90-34-6 | N-(5-aminopentan-2-yl)-6-methoxyquinolin-8-amine

Packsize	Purity	Availability	Price	Discounted Price
100mg	95%	in stock	$89.00	$62.00
250mg	95%	in stock	$128.00	$89.00
1g	95%	in stock	$129.00	$90.00
5g	95%	in stock	$471.00	$330.00
25g	95%	in stock	$1,847.00	$1,293.00

Description

• Catalog Number: AI60273
• Chemical Name: N-(5-aminopentan-2-yl)-6-methoxyquinolin-8-amine
• CAS Number: 90-34-6
• Molecular Formula: C15H21N3O
• Molecular Weight: 259.3467
• MDL Number: MFCD00598906
• SMILES: NCCCC(Nc1cc(OC)cc2c1nccc2)C
• NSC Number: 27296

Computed Properties

• Complexity: 262
• Covalently-Bonded Unit Count: 1
• Heavy Atom Count: 19
• Hydrogen Bond Acceptor Count: 4
• Hydrogen Bond Donor Count: 2
• Rotatable Bond Count: 6
• Undefined Atom Stereocenter Count: 1
• XLogP3: 2.2

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• Alteration of platelet counts and lipid profiles after treatment of acute Plasmodium vivax.

  Acta tropica 20080401

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  Medecine et maladies infectieuses 20080401

• Novel triazine JPC-2067-B inhibits Toxoplasma gondii in vitro and in vivo.

  PLoS neglected tropical diseases 20080301

• Formulation, antimalarial activity and biodistribution of oral lipid nanoemulsion of primaquine.

  International journal of pharmaceutics 20080122

• Development and validation of UPLC method for determination of primaquine phosphate and its impurities.

  Journal of pharmaceutical and biomedical analysis 20080122

• Anti-Pneumocystis carinii and antiplasmodial activities of primaquine-derived imidazolidin-4-ones.

  Bioorganic & medicinal chemistry letters 20080115

• HepaRG cells as an in vitro model for evaluation of cytochrome P450 induction in humans.

  Drug metabolism and disposition: the biological fate of chemicals 20080101

• Atypical Plasmodium vivax malaria in a traveler: bilateral hydronephrosis, severe thrombocytopenia, and hypotension.

  Journal of travel medicine 20080101

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  Revista da Sociedade Brasileira de Medicina Tropical 20080101

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  Meditsinskaia parazitologiia i parazitarnye bolezni 20080101

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  Malaria journal 20080101

• Development of a capillary electrophoresis method for the enantioselective estimation of primaquine in pharmaceutical formulations.

  Journal of AOAC International 20080101

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  The Southeast Asian journal of tropical medicine and public health 20080101

• A randomised trial of an eight-week, once weekly primaquine regimen to prevent relapse of plasmodium vivax in Northwest Frontier Province, Pakistan.

  PloS one 20080101

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  Molecular pharmaceutics 20080101

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  Meditsinskaia parazitologiia i parazitarnye bolezni 20080101

• Targeting the plasmepsin 4 orthologs of Plasmodium sp. with 'double drug' inhibitors.

  Protein and peptide letters 20080101

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  Revista da Sociedade Brasileira de Medicina Tropical 20080101

• The role of anti-malarial drugs in eliminating malaria.

  Malaria journal 20080101

• Synthesis and evaluation of naphthyridine compounds as antimalarial agents.

  Bioorganic & medicinal chemistry letters 20071115

• Neglect of Plasmodium vivax malaria.

  Trends in parasitology 20071101

• Clinical inquiries. When should travelers begin malaria prophylaxis?

  The Journal of family practice 20071101

• Apparent relapse of imported Plasmodium ovale malaria in a pregnant woman.

  The American journal of tropical medicine and hygiene 20071101

• Congenital malaria in the United States: a review of cases from 1966 to 2005.

  Archives of pediatrics & adolescent medicine 20071101

• Recent patent reviews on small molecule-based antimalarial drugs.

  Recent patents on anti-infective drug discovery 20071101

• Exploring biosynthetic diversity with trichodiene synthase.

  Archives of biochemistry and biophysics 20071015

• Pulmonary edema due to Plasmodium vivax malaria in an American missionary.

  Infection 20071001

• Primaquine-induced differential gene expression analysis in mice liver using DNA microarrays.

  Toxicology 20070924

• Cytoplasmic remodeling of erythrocyte raft lipids during infection by the human malaria parasite Plasmodium falciparum.

