Biomedica : revista del Instituto Nacional de Salud 20060901

• A simple technique for the detection of anti-malarial drug formulations and their presence in human urine.

  Tanzania health research bulletin 20060901

• Imported non-Plasmodium falciparum malaria: a five-year prospective study in a European referral center.

  The American journal of tropical medicine and hygiene 20060701

• Chloroquine and primaquine: combining old drugs as a new weapon against falciparum malaria?

  Trends in parasitology 20060601

• Cerebral malaria owing to Plasmodium vivax: case report.

  Annals of tropical paediatrics 20060601

• Does gender, food or grapefruit juice alter the pharmacokinetics of primaquine in healthy subjects?

  British journal of clinical pharmacology 20060601

• Lack of sex effect on the pharmacokinetics of primaquine.

  The American journal of tropical medicine and hygiene 20060601

• Pneumocystis pneumonia in people with HIV.

  Clinical evidence 20060601

• Pharmacokinetics of piperaquine after repeated oral administration of the antimalarial combination CV8 in 12 healthy male subjects.

  European journal of clinical pharmacology 20060501

• [Haemolysis due to primaquine in 3 cases].

  Zhongguo ji sheng chong xue yu ji sheng chong bing za zhi = Chinese journal of parasitology & parasitic diseases 20060227

• Do apoptotic Plasmodium-infected hepatocytes initiate protective immune responses?

  The Journal of infectious diseases 20060101

• Are multiple gametocyte infections in malarial parasites an adaptation to ensure fertility?

  Parasitology 20060101

• A randomized, parallel study of the safety and efficacy of 45 mg primaquine versus 75 mg bulaquine as gametocytocidal agents in adults with blood schizonticide-responsive uncomplicated falciparum malaria [ISCRTN50134587].

  BMC infectious diseases 20060101

• [How much primaquine is needed to eradicate Plasmodium vivax hypnozoites?].

  Enfermedades infecciosas y microbiologia clinica 20060101

• Frequency of malaria and glucose-6-phosphate dehydrogenase deficiency in Tajikistan.

  Malaria journal 20060101

• Combined chloroquine, sulfadoxine/pyrimethamine and primaquine against Plasmodium falciparum in Central Java, Indonesia.

  Malaria journal 20060101

• Primaquine-induced hemolytic anemia: role of splenic macrophages in the fate of 5-hydroxyprimaquine-treated rat erythrocytes.

  The Journal of pharmacology and experimental therapeutics 20051201

• A double-blind, randomized study of azithromycin compared to chloroquine for the treatment of Plasmodium vivax malaria in India.

  The American journal of tropical medicine and hygiene 20051201

• A 57-year-old man with a 6-day headache and fatigue.

  The American journal of medicine 20051201

• Failure of primaquine therapy for the treatment of Plasmodium ovale malaria.

  Clinical infectious diseases : an official publication of the Infectious Diseases Society of America 20051115

• Primaquine synergises the activity of chloroquine against chloroquine-resistant P. falciparum.

  Biochemical pharmacology 20051015

• Targeting primaquine into liver using chylomicron emulsions for potential vivax malaria therapy.

  International journal of pharmaceutics 20051013

• Evaluation of anti-malarial effects of mass chemoprophylaxis in the Republic of Korea army.

  Journal of Korean medical science 20051001

• Application of GC-EI-MS for the identification and investigation of positional isomer in primaquine, an antimalarial drug.

  Journal of pharmaceutical and biomedical analysis 20050901

• Plasmodium cynomolgi: gametocytocidal activity of the anti-malarial compound CDRI 80/53 (elubaquine) in rhesus monkeys.

  Experimental parasitology 20050901

• Primaquine-induced hemolytic anemia: role of membrane lipid peroxidation and cytoskeletal protein alterations in the hemotoxicity of 5-hydroxyprimaquine.

  The Journal of pharmacology and experimental therapeutics 20050801

• Pseudo-borreliosis in patients with malaria.

  The American journal of tropical medicine and hygiene 20050701

• Photoreactivity of biologically active compounds. XVII. Influence of solvent interactions on spectroscopic properties and photostability of primaquine.

  Die Pharmazie 20050601

• Pneumocystis pneumonia in people with HIV.

  Clinical evidence 20050601

• Glycodendrimeric nanoparticulate carriers of primaquine phosphate for liver targeting.

  International journal of pharmaceutics 20050513

• Effectiveness of antimalarial drugs.

