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Fetal bovine serum and human constitutive androstane receptor: evidence for activation of the SV23 splice variant by artemisinin, artemether, and arteether in a serum-free cell culture system.
Toxicology and applied pharmacology 20140601
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Synthesis and insight into the structure-activity relationships of chalcones as antimalarial agents.
Journal of medicinal chemistry 20130110
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Bile acid-based 1,2,4-trioxanes: synthesis and antimalarial assessment.
Journal of medicinal chemistry 20121213
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Formulation design and in vivo antimalarial evaluation of lipid-based drug delivery systems for oral delivery of β-arteether.
European journal of pharmaceutics and biopharmaceutics : official journal of Arbeitsgemeinschaft fur Pharmazeutische Verfahrenstechnik e.V 20120901
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Curcuminoids-loaded liposomes in combination with arteether protects against Plasmodium berghei infection in mice.
Experimental parasitology 20120701
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Linker-based hemisuccinate derivatives of artemisinin: synthesis and antimalarial assessment against multidrug-resistant Plasmodium yoelii nigeriensis in mice.
Journal of medicinal chemistry 20120209
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Curcumin-arteether combination therapy of Plasmodium berghei-infected mice prevents recrudescence through immunomodulation.
PloS one 20120101
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Plasmodium vinckei: infectivity of arteether-sensitive and arteether-resistant parasites in different strains of mice.
Parasitology research 20111001
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Neurological assessments after treatment with the antimalarial β-arteether in neonatal and adult rats.
Neurotoxicology 20110801
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A phase III clinical trial of alpha, beta-arteether injection 150 mg/ml in patients of P falciparum malaria.
Journal of the Indian Medical Association 20110801
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Preparation of molecularly imprinted polymers for artemisinin based on the surfaces of silica gel.
Journal of biotechnology 20110420
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Toxicokinetic and toxicodynamic (TK/TD) evaluation to determine and predict the neurotoxicity of artemisinins.
Toxicology 20110111
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Implication of intracellular glutathione and its related enzymes on resistance of malaria parasites to the antimalarial drug arteether.
Parasitology international 20110101
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Synthesis and antimalarial assessment of a new series of orally active amino-functionalized spiro 1,2,4-trioxanes.
Journal of medicinal chemistry 20101111
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Self-microemulsifiyng suppository formulation of β-artemether.
AAPS PharmSciTech 20100901
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6-(4'-Aryloxy-phenyl)vinyl-1,2,4-trioxanes: a new series of orally active peroxides effective against multidrug-resistant Plasmodium yoelii in Swiss mice.
Bioorganic & medicinal chemistry letters 20100801
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Toxicity of the antimalarial artemisinin and its dervatives.
Critical reviews in toxicology 20100501
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Efficacy of novel oral formulations of α/β arteether against multidrug-resistant malaria in mice.
Chemotherapy 20100101
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Indolizidine, antiinfective and antiparasitic compounds from Prosopis glandulosa var. glandulosa.
Journal of natural products 20090101
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alpha/beta-Arteether-induced mania in a predisposed adolescent.
General hospital psychiatry 20090101
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New functionalized 1,2,4-trioxepanes: synthesis and antimalarial activity against multi-drug resistant P. yoelii in mice.
Bioorganic & medicinal chemistry letters 20081001
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Developmental toxicity of artesunate in the rat: comparison to other artemisinins, comparison of embryotoxicity and kinetics by oral and intravenous routes, and relationship to maternal reticulocyte count.
Birth defects research. Part B, Developmental and reproductive toxicology 20080801
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A model based assessment of the CYP2B6 and CYP2C19 inductive properties by artemisinin antimalarials: implications for combination regimens.
Journal of pharmacokinetics and pharmacodynamics 20080401
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Distribution of C14-labelled arteether in kidneys and livers of experimental mice after intramuscular injection.
The Southeast Asian journal of tropical medicine and public health 20080301
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Orally active 1,2,4-trioxepanes: synthesis and antimalarial activity of a series of 7-arylvinyl-1,2,4-trioxepanes against multidrug-resistant Plasmodium yoelii in Swiss mice.
