-
Ring splitting of azetidin-2-ones via radical anions.
Organic & biomolecular chemistry 20121021
-
An expeditious iodine-catalyzed synthesis of 3-pyrrole-substituted 2-azetidinones.
Molecules (Basel, Switzerland) 20120928
-
Photoelectron spectra of some antibiotic building blocks: 2-azetidinone and thiazolidine-carboxylic acid.
The journal of physical chemistry. A 20120823
-
An expeditious route to eight-membered heterocycles by nickel-catalyzed cycloaddition: low-temperature C(sp)2-C(sp)3 bond cleavage.
Angewandte Chemie (International ed. in English) 20120820
-
Kappa agonist CovX-Bodies.
Bioorganic & medicinal chemistry letters 20120615
-
Regioselective cycloaddition of 3-azetidinones and 3-oxetanones with alkynes through nickel-catalysed carbon-carbon bond activation.
Chemistry (Weinheim an der Bergstrasse, Germany) 20120319
-
Synthesis and bioactivities of 2-azetidinone derivatives as cholesterol absorption inhibitors.
Medicinal chemistry (Shariqah (United Arab Emirates)) 20111101
-
Antibacterial agents and cystic fibrosis: synthesis and antimicrobial evaluation of a series of N-thiomethylazetidinones.
ChemMedChem 20111004
-
Antiplasmodial and cytotoxicity evaluation of 3-functionalized 2-azetidinone derivatives.
Bioorganic & medicinal chemistry letters 20110801
-
Synthesis of spirocyclic β-keto-lactams: copper catalyzed process.
Chemical communications (Cambridge, England) 20110507
-
Synthesis, evaluation and structural studies of antiproliferative tubulin-targeting azetidin-2-ones.
Bioorganic & medicinal chemistry 20110401
-
Monocyclic β-lactams: new structures for new biological activities.
Current medicinal chemistry 20110101
-
2-Azetidinone--a new profile of various pharmacological activities.
European journal of medicinal chemistry 20101201
-
Synthesis of chlorinated bicyclic C-fused tetrahydrofuro[3,2-c]azetidin-2-ones.
The Journal of organic chemistry 20101105
-
Ferrier-Petasis rearrangement of 4-(vinyloxy)azetidin-2-ones: an entry to carbapenams and carbacephams.
The Journal of organic chemistry 20101015
-
T-type calcium channel blockers: spiro-piperidine azetidines and azetidinones-optimization, design and synthesis.
Bioorganic & medicinal chemistry letters 20100801
-
Azetidinone-isothiazolidinones: stereoselective synthesis and antibacterial evaluation of new monocyclic beta-lactams.
Bioorganic & medicinal chemistry 20100501
-
Synthesis, in-vitro antimicrobial and cytotoxic studies of novel azetidinone derivatives.
Archiv der Pharmazie 20100401
-
Suppressed beta-effect of silicon in 3-silylated monocyclic beta-lactams: the role of antiaromaticity.
Organic letters 20091217
-
Design, synthesis and bioactivity of catechin/epicatechin and 2-azetidinone derived chimeric molecules.
Bioorganic & medicinal chemistry letters 20091215
-
2-Azetidinone derivatives: design, synthesis, in vitro anti-microbial, cytotoxic activities and DNA cleavage study.
European journal of medicinal chemistry 20091201
-
Azetidinones as zinc-binding groups to design selective HDAC8 inhibitors.
ChemMedChem 20091201
-
Lewis acid-assisted ene cyclization of 2-azetidinone-tethered enals: synthesis of enantiopure carbacepham derivatives.
Chemistry, an Asian journal 20091005
-
Staudinger ketene-imine cycloaddition, RCM approach to macrocrocyclic bisazetidinones.
The Journal of organic chemistry 20090605
-
Large ring 1,3-bridged 2-azetidinones: experimental and theoretical studies.
European journal of medicinal chemistry 20090501
-
2-Azetidinone derivatives: design, synthesis and evaluation of cholesterol absorption inhibitors.