  The New England journal of medicine 20050414

• A novel incubation direct injection LC/MS/MS technique for in vitro drug metabolism screening studies involving the CYP 2D6 and the CYP 3A4 isozymes.

  Journal of pharmaceutical and biomedical analysis 20050401

• Glucose-6-phosphate dehydrogenase deficiency in two returning Operation Iraqi Freedom soldiers who developed hemolytic anemia while receiving primaquine prophylaxis for malaria.

  Military medicine 20050401

• Differential toxicity of reactive metabolites of clindamycin and sulfonamides in HIV-infected cells: influence of HIV infection on clindamycin toxicity in vitro.

  Journal of clinical pharmacology 20050301

• Imidazolidin-4-one derivatives of primaquine as novel transmission-blocking antimalarials.

  Journal of medicinal chemistry 20050210

• Raising antibodies in chickens against primaquine, pyrimethamine, dapsone, tetracycline, and doxycycline.

  Immunological investigations 20050101

• Diagnostic and prognostic utility of an inexpensive rapid on site malaria diagnostic test (ParaHIT f) among ethnic tribal population in areas of high, low and no transmission in central India.

  BMC infectious diseases 20050101

• Adequate primaquine for vivax malaria.

  Journal of travel medicine 20050101

• Glucose-6-phosphate dehydrogenase (G6PD) mutations in Cambodia: G6PD Viangchan (871G>A) is the most common variant in the Cambodian population.

  Journal of human genetics 20050101

• Antimalarials inhibit human erythrocyte membrane acetylcholinesterase.

  Drug and chemical toxicology 20050101

• Primaquine therapy for malaria.

  Clinical infectious diseases : an official publication of the Infectious Diseases Society of America 20041101

• Randomized trial of 3-dose regimens of tafenoquine (WR238605) versus low-dose primaquine for preventing Plasmodium vivax malaria relapse.

  Clinical infectious diseases : an official publication of the Infectious Diseases Society of America 20041015

• Declining mefloquine sensitivity of Plasmodium falciparum along the Thai-Myanmar border.

  The Southeast Asian journal of tropical medicine and public health 20040901

• Assessment of therapeutic efficacy of chloroquine for vivax malaria in Thailand.

  The Southeast Asian journal of tropical medicine and public health 20040901

• Therapeutic efficacy of artesunate in Plasmodium vivax malaria in Thailand.

  The Southeast Asian journal of tropical medicine and public health 20040901

• Changes in Haemoproteus sex ratios: fertility insurance or differential sex lifespan?

  Proceedings. Biological sciences 20040807

• Enantioselective analysis of primaquine and its metabolite carboxyprimaquine by capillary electrophoresis.

  Electrophoresis 20040801

• PKD1/PKCmu promotes alphavbeta3 integrin recycling and delivery to nascent focal adhesions.

  The EMBO journal 20040707

• A prospective study evaluating the efficacy of a single, 45-mg dose of primaquine, as a gametocytocidal agent, in patients with Plasmodium falciparum malaria in Mumbai, India.

  Annals of tropical medicine and parasitology 20040701

• Preliminary report of the evaluation of the gametocytocidal action of bulaquine, in adult patients with acute, Plasmodium falciparum malaria.

  Annals of tropical medicine and parasitology 20040701

• Plasmepsin II inhibition and antiplasmodial activity of Primaquine-Statine 'double-drugs'.

  Bioorganic & medicinal chemistry letters 20040607

• In vitro and in vivo evaluation of albumin-encapsulated primaquine diphosphate prepared by nebulization into heated oil.

  Journal of microencapsulation 20040601

• Pneumocystis carinii pneumonia treatment in people infected with HIV.

  Clinical evidence 20040601

• Pharmacokinetics of primaquine and carboxyprimaquine in Korean patients with vivax malaria.

  Archives of pharmacal research 20040501

• Kinetic mechanism of quinone oxidoreductase 2 and its inhibition by the antimalarial quinolines.

  Biochemistry 20040420

• Primaquine-induced hemolytic anemia: susceptibility of normal versus glutathione-depleted rat erythrocytes to 5-hydroxyprimaquine.

  The Journal of pharmacology and experimental therapeutics 20040401

• A large focus of naturally acquired Plasmodium knowlesi infections in human beings.

  Lancet (London, England) 20040327

• Synthesis and blood-schizontocidal antimalarial activities of 2-substituted/2,5-disubstituted-8-quinolinamines and some of their amino acid conjugates.