  Blood 20070915

• Management of vivax malaria with primaquine.

  The Journal of infection 20070901

• Clinical signs and response to primaquine in falcons with Haemoproteus tinnunculi infection.

  The Veterinary record 20070811

• Role of calcium messenger systems in ACTH-induced cortisol production in bovine adrenal fasciculo-reticularis cells.

  Endocrine journal 20070801

• Methaemoglobinaemia causing progressive dyspnoea and cyanosis during treatment of Pneumocystis jirovecii pneumonia.

  International journal of STD & AIDS 20070801

• In Vitro and In Vivo pharmacokinetic studies of bulaquine (analogue of primaquine), a novel antirelapse antimalarial, in rat, rabbit and monkey--highlighting species similarities and differences.

  Biopharmaceutics & drug disposition 20070701

• Persistent binding of ligands to the aryl hydrocarbon receptor.

  Toxicological sciences : an official journal of the Society of Toxicology 20070701

• Chloroquine-resistant Plasmodium vivax, Brazilian Amazon.

  Emerging infectious diseases 20070701

• Vivax malaria: preliminary observations following a shorter course of treatment with artesunate plus primaquine.

  Transactions of the Royal Society of Tropical Medicine and Hygiene 20070601

• Clinical efficacy of chloroquine versus artemether-lumefantrine for Plasmodium vivax treatment in Thailand.

  The Korean journal of parasitology 20070601

• Unanticipated stereoselectivity in the reaction of primaquine alpha-aminoamides with substituted benzaldehydes: a computational and experimental study.

  The Journal of organic chemistry 20070525

• Controversies and misconceptions in malaria chemoprophylaxis for travelers.

  JAMA 20070523

• Can the host immune system promote multiple invasions of erythrocytes in vivo? Differential effects of medication and host sex in a wild malaria-like model.

  Parasitology 20070501

• Relapses of Plasmodium vivax infection usually result from activation of heterologous hypnozoites.

  The Journal of infectious diseases 20070401

• A background and critical analysis of the treatment of pneumocystis carinii pneumonia (PCP) in HIV/AIDS.

  Australian nursing journal (July 1993) 20070401

• Management of vivax malaria with low sensitivity to primaquine.

  The Journal of infection 20070301

• A case of symptomatic splenic infarction in vivax malaria.

  The Korean journal of parasitology 20070301

• Nature of the main contaminant in the drug primaquine diphosphate: SFC and SFC-MS methods of analysis.

  Journal of pharmaceutical and biomedical analysis 20070219

• When the book is wrong.

  Lancet (London, England) 20070203

• A rare glimpse at the efficacy of primaquine.

  The American journal of tropical medicine and hygiene 20070201

• Regional differences in the response of Plasmodium vivax malaria to primaquine as anti-relapse therapy.

  The American journal of tropical medicine and hygiene 20070201

• Primaquine for preventing relapses in people with Plasmodium vivax malaria.

  The Cochrane database of systematic reviews 20070124

• Synthesis, antimalarial, antileishmanial, antimicrobial, cytotoxicity, and methemoglobin (MetHB) formation activities of new 8-quinolinamines.

  Bioorganic & medicinal chemistry 20070115

• Self-gelling primaquine-gum arabic conjugate: an injectable controlled delivery system for primaquine.

  Biomacromolecules 20070101

• Operational feasibility of rapid diagnostic kits & blister packs use for malaria control in high transmission areas of Orissa & Chhattisgarh.

  The Indian journal of medical research 20070101

• Primaquine clears submicroscopic Plasmodium falciparum gametocytes that persist after treatment with sulphadoxine-pyrimethamine and artesunate.

  PloS one 20070101

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  Revista da Sociedade Brasileira de Medicina Tropical 20070101

• Relapsing vivax malaria after 6 months of daily atovaquone/proguanil in Afghanistan: the case for expanded use of primaquine as a causal prophylactic.

  Journal of travel medicine 20070101

• Photophysical properties and photobiological behavior of amodiaquine, primaquine and chloroquine.

  Photochemistry and photobiology 20070101

• A randomized open-label trial of artesunate- sulfadoxine-pyrimethamine with or without primaquine for elimination of sub-microscopic P. falciparum parasitaemia and gametocyte carriage in eastern Sudan.

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  Bioinformation 20070101

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  Emerging infectious diseases 20061101

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  Haematologica 20061001

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  The American journal of tropical medicine and hygiene 20061001

• Primaquine: report from CDC expert meeting on malaria chemoprophylaxis I.