European journal of medicinal chemistry 20090401
-
Spiro-piperidine azetidinones as potent TRPV1 antagonists.
Bioorganic & medicinal chemistry letters 20090201
-
Deeper insight into the mechanism of the reaction of photogenerated metallaketenes and imines.
Journal of the American Chemical Society 20081022
-
Novel syntheses of azetidines and azetidinones.
Chemical reviews 20080901
-
3-Alkenyl-2-azetidinones as fatty acid amide hydrolase inhibitors.
Bioorganic & medicinal chemistry letters 20080715
-
Total synthesis of (-)-kainic acid via intramolecular Michael addition: a second-generation route.
Organic letters 20080501
-
Discovery of azetidinone acids as conformationally-constrained dual PPARalpha/gamma agonists.
Bioorganic & medicinal chemistry letters 20080315
-
New regiocontrolled synthesis of functionalized pyrroles from 2-azetidinone-tethered allenols.
Chemistry (Weinheim an der Bergstrasse, Germany) 20080101
-
Synthesis and biological activity of N-substituted-3-chloro-2-azetidinones.
Molecules (Basel, Switzerland) 20071112
-
Synthesis of novel N-(4-ethoxyphenyl) azetidin-2-ones and their oxidative N-deprotection by ceric ammonium nitrate.
Molecules (Basel, Switzerland) 20071025
-
Synthesis of 3-[4'-(p-chlorophenyl)-thiazol-2'-yl]-2-[(substituted azetidinone/thiazolidinone)-aminomethyl]-6-bromoquinazolin-4-ones as anti-inflammatory agent.
Bioorganic & medicinal chemistry 20070415
-
Azetidinones as vasopressin V1a antagonists.
Bioorganic & medicinal chemistry 20070301
-
Indium-mediated selective introduction of a 1,3-butadien-2-yl group at the C4-position in 2-azetidinones and application of 1,3-diene-tethered 2-azetidinones in the Diels-Alder reaction.
Chemistry (Weinheim an der Bergstrasse, Germany) 20070101
-
A theoretical proposal for the synthesis of carbapenems from 4-(2-propynyl)azetidinones promoted by [W(CO)5] as an alternative to the Ag+-assisted process.
Chemistry (Weinheim an der Bergstrasse, Germany) 20061016
-
Structures of (S)-(-)-4-oxo-2-azetidinecarboxylic acid and 3-azetidinecarboxylic acid from powder synchrotron diffraction data.
Acta crystallographica. Section B, Structural science 20060801
-
Synthesis of strained tricyclic beta-lactams by intramolecular [2+2] cycloaddition reactions of 2-azetidinone-tethered enallenols: control of regioselectivity by selective alkene substitution.
Chemistry (Weinheim an der Bergstrasse, Germany) 20060201
-
The polymer-supported and combinatorial synthesis of beta-lactam compounds: an update.
Mini reviews in medicinal chemistry 20060101
-
Rabbit small intestine does not contain an annexin II/caveolin 1 complex as a target for 2-azetidinone cholesterol absorption inhibitors.
Biochimica et biophysica acta 20060101
-
Synthesis of 2-azetidinones from 2-diazo-1, 2-diarylethanones and N-(2-thienylidene)imines as possible antimicrobial agents.
Farmaco (Societa chimica italiana : 1989) 20050901
-
The indium-mediated selective introduction of allenyl and propargyl groups at the C4-position of 2-azetidinones and the AuCl3-catalyzed cyclization of 4-allenyl-2-azetidinones.
Angewandte Chemie (International ed. in English) 20050311
-
3,4-disubstituted azetidinones as selective inhibitors of the cysteine protease cathepsin K. Exploring P3 elements for potency and selectivity.
Bioorganic & medicinal chemistry letters 20050301
-
Kinetics and mechanism of hydrolysis of N-acyloxymethyl derivatives of azetidin-2-one.