  Bioorganic & medicinal chemistry 20040301

• Compliance with 14-day primaquine therapy for radical cure of vivax malaria--a randomized placebo-controlled trial comparing unsupervised with supervised treatment.

  Transactions of the Royal Society of Tropical Medicine and Hygiene 20040301

• Nature of the main contaminant in the anti malaria drug primaquine diphosphate: a qualitative isomer analysis.

  Journal of chromatography. B, Analytical technologies in the biomedical and life sciences 20040205

• Treatment with antimalarials adversely affects the oxidative energy metabolism in rat liver mitochondria.

  Drug and chemical toxicology 20040201

• CV8, a new combination of dihydroartemisinin, piperaquine, trimethoprim and primaquine, compared with atovaquone-proguanil against falciparum malaria in Vietnam.

  Tropical medicine & international health : TM & IH 20040201

• Discovery of a bulky 2-tert-butyl group containing primaquine analogue that exhibits potent blood-schizontocidal antimalarial activities and complete elimination of methemoglobin toxicity.

  Journal of medicinal chemistry 20040115

• [Cerebral Malaria in Ceará: a case report].

  Revista da Sociedade Brasileira de Medicina Tropical 20040101

• Preparation and in vitro evaluation of primaquine-conjugated gum arabic microspheres.

  Biomacromolecules 20040101

• [Clinical and laboratorial alterations in Plasmodium vivax malaria patients and glucose-6-phosphate dehydrogenase deficiency treated with primaquine at 0.50 mg/kg/day].

  Revista da Sociedade Brasileira de Medicina Tropical 20040101

• Primaquine for prevention of malaria in travelers.

  Clinical infectious diseases : an official publication of the Infectious Diseases Society of America 20031215

• Military aviators, special operations forces, and causal malaria prophylaxis.

  Military medicine 20031201

• HPLC and HPTLC assays for the antimalarial agents chloroquine, primaquine and bulaquine.

  Journal of pharmaceutical and biomedical analysis 20031124

• Transmission-blocking activity of tafenoquine (WR-238605) and artelinic acid against naturally circulating strains of Plasmodium vivax in Thailand.

  The American journal of tropical medicine and hygiene 20031101

• Mechanism of C2-toxin inhibition by fluphenazine and related compounds: investigation of their binding kinetics to the C2II-channel using the current noise analysis.

  Journal of molecular biology 20031024

• Two worlds of malaria.

  The New England journal of medicine 20031016

• Real-time investigation of the interaction between primaquine phosphate and bovine serum albumin (BSA) by piezoelectric quartz crystal impedance analysis.

  Journal of biotechnology 20031009

• Problems in the therapy for imported malaria in the United States.

  Archives of internal medicine 20030922

• Clinical efficacy of chloroquine followed by primaquine for Plasmodium vivax treatment in Azerbaijan.

  Acta tropica 20030901

• Monitoring the therapeutic efficacy of antimalarials against uncomplicated falciparum malaria in Thailand.

  The Southeast Asian journal of tropical medicine and public health 20030901

• Liquid chromatography-tandem mass spectrometric assay with a novel method of quantitation for the simultaneous determination of bulaquine and its metabolite, primaquine, in monkey plasma.

  Journal of chromatography. B, Analytical technologies in the biomedical and life sciences 20030815

• Cooperative actions to achieve malaria control without the use of DDT.

  International journal of hygiene and environmental health 20030801

• Vivax malaria: a continuing health threat to the Republic of Korea.

  The American journal of tropical medicine and hygiene 20030801

• The impact of Malarone and primaquine on psychomotor performance.

  Aviation, space, and environmental medicine 20030701

• Clinical trial of oral artesunate with or without high-dose primaquine for the treatment of vivax malaria in Thailand.

  The American journal of tropical medicine and hygiene 20030701

• Primaquine induced methemoglobinemia.

  Indian journal of pediatrics 20030601

• Correlation between Plasmodium vivax variants in Belém, Pará State, Brazil and symptoms and clearance of parasitaemia.

  The Brazilian journal of infectious diseases : an official publication of the Brazilian Society of Infectious Diseases 20030601

• Binding of primaquine to epidermal membranes and keratin.

  International journal of pharmaceutics 20030512

• The efficacy of combined mefloquine-artesunate versus mefloquine-primaquine on subsequent development of Plasmodium falciparum gametocytemia.