  The American journal of tropical medicine and hygiene 20060901

• Cost considerations of malaria chemoprophylaxis including use of primaquine for primary or terminal chemoprophylaxis.

  The American journal of tropical medicine and hygiene 20060901

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  Biomedica : revista del Instituto Nacional de Salud 20060901

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  Tanzania health research bulletin 20060901

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  The American journal of tropical medicine and hygiene 20060701

• Chloroquine and primaquine: combining old drugs as a new weapon against falciparum malaria?

  Trends in parasitology 20060601

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  Annals of tropical paediatrics 20060601

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  British journal of clinical pharmacology 20060601

• Lack of sex effect on the pharmacokinetics of primaquine.

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  Malaria journal 20060101

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  The American journal of medicine 20051201

• Failure of primaquine therapy for the treatment of Plasmodium ovale malaria.

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  Biochemical pharmacology 20051015

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  International journal of pharmaceutics 20051013

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  Journal of Korean medical science 20051001

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  Journal of pharmaceutical and biomedical analysis 20050901

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  Experimental parasitology 20050901

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  The Journal of pharmacology and experimental therapeutics 20050801

• Pseudo-borreliosis in patients with malaria.

  The American journal of tropical medicine and hygiene 20050701

• Photoreactivity of biologically active compounds. XVII. Influence of solvent interactions on spectroscopic properties and photostability of primaquine.

  Die Pharmazie 20050601

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  Clinical evidence 20050601

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  International journal of pharmaceutics 20050513

• Effectiveness of antimalarial drugs.

  The New England journal of medicine 20050414

• A novel incubation direct injection LC/MS/MS technique for in vitro drug metabolism screening studies involving the CYP 2D6 and the CYP 3A4 isozymes.

  Journal of pharmaceutical and biomedical analysis 20050401

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  Military medicine 20050401

• Differential toxicity of reactive metabolites of clindamycin and sulfonamides in HIV-infected cells: influence of HIV infection on clindamycin toxicity in vitro.

  Journal of clinical pharmacology 20050301

• Imidazolidin-4-one derivatives of primaquine as novel transmission-blocking antimalarials.

  Journal of medicinal chemistry 20050210

• Piperaquine: a resurgent antimalarial drug.

  Drugs 20050101

• Raising antibodies in chickens against primaquine, pyrimethamine, dapsone, tetracycline, and doxycycline.

  Immunological investigations 20050101

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  Journal of human genetics 20050101

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  Drug and chemical toxicology 20050101

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  Irish veterinary journal 20050101

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  Clinical infectious diseases : an official publication of the Infectious Diseases Society of America 20041015

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  Annals of the New York Academy of Sciences 20041001

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  The EMBO journal 20040707

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  Journal of microencapsulation 20040601

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  Clinical evidence 20040601

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  The Journal of pharmacology and experimental therapeutics 20040401

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  Lancet (London, England) 20040327

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  Bioorganic & medicinal chemistry 20040301

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  Transactions of the Royal Society of Tropical Medicine and Hygiene 20040301

• Nature of the main contaminant in the anti malaria drug primaquine diphosphate: a qualitative isomer analysis.

  Journal of chromatography. B, Analytical technologies in the biomedical and life sciences 20040205

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  Molecular pharmacology 20040201

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  Drug and chemical toxicology 20040201

• CV8, a new combination of dihydroartemisinin, piperaquine, trimethoprim and primaquine, compared with atovaquone-proguanil against falciparum malaria in Vietnam.

  Tropical medicine & international health : TM & IH 20040201

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  The American journal of tropical medicine and hygiene 20031101

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• Two worlds of malaria.

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  Journal of chromatography. B, Analytical technologies in the biomedical and life sciences 20030815

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  International journal of hygiene and environmental health 20030801

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  Indian journal of pediatrics 20030601

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  The Brazilian journal of infectious diseases : an official publication of the Brazilian Society of Infectious Diseases 20030601

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  The American journal of tropical medicine and hygiene 20030501

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  Journal of immunology (Baltimore, Md. : 1950) 20030401

• Toxicity related to chloroquine treatment of resistant vivax malaria.

  The Annals of pharmacotherapy 20030401

• Blood schizontocidal activity of WR 238605 (Tafenoquine) against Plasmodium cynomolgi and Plasmodium fragile infections in rhesus monkeys.

  Acta tropica 20030401

• The chemotherapy of rodent malaria. LXI. Drug combinations to impede the selection of drug resistance, part 4: the potential role of 8-aminoquinolines.