Bioorganic & medicinal chemistry 20080215
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Orally active esters of dihydroartemisinin: Synthesis and antimalarial activity against multidrug-resistant Plasmodium yoelii in mice.
Bioorganic & medicinal chemistry letters 20080215
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Orally active antimalarials: synthesis and bioevaluation of a new series of steroid-based 1,2,4-trioxanes against multi-drug resistant malaria in mice.
Bioorganic & medicinal chemistry letters 20070801
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Efficacy of combined treatment with alpha/beta-arteether and sulfadoxine-pyrimethamine, for cases of Plasmodium falciparum malaria in Jharkhand, India.
Annals of tropical medicine and parasitology 20070401
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New adamantane-based spiro 1,2,4-trioxanes orally effective against rodent and simian malaria.
Journal of medicinal chemistry 20070208
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Quality control of active ingredients in artemisinin-derivative antimalarials within Kenya and DR Congo.
Tropical medicine & international health : TM & IH 20070101
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New orally active derivatives of artemisinin with high efficacy against multidrug-resistant malaria in mice.
Journal of medicinal chemistry 20061130
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Reactions of artemisinin and arteether with acid: implications for stability and mode of antimalarial action.
Journal of medicinal chemistry 20061005
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Plasmodium vinckei: selection of a strain exhibiting stable resistance to arteether.
Experimental parasitology 20061001
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Simultaneous quantification of alpha-/beta-diastereomers of arteether, sulphadoxine and pyrimethamine: a promising anti-relapse antimalarial therapeutic combination, by liquid chromatography tandem mass spectrometry.
Journal of chromatography. B, Analytical technologies in the biomedical and life sciences 20060914
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Efficacy and safety of beta-arteether and alpha/beta-arteether for treatment of acute Plasmodium falciparum malaria.
The American journal of tropical medicine and hygiene 20060701
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Malaria: severe, life threatening.
Clinical evidence 20060601
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Orally active 1,2,4-trioxanes: synthesis and antimalarial assessment of a new series of 9-functionalized 3-(1-arylvinyl)-1,2,5-trioxaspiro[5.5]undecanes against multi-drug-resistant plasmodium yoelii nigeriensis in mice.
Journal of medicinal chemistry 20060504
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Antiangiogenic activity of deoxoartemisinin derivatives on chorioallantoic membrane.
Bioorganic & medicinal chemistry letters 20060301
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Effects of artemisinin, artemether, and arteether on the pharmacokinetics of phenytoin.
Methods and findings in experimental and clinical pharmacology 20060301
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Effects of artemisinin, artemether, arteether on the pharmacokinetics of carbamazepine.
Pharmacology 20060101
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Unambiguous synthesis and prophylactic antimalarial activities of imidazolidinedione derivatives.
Journal of medicinal chemistry 20051006
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Pharmacokinetics of the diastereomers of arteether, a potent antimalarial drug, in rats.
Biopharmaceutics & drug disposition 20050901
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Blood schizontocidal activity of azithromycin and its combination with alpha/beta arteether against multi-drug resistant Plasmodium yoelii nigeriensis, a novel MDR parasite model for antimalarial screening.
Parasitology 20050901
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Antifungal activity of artemisinin derivatives.
Journal of natural products 20050801
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Convenient access both to highly antimalaria-active 10-arylaminoartemisinins, and to 10-alkyl ethers including artemether, arteether, and artelinate.
Chembiochem : a European journal of chemical biology 20050401
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Studies on drug metabolizing enzymes during arteether treatment of Plasmodium yoelii nigeriensis infected mice cerebral microvessels.
The Journal of communicable diseases 20050301
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Clinical pharmacokinetics of the diastereomers of arteether in healthy volunteers.
Clinical pharmacokinetics 20050101
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Pharmacokinetic investigation on the therapeutic potential of artemotil (beta-arteether) in Thai patients with severe Plasmodium falciparum malaria.
The American journal of tropical medicine and hygiene 20041201
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Intramuscular arteether for treating severe malaria.