The Journal of organic chemistry 20040514
-
Examination of the 1,4-disubstituted azetidinone ring system as a template for combretastatin A-4 conformationally restricted analogue design.
Bioorganic & medicinal chemistry letters 20040503
-
Solid-phase synthesis and SAR of 4-carboxy-2-azetidinone mechanism-based tryptase inhibitors.
Bioorganic & medicinal chemistry letters 20040503
-
Synthesis of optically pure highly functionalized gamma-lactams via 2-azetidinone-tethered iminophosphoranes.
The Journal of organic chemistry 20040206
-
Synthesis of antitumor 6-alkylidenepenicillanate sulfones and related 3-alkylidene-2-azetidinones.
Bioorganic & medicinal chemistry letters 20040105
-
Synthesis and evaluation of N1/C4-substituted beta-lactams as PPE and HLE inhibitors.
Bioorganic & medicinal chemistry 20040102
-
Synthesis of cryptophycins via an N-acyl-beta-lactam macrolactonization.
The Journal of organic chemistry 20031212
-
Synthesis of a biotin-tagged photoaffinity probe of 2-azetidinone cholesterol absorption inhibitors.
Bioorganic & medicinal chemistry 20030417
-
Catalysts with mixed ligands on immobilized supports. Electronic and steric advantages.
Organic letters 20030220
-
Synthesis and SAR of 4-carboxy-2-azetidinone mechanism-based tryptase inhibitors.
Bioorganic & medicinal chemistry letters 20021104
-
A stereoselective synthesis of BMS-262084, an azetidinone-based tryptase inhibitor.
The Journal of organic chemistry 20020531
-
General approach for the stereocontrolled construction of the beta-lactam ring in amino acid-derived 4-alkyl-4-carboxy-2-azetidinones.
The Journal of organic chemistry 20020531
-
Water-assisted alkaline hydrolysis of monobactams: a theoretical study.
Chemistry (Weinheim an der Bergstrasse, Germany) 20020215
-
Synthesis of iodinated biochemical tools related to the 2-azetidinone class of cholesterol absorption inhibitors.
Bioorganic & medicinal chemistry letters 20020211
-
Synthesis of fluorescent biochemical tools related to the 2-azetidinone class of cholesterol absorption inhibitors.
Bioorganic & medicinal chemistry letters 20020211
-
Design, synthesis and pharmacological evaluation of 3-benzylazetidine-2-one-based human chymase inhibitors.
Bioorganic & medicinal chemistry 20011101
-
Metal-promoted allylation, propargylation, or allenylation of azetidine-2,3-diones in aqueous and anhydrous media. Application to the asymmetric synthesis of densely functionalized 3-substituted 3-hydroxy-beta-lactams.
The Journal of organic chemistry 20010727
-
Crystal structure of 3,3-dichloro-N-p-methoxyphenyl-4-(2-phenylstryl)-2-azetidinone.
Analytical sciences : the international journal of the Japan Society for Analytical Chemistry 20010701
-
Entry to new conformationally constrained amino acids. First synthesis of 3-unsubstituted 4-alkyl-4-carboxy-2-azetidinone derivatives via an intramolecular N(alpha)-C(alpha)-cyclization strategy.
The Journal of organic chemistry 20010518
-
beta-lactam derivatives as enzyme inhibitors: carboxy peptidyl derivatives of (S)-4-oxoazetidine-2-carboxylate as peptidomimetics.
Archiv der Pharmazie 20010501
-
Design, synthesis and stability of N-acyloxymethyl- and N-aminocarbonyloxymethyl-2-azetidinones as human leukocyte elastase inhibitors.
Bioorganic & medicinal chemistry letters 20010423
-
Synthesis of trans-4-aryl-3-(omega-chloroalkyl) -2-azetidinones.
Mededelingen (Rijksuniversiteit te Gent. Fakulteit van de Landbouwkundige en Toegepaste Biologische Wetenschappen) 20010101