  The American journal of tropical medicine and hygiene 20030501

• Analysis and pharmacokinetics of bulaquine and its major metabolite primaquine in rabbits using an LC-UV method--a pilot study.

  Journal of pharmaceutical and biomedical analysis 20030424

• Presentation by recycling MHC class II molecules of an influenza hemagglutinin-derived epitope that is revealed in the early endosome by acidification.

  Journal of immunology (Baltimore, Md. : 1950) 20030401

• Toxicity related to chloroquine treatment of resistant vivax malaria.

  The Annals of pharmacotherapy 20030401

• Blood schizontocidal activity of WR 238605 (Tafenoquine) against Plasmodium cynomolgi and Plasmodium fragile infections in rhesus monkeys.

  Acta tropica 20030401

• The chemotherapy of rodent malaria. LXI. Drug combinations to impede the selection of drug resistance, part 4: the potential role of 8-aminoquinolines.

  Annals of tropical medicine and parasitology 20030401

• A mathematical model for the transmission of Plasmodium vivax malaria.

  Parasitology international 20030301

• Can primaquine therapy for vivax malaria be improved?

  Trends in parasitology 20030301

• Efficacy of a five-day course of primaquine in preventing relapses in Plasmodium vivax malaria--a pilot study.

  The Ceylon medical journal 20030301

• Case report: An unusual late relapse of Plasmodium vivax malaria.

  The American journal of tropical medicine and hygiene 20030201

• [Antiprotozoal drugs].

  Nihon rinsho. Japanese journal of clinical medicine 20030201

• [Short course schemes for vivax malaria treatment].

  Revista da Sociedade Brasileira de Medicina Tropical 20030101

• [Internal validity of clinical trials for Plasmodium vivax malaria treatment: analysis of evaluation study of in vivo Plasmodium vivax emergence of resistance to standard doses of primaquine].

  Revista da Sociedade Brasileira de Medicina Tropical 20030101

• Efficacy of a 14-day primaquine regimen in preventing relapses in patients with Plasmodium vivax malaria in Mumbai, India.

  Transactions of the Royal Society of Tropical Medicine and Hygiene 20030101

• Effectiveness of primaquine terminal prophylaxis against late primary attacks of Plasmodium vivax malaria: a case-control study among troops of the Republic of Korea army.

  Transactions of the Royal Society of Tropical Medicine and Hygiene 20030101

• Isolation and antimalarial activity of peroxydisulfate oxidation products of primaquine.

  Bioorganic & medicinal chemistry letters 20021216

• Discovery of novel targets of quinoline drugs in the human purine binding proteome.

  Molecular pharmacology 20021201

• Primaquine-induced hemolytic anemia: formation of free radicals in rat erythrocytes exposed to 6-methoxy-8-hydroxylaminoquinoline.

  The Journal of pharmacology and experimental therapeutics 20021201

• Plasmodium ovale malaria acquired in central Spain.

  Emerging infectious diseases 20021201

• The clinical and epidemiological features of childhood malaria in a moderately endemic area of Sri Lanka.

  The Southeast Asian journal of tropical medicine and public health 20021201

• Cytochrome P450 1A1/2 induction by antiparasitic drugs: dose-dependent increase in ethoxyresorufin O-deethylase activity and mRNA caused by quinine, primaquine and albendazole in HepG2 cells.

  European journal of clinical pharmacology 20021101

• Pancytopenia resulting from hemophagocytosis in malaria.

  The Pediatric infectious disease journal 20021101

• Primaquine-induced hemolytic anemia: effect of 6-methoxy-8-hydroxylaminoquinoline on rat erythrocyte sulfhydryl status, membrane lipids, cytoskeletal proteins, and morphology.

  The Journal of pharmacology and experimental therapeutics 20021001

• Radical curative efficacy of five-day regimen of primaquine for treatment of Plasmodium vivax malaria in India.

  The Journal of parasitology 20021001

• Sensitivity of Plasmodium vivax to chloroquine in Sa Kaeo Province, Thailand.

  Acta tropica 20020801

• Does radical cure of asymptomatic Plasmodium falciparum place adults in endemic areas at increased risk of recurrent symptomatic malaria?

  Tropical medicine & international health : TM & IH 20020701

• Recycling CD1d1 molecules present endogenous antigens processed in an endocytic compartment to NKT cells.

  Journal of immunology (Baltimore, Md. : 1950) 20020601

• Coronary bypass surgery in patient with malaria.