  Annals of tropical medicine and parasitology 20030401

• Conductometric and indirect AAS determination of antimalarials.

  Journal of pharmaceutical and biomedical analysis 20030326

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  Parasitology international 20030301

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  Trends in parasitology 20030301

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  American journal of physiology. Cell physiology 20030201

• Time-dependent transcriptional induction of CYP1A1, CYP1A2 and CYP1B1 mRNAs by H+/K+ -ATPase inhibitors and other xenobiotics.

  Xenobiotica; the fate of foreign compounds in biological systems 20030201

• Case report: An unusual late relapse of Plasmodium vivax malaria.

  The American journal of tropical medicine and hygiene 20030201

• [Antiprotozoal drugs].

  Nihon rinsho. Japanese journal of clinical medicine 20030201

• [Short course schemes for vivax malaria treatment].

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  Revista da Sociedade Brasileira de Medicina Tropical 20030101

• Efficacy of a 14-day primaquine regimen in preventing relapses in patients with Plasmodium vivax malaria in Mumbai, India.

  Transactions of the Royal Society of Tropical Medicine and Hygiene 20030101

• Effectiveness of primaquine terminal prophylaxis against late primary attacks of Plasmodium vivax malaria: a case-control study among troops of the Republic of Korea army.

  Transactions of the Royal Society of Tropical Medicine and Hygiene 20030101

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  Bioorganic & medicinal chemistry letters 20021216

• Discovery of novel targets of quinoline drugs in the human purine binding proteome.

  Molecular pharmacology 20021201

• Primaquine-induced hemolytic anemia: formation of free radicals in rat erythrocytes exposed to 6-methoxy-8-hydroxylaminoquinoline.

  The Journal of pharmacology and experimental therapeutics 20021201

• Plasmodium ovale malaria acquired in central Spain.

  Emerging infectious diseases 20021201

• The clinical and epidemiological features of childhood malaria in a moderately endemic area of Sri Lanka.

  The Southeast Asian journal of tropical medicine and public health 20021201

• Cytochrome P450 1A1/2 induction by antiparasitic drugs: dose-dependent increase in ethoxyresorufin O-deethylase activity and mRNA caused by quinine, primaquine and albendazole in HepG2 cells.

  European journal of clinical pharmacology 20021101

• Pancytopenia resulting from hemophagocytosis in malaria.

  The Pediatric infectious disease journal 20021101

• Primaquine-induced hemolytic anemia: effect of 6-methoxy-8-hydroxylaminoquinoline on rat erythrocyte sulfhydryl status, membrane lipids, cytoskeletal proteins, and morphology.

  The Journal of pharmacology and experimental therapeutics 20021001

• Radical curative efficacy of five-day regimen of primaquine for treatment of Plasmodium vivax malaria in India.

  The Journal of parasitology 20021001

• Sensitivity of Plasmodium vivax to chloroquine in Sa Kaeo Province, Thailand.

  Acta tropica 20020801

• Does radical cure of asymptomatic Plasmodium falciparum place adults in endemic areas at increased risk of recurrent symptomatic malaria?

  Tropical medicine & international health : TM & IH 20020701

• Recycling CD1d1 molecules present endogenous antigens processed in an endocytic compartment to NKT cells.

  Journal of immunology (Baltimore, Md. : 1950) 20020601

• Coronary bypass surgery in patient with malaria.

  Asian cardiovascular & thoracic annals 20020601

• Short report: therapeutic efficacy of chloroquine combined with primaquine against Plasmodium falciparum in northeastern Papua, Indonesia.

  The American journal of tropical medicine and hygiene 20020601

• Relapsing vivax malaria.

  The Medical journal of Australia 20020520

• Enantiomeric separation of primaquine, an anti-malarial drug, by cyclodextrin-modified micellar electrokinetic capillary chromatography.

  Analytical sciences : the international journal of the Japan Society for Analytical Chemistry 20020501

• In vitro cultivation of Chinese strains of Babesia spp.

  Parasitology research 20020501

• Effect of antimalarial drugs on plasmodia cell-free protein synthesis.

  Memorias do Instituto Oswaldo Cruz 20020401

• Relapse pattern of Plasmodium vivax in Mumbai: a study of 283 cases of vivax malaria.

  The Journal of the Association of Physicians of India 20020301

• Methemoglobin reductase activity and in vitro sensitivity towards oxidant induced methemoglobinemia in swiss mice and beagle dogs erythrocytes.