The Cochrane database of systematic reviews 20041018
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[Combined antimalarial therapy using artemisinin].
Parassitologia 20040601
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Efficacy of arteether in chloroquine resistant falciparum malaria in eastern India.
The Indian journal of medical research 20040101
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Growth inhibition activity of thioacetal artemisinin derivatives against human umbilical vein endothelial cells.
Bioorganic & medicinal chemistry letters 20031103
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An HPLC-MS method for simultaneous estimation of alpha,beta-arteether and its metabolite dihydroartemisinin, in rat plasma for application to pharmacokinetic study.
Biomedical chromatography : BMC 20031001
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Densitometric thin-layer chromatographic determination of artemisinin and its lipophilic derivatives, artemether and arteether.
Journal of chromatographic science 20030801
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Neuropathological assessment of artemether-treated severe malaria.
Lancet (London, England) 20030726
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A sensitive and selective liquid chromatographic/electrospray ionization tandem mass spectrometric assay for the simultaneous quantification of alpha-,beta-arteether and its metabolite dihydroartemisinin in plasma, useful for pharmacokinetic studies.
Journal of mass spectrometry : JMS 20030701
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A short synthesis and biological evaluation of potent and nontoxic antimalarial bridged bicyclic beta-sulfonyl-endoperoxides.
Journal of medicinal chemistry 20030605
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[Three newly registered drugs in the Netherlands for the treatment and chemoprophylaxis of malaria: atovaquone-proguanil, artemether-lumefantrine and artemotil].
Nederlands tijdschrift voor geneeskunde 20030215
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Liquid chromatographic-mass spectrometric method for the determination of alpha-,beta-arteether in rat serum.
Journal of chromatography. B, Analytical technologies in the biomedical and life sciences 20030115
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Synthesis, stability, and antimalarial activity of new hydrolytically stable and water-soluble (+)-deoxoartelinic acid.
Journal of medicinal chemistry 20021024
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mRNA expression profiles for the response of human tumor cell lines to the antimalarial drugs artesunate, arteether, and artemether.
Biochemical pharmacology 20020815
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Mixed steroidal 1,2,4,5-tetraoxanes: antimalarial and antimycobacterial activity.
Journal of medicinal chemistry 20020801
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Efficacy of alpha, beta - Arteether in children with cerebral malaria in forested tribal belt.
Indian pediatrics 20020601
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Dose-finding and efficacy study for i.m. artemotil (beta-arteether) and comparison with i.m. artemether in acute uncomplicated P. falciparum malaria.
British journal of clinical pharmacology 20020501
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Neurotoxicity and efficacy of arteether related to its exposure times and exposure levels in rodents.
The American journal of tropical medicine and hygiene 20020501
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Artemotil Artecef.
Current opinion in investigational drugs (London, England : 2000) 20020401
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Post-marketing surveillance of arteether in malaria.
The Journal of the Association of Physicians of India 20020401
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Multicentric clinical trials for safety and efficacy evaluation of alpha;beta arteether in complicated P. falciparum malaria.
The Journal of the Association of Physicians of India 20011201
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Antimalarial simplified 3-aryltrioxanes: synthesis and preclinical efficacy/toxicity testing in rodents.
Journal of medicinal chemistry 20010913
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Arteether in therapy of malaria.
The Journal of the Association of Physicians of India 20010701
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A multicentric study with arteether in patients of uncomplicated falciparum malaria.
The Journal of the Association of Physicians of India 20010701
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Effect of beta-arteether treatment on erythrocytic methemoglobin reductase system in Plasmodium yoelii nigeriensis infected mice.
Drug and chemical toxicology 20010501
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Effects of arteether on an auditory radial-arm maze task in rats.
Physiology & behavior 20010501
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Clinical trial of beta-arteether versus quinine for the treatment of cerebral malaria in children in Yaounde, Cameroon.
The American journal of tropical medicine and hygiene 20010101
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Comparison of beta-artemether and beta-arteether against malaria parasites in vitro and in vivo.
The American journal of tropical medicine and hygiene 19930301