  Asian cardiovascular & thoracic annals 20020601

• Short report: therapeutic efficacy of chloroquine combined with primaquine against Plasmodium falciparum in northeastern Papua, Indonesia.

  The American journal of tropical medicine and hygiene 20020601

• Relapsing vivax malaria.

  The Medical journal of Australia 20020520

• Enantiomeric separation of primaquine, an anti-malarial drug, by cyclodextrin-modified micellar electrokinetic capillary chromatography.

  Analytical sciences : the international journal of the Japan Society for Analytical Chemistry 20020501

• Effect of antimalarial drugs on plasmodia cell-free protein synthesis.

  Memorias do Instituto Oswaldo Cruz 20020401

• Relapse pattern of Plasmodium vivax in Mumbai: a study of 283 cases of vivax malaria.

  The Journal of the Association of Physicians of India 20020301

• Methemoglobin reductase activity and in vitro sensitivity towards oxidant induced methemoglobinemia in swiss mice and beagle dogs erythrocytes.

  Molecular and cellular biochemistry 20020301

• Prevalence of malaria in Aligarh.

  The Journal of communicable diseases 20020301

• Inhibition of cardiac Na+ current by primaquine.

  British journal of pharmacology 20020201

• Mutagenic activity and mutational specificity of antiprotozoal drugs with and without nitrite treatment.

  Environmental and molecular mutagenesis 20020101

• Control of malaria: a successful experience from Viet Nam.

  Bulletin of the World Health Organization 20020101

• Comparison of tafenoquine (WR238605) and primaquine in the post-exposure (terminal) prophylaxis of vivax malaria in Australian Defence Force personnel.

  Transactions of the Royal Society of Tropical Medicine and Hygiene 20020101

• Randomized, parallel placebo-controlled trial of primaquine for malaria prophylaxis in Papua, Indonesia.

  Clinical infectious diseases : an official publication of the Infectious Diseases Society of America 20011215

• Effect of primaquine standard dose (15 mg/day for 14 days) in the treatment of vivax malaria patients in Thailand.

  The Southeast Asian journal of tropical medicine and public health 20011201

• Current drugs for antimalarial chemoprophylaxis: a review of efficacy and safety.

  Journal of travel medicine 20011201

• Association of subtherapeutic dosages of a standard drug regimen with failures in preventing relapses of vivax malaria.

  The American journal of tropical medicine and hygiene 20011101

• Plasmodium vivax relapses after 5 days of primaquine treatment, in some industrial complexes of India.

  Annals of tropical medicine and parasitology 20011001

• Plasmodium vivax polymorphism in a clinical drug trial.

  Clinical and diagnostic laboratory immunology 20010901

• Malaria chemoprophylaxis in the age of drug resistance. II. Drugs that may be available in the future.

  Clinical infectious diseases : an official publication of the Infectious Diseases Society of America 20010801

• Plasmodium vivax clinically resistant to chloroquine in Colombia.

  The American journal of tropical medicine and hygiene 20010801

• Malaria chemoprophylaxis in the age of drug resistance. I. Currently recommended drug regimens.

  Clinical infectious diseases : an official publication of the Infectious Diseases Society of America 20010715

• The antileishmanial properties of surface-modified, primaquine-loaded nanocapsules tested against intramacrophagic Leishmania donovani amastigotes in vitro.

  Annals of tropical medicine and parasitology 20010701

• Treating malaria may be too expensive.

  Australian family physician 20010601

• Primaquine-induced hemolytic anemia: formation and hemotoxicity of the arylhydroxylamine metabolite 6-methoxy-8-hydroxylaminoquinoline.

  The Journal of pharmacology and experimental therapeutics 20010501

• Transcriptional and post-translational regulation of CYP1A1 by primaquine.

  The Journal of pharmacology and experimental therapeutics 20010401

• Oxidative stress participates in the breakdown of neuronal phenotype in experimental diabetic neuropathy.

  Diabetologia 20010401

• Functional integrity of the vesicle transporting machinery is required for complete activation of cFTR expressed in xenopus laevis oocytes.

  Pflugers Archiv : European journal of physiology 20010301

• [Does the brief treatment with antimalarials favorably influence drug resistance and recurrences?].

  Revista panamericana de salud publica = Pan American journal of public health 20010301

• Dissociation and electrooxidation of primaquine diphosphate as an approach to the study of anti-chagas prodrugs mechanism of action.

  Bioelectrochemistry (Amsterdam, Netherlands) 20010101

• Immunological alterations associated with Plasmodium vivax malaria in South Korea.