  Molecular and cellular biochemistry 20020301

• Prevalence of malaria in Aligarh.

  The Journal of communicable diseases 20020301

• Inhibition of cardiac Na+ current by primaquine.

  British journal of pharmacology 20020201

• Mutagenic activity and mutational specificity of antiprotozoal drugs with and without nitrite treatment.

  Environmental and molecular mutagenesis 20020101

• Control of malaria: a successful experience from Viet Nam.

  Bulletin of the World Health Organization 20020101

• Comparison of tafenoquine (WR238605) and primaquine in the post-exposure (terminal) prophylaxis of vivax malaria in Australian Defence Force personnel.

  Transactions of the Royal Society of Tropical Medicine and Hygiene 20020101

• Randomized, parallel placebo-controlled trial of primaquine for malaria prophylaxis in Papua, Indonesia.

  Clinical infectious diseases : an official publication of the Infectious Diseases Society of America 20011215

• Effect of primaquine standard dose (15 mg/day for 14 days) in the treatment of vivax malaria patients in Thailand.

  The Southeast Asian journal of tropical medicine and public health 20011201

• Current drugs for antimalarial chemoprophylaxis: a review of efficacy and safety.

  Journal of travel medicine 20011201

• A systematic gene expression screen of Caenorhabditis elegans cytochrome P450 genes reveals CYP35 as strongly xenobiotic inducible.

  Archives of biochemistry and biophysics 20011115

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  The American journal of tropical medicine and hygiene 20011101

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  Annals of tropical medicine and parasitology 20011001

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  Clinical and diagnostic laboratory immunology 20010901

• Malaria chemoprophylaxis in the age of drug resistance. II. Drugs that may be available in the future.

  Clinical infectious diseases : an official publication of the Infectious Diseases Society of America 20010801

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  The American journal of tropical medicine and hygiene 20010801

• Malaria chemoprophylaxis in the age of drug resistance. I. Currently recommended drug regimens.

  Clinical infectious diseases : an official publication of the Infectious Diseases Society of America 20010715

• The antileishmanial properties of surface-modified, primaquine-loaded nanocapsules tested against intramacrophagic Leishmania donovani amastigotes in vitro.

  Annals of tropical medicine and parasitology 20010701

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  Archives of internal medicine 20010625

• Treating malaria may be too expensive.

  Australian family physician 20010601

• Primaquine-induced hemolytic anemia: formation and hemotoxicity of the arylhydroxylamine metabolite 6-methoxy-8-hydroxylaminoquinoline.

  The Journal of pharmacology and experimental therapeutics 20010501

• Transcriptional and post-translational regulation of CYP1A1 by primaquine.

  The Journal of pharmacology and experimental therapeutics 20010401

• Oxidative stress participates in the breakdown of neuronal phenotype in experimental diabetic neuropathy.

  Diabetologia 20010401

• Functional integrity of the vesicle transporting machinery is required for complete activation of cFTR expressed in xenopus laevis oocytes.

  Pflugers Archiv : European journal of physiology 20010301

• [Does the brief treatment with antimalarials favorably influence drug resistance and recurrences?].

  Revista panamericana de salud publica = Pan American journal of public health 20010301

• Dissociation and electrooxidation of primaquine diphosphate as an approach to the study of anti-chagas prodrugs mechanism of action.

  Bioelectrochemistry (Amsterdam, Netherlands) 20010101

• Immunological alterations associated with Plasmodium vivax malaria in South Korea.

  Annals of tropical medicine and parasitology 20010101

• Antimalarial chemoprophylaxis in infants and children.

  Paediatric drugs 20010101

• [Primaquine].

  Medecine tropicale : revue du Corps de sante colonial 20010101

• Malaria prophylaxis/radical cure: recent experiences of the Australian Defence Force.

  Medecine tropicale : revue du Corps de sante colonial 20010101

• [Effect of daphnetin on the exo-erythrocytic stage of rodent malaria].

  Zhongguo ji sheng chong xue yu ji sheng chong bing za zhi = Chinese journal of parasitology & parasitic diseases 20010101

• [A study of artemether combined with primaquine in the treatment of falciparum malaria].

  Zhongguo ji sheng chong xue yu ji sheng chong bing za zhi = Chinese journal of parasitology & parasitic diseases 20010101

• Potential inhibitors of HIV integrase.

  Nucleosides & nucleotides 19990101

• Prediction of aryl hydrocarbon receptor-mediated enzyme induction of drugs and chemicals by mRNA quantification.