  Annals of tropical medicine and parasitology 20010101

• Antimalarial chemoprophylaxis in infants and children.

  Paediatric drugs 20010101

• [Primaquine].

  Medecine tropicale : revue du Corps de sante colonial 20010101

• Malaria prophylaxis/radical cure: recent experiences of the Australian Defence Force.

  Medecine tropicale : revue du Corps de sante colonial 20010101

• [Effect of daphnetin on the exo-erythrocytic stage of rodent malaria].

  Zhongguo ji sheng chong xue yu ji sheng chong bing za zhi = Chinese journal of parasitology & parasitic diseases 20010101

• [A study of artemether combined with primaquine in the treatment of falciparum malaria].

  Zhongguo ji sheng chong xue yu ji sheng chong bing za zhi = Chinese journal of parasitology & parasitic diseases 20010101

• [Hemolysis and primaquine treatment. Preliminary report].

  Revista cubana de medicina tropical 19970101

• Dapsone- and primaquine-induced methemoglobinemia in HIV-infected individuals.

  Journal of acquired immune deficiency syndromes and human retrovirology : official publication of the International Retrovirology Association 19960815

• [Primaquine and travelers from the Arab world. A report and recommendations].

  Revista cubana de medicina tropical 19950101

• In vitro effects of artemisinin ether, cycloguanil hydrochloride (alone and in combination with sulfadiazine), quinine sulfate, mefloquine, primaquine phosphate, trifluoperazine hydrochloride, and verapamil on Toxoplasma gondii.

  Antimicrobial agents and chemotherapy 19940601

• [Comparative study on hemolytic toxicity of trifluoroacetoprimaquine and primaquine in rabbits].

  Zhongguo ji sheng chong xue yu ji sheng chong bing za zhi = Chinese journal of parasitology & parasitic diseases 19940101

• Acute intravascular haemolysis in Vanuatu following a single dose of primaquine in individuals with glucose-6-phosphate dehydrogenase deficiency.

  The Journal of tropical medicine and hygiene 19921001

• 8-Aminoquinolines from Walter Reed Army Institute for Research for treatment and prophylaxis of Pneumocystis pneumonia in rat models.

  Antimicrobial agents and chemotherapy 19910201

• The effect of primaquine on the ultrastructural morphology of Pneumocystis carinii.

  The Journal of protozoology 19910101

• Detection of antidrug IgG antibodies in patients with adverse drug reactions to amodiaquine.

  International archives of allergy and applied immunology 19910101

• Primaquine induced hemolysis in a Thai soldier.

  The Southeast Asian journal of tropical medicine and public health 19891201

• Activity of clindamycin with primaquine against Pneumocystis carinii in vitro and in vivo.

  Antimicrobial agents and chemotherapy 19880601

• [Hemolytic reaction due to administration of primaquine].

  Zhonghua liu xing bing xue za zhi = Zhonghua liuxingbingxue zazhi 19860401

• Pharmacokinetics of primaquine in man. I. Studies of the absolute bioavailability and effects of dose size.

  British journal of clinical pharmacology 19850601

• Primaquine-chloroquine prophylaxis against malaria in Southeast-Asian refugees entering South Australia.

  The Medical journal of Australia 19840317

• The treatment of malaria in glucose-6-phosphate dehydrogenase deficient patients in Sabah.

  Annals of tropical medicine and parasitology 19811201

• Reaction to primaquine.

  Annals of internal medicine 19800301

• Antimalarial activities of various 4-quinolonemethanols with special attention to WR-142,490 (mefloquine).

  Antimicrobial agents and chemotherapy 19780601

• Hemolysis in dialyzed patients: tap water-induced red blood cell metabolic deficiency.

  Transactions - American Society for Artificial Internal Organs 19720101

• Simultaneous drug reactions in the same patient. Chloroquine-Primaquine sensitivity.

  JAMA 19700427

• Methemoglobinemia provoked by malarial chemoprophylaxis in Vietnam.

  The New England journal of medicine 19681121

• The haemolytic effect of various regimens of primaquine with chloroquine in American Negroes with G6PD deficiency and the lack of an effect of various antimalarial suppressive agents on erythrocyte metabolism.

  Bulletin of the World Health Organization 19670101

• Potentiation of the curative action of primaquine in vivax malaria by quinine and chloroquine.

  The Journal of laboratory and clinical medicine 19550801