  Chemical research in toxicology 19981201

• [Hemolysis and primaquine treatment. Preliminary report].

  Revista cubana de medicina tropical 19970101

• Efficacy of 101 antimicrobials and other agents on the development of Cryptosporidium parvum in vitro.

  Annals of tropical medicine and parasitology 19961201

• Dapsone- and primaquine-induced methemoglobinemia in HIV-infected individuals.

  Journal of acquired immune deficiency syndromes and human retrovirology : official publication of the International Retrovirology Association 19960815

• Drug-induced methaemoglobinaemia. Treatment issues.

  Drug safety 19960601

• New drug developments for opportunistic infections in immunosuppressed patients: Pneumocystis carinii.

  Journal of medicinal chemistry 19951124

• [Primaquine and travelers from the Arab world. A report and recommendations].

  Revista cubana de medicina tropical 19950101

• In vitro effects of artemisinin ether, cycloguanil hydrochloride (alone and in combination with sulfadiazine), quinine sulfate, mefloquine, primaquine phosphate, trifluoperazine hydrochloride, and verapamil on Toxoplasma gondii.

  Antimicrobial agents and chemotherapy 19940601

• [Comparative study on hemolytic toxicity of trifluoroacetoprimaquine and primaquine in rabbits].

  Zhongguo ji sheng chong xue yu ji sheng chong bing za zhi = Chinese journal of parasitology & parasitic diseases 19940101

• Inhibitors of human immunodeficiency virus integrase.

  Proceedings of the National Academy of Sciences of the United States of America 19930315

• Acute intravascular haemolysis in Vanuatu following a single dose of primaquine in individuals with glucose-6-phosphate dehydrogenase deficiency.

  The Journal of tropical medicine and hygiene 19921001

• 8-Aminoquinolines from Walter Reed Army Institute for Research for treatment and prophylaxis of Pneumocystis pneumonia in rat models.

  Antimicrobial agents and chemotherapy 19910201

• Isolation and characterization of rat lung Pneumocystis carinii gp120.

  The Journal of protozoology 19910101

• The effect of primaquine on the ultrastructural morphology of Pneumocystis carinii.

  The Journal of protozoology 19910101

• Detection of antidrug IgG antibodies in patients with adverse drug reactions to amodiaquine.

  International archives of allergy and applied immunology 19910101

• Immunogenicity of amodiaquine in the rat.

  International archives of allergy and applied immunology 19900101

• Primaquine induced hemolysis in a Thai soldier.

  The Southeast Asian journal of tropical medicine and public health 19891201

• Activity of clindamycin with primaquine against Pneumocystis carinii in vitro and in vivo.

  Antimicrobial agents and chemotherapy 19880601

• [Hemolytic reaction due to administration of primaquine].

  Zhonghua liu xing bing xue za zhi = Zhonghua liuxingbingxue zazhi 19860401

• Drug- and chemical-induced methaemoglobinaemia. Clinical features and management.

  Medical toxicology 19860101

• Pharmacokinetics of primaquine in man. I. Studies of the absolute bioavailability and effects of dose size.

  British journal of clinical pharmacology 19850601

• Primaquine-chloroquine prophylaxis against malaria in Southeast-Asian refugees entering South Australia.

  The Medical journal of Australia 19840317

• The treatment of malaria in glucose-6-phosphate dehydrogenase deficient patients in Sabah.

  Annals of tropical medicine and parasitology 19811201

• Reaction to primaquine.

  Annals of internal medicine 19800301

• Antimalarial activities of various 4-quinolonemethanols with special attention to WR-142,490 (mefloquine).

  Antimicrobial agents and chemotherapy 19780601

• Hemolysis in dialyzed patients: tap water-induced red blood cell metabolic deficiency.

  Transactions - American Society for Artificial Internal Organs 19720101

• Simultaneous drug reactions in the same patient. Chloroquine-Primaquine sensitivity.

  JAMA 19700427

• Methemoglobinemia provoked by malarial chemoprophylaxis in Vietnam.

  The New England journal of medicine 19681121

• The haemolytic effect of various regimens of primaquine with chloroquine in American Negroes with G6PD deficiency and the lack of an effect of various antimalarial suppressive agents on erythrocyte metabolism.

  Bulletin of the World Health Organization 19670101

• Potentiation of the curative action of primaquine in vivax malaria by quinine and chloroquine.

  The Journal of laboratory and clinical medicine 19